-
1دورية أكاديمية
المؤلفون: Terence G Hall, Yi Yu, Sudharshan Eathiraj, Yunxia Wang, Ronald E Savage, Jean-Marc Lapierre, Brian Schwartz, Giovanni Abbadessa
المصدر: PLoS ONE, Vol 11, Iss 9, p e0162594 (2016)
وصف الملف: electronic resource
-
2
المؤلفون: Jean-Marc Lapierre, Cathy O. Bull, Ronald E. Savage, Sudharshan Eathiraj, David Vensel, Sapna Makhija, Eugene Kelleher, Neil Westlund, Jeff Szwaya, Yanbin Liu, Steffi Koerner, Magdi Moussa, Susan Cornell-Kennon, Akihisa Matsuda, Darin Kizer, Nivedita Namdev, Hui Wu, Shin Iimura, Brian Schwartz, Erika Volckova
المصدر: Journal of Medicinal Chemistry. 59:6455-6469
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Allosteric regulation, Administration, Oral, Aminopyridines, AKT1, Antineoplastic Agents, AKT2, Mice, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Allosteric Regulation, Drug Discovery, Animals, Humans, Moiety, Protein Kinase Inhibitors, Protein kinase B, Cell Proliferation, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, Kinase, Imidazoles, Neoplasms, Experimental, Endometrial Neoplasms, 030104 developmental biology, Enzyme, chemistry, 030220 oncology & carcinogenesis, embryonic structures, Molecular Medicine, Phosphorylation, Female, Drug Screening Assays, Antitumor, Carcinoma, Endometrioid, Proto-Oncogene Proteins c-akt
-
3
المؤلفون: Tom O'Shea, Kevin Mills, Jean-Marc Lapierre, Melinda Day
المصدر: Cancer Research. 79:C14-C14
مصطلحات موضوعية: Genome instability, Cancer Research, biology, DNA repair, Cancer, Cytidine deaminase, Synthetic lethality, medicine.disease_cause, medicine.disease, Oncology, Pancreatic cancer, Activation-induced (cytidine) deaminase, biology.protein, medicine, Cancer research, Carcinogenesis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::eac41465559b00f84c2654fda617674d
https://doi.org/10.1158/1538-7445.panca19-c14 -
4
المؤلفون: Mark A. Ashwell, Jean-Marc Lapierre, Christopher Brassard, Karen Bresciano, Cathy Bull, Susan Cornell-Kennon, Sudharshan Eathiraj, Dennis S. France, Terence Hall, Jason Hill, Eoin Kelleher, Sampada Khanapurkar, Darin Kizer, Steffi Koerner, Jeff Link, Yanbin Liu, Sapna Makhija, Magdi Moussa, Nivedita Namdev, Khanh Nguyen, Robert Nicewonger, Rocio Palma, Jeff Szwaya, Manish Tandon, Uma Uppalapati, David Vensel, Laurie P. Volak, Erika Volckova, Neil Westlund, Hui Wu, Rui-Yang Yang, Thomas C. K. Chan
المصدر: Journal of Medicinal Chemistry. 55:5291-5310
مصطلحات موضوعية: Models, Molecular, Protein Conformation, Pyridines, Administration, Oral, Biological Availability, AKT1, Antineoplastic Agents, Plasma protein binding, Pharmacology, Crystallography, X-Ray, Mice, Structure-Activity Relationship, Adenosine Triphosphate, In vivo, Catalytic Domain, Cell Line, Tumor, Drug Discovery, Animals, Humans, Structure–activity relationship, Phosphorylation, Protein kinase B, Adaptor Proteins, Signal Transducing, Cell Proliferation, Effector, Chemistry, Imidazoles, Ribosomal Protein S6 Kinases, 70-kDa, Small molecule, Biochemistry, Microsomes, Liver, Molecular Medicine, Proto-Oncogene Proteins c-akt, Protein Binding
-
5
المؤلفون: Tara Mirzadegan, Frank Diehl, Bettina Ebi, Sunil Bhakta, Irene Polsky, Deborah McCarley, Mary Mulkins, Gabe S. Weatherhead, Jean-Marc Lapierre, John Dankwardt, David Morgans, Robert Wilhelm, Kurt Jarnagin
المصدر: Journal of Biological Chemistry. 275:25562-25571
مصطلحات موضوعية: CCR1, CCR2, Chemistry, Stereochemistry, C-C chemokine receptor type 7, Chemotaxis, Cell Biology, Biochemistry, Chemokine receptor, Binding site, Receptor, Molecular Biology, Leukocyte chemotaxis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::18289e24da7320fd7e0390483ec5e81b
https://doi.org/10.1074/jbc.m000692200 -
6
المؤلفون: Dieter Seebach, Guy Greiveldinger, Jean-Marc Lapierre, Peter Murer
المصدر: Helvetica Chimica Acta. 80:1648-1681
مصطلحات موضوعية: Stereochemistry, Organic Chemistry, Dispersity, Diastereomer, Branching (polymer chemistry), Biochemistry, Catalysis, Stereocenter, Inorganic Chemistry, chemistry.chemical_compound, Molecular recognition, chemistry, Dendrimer, Drug Discovery, Hydroxymethyl, Physical and Theoretical Chemistry, Enantiomer
-
7
المصدر: Helvetica Chimica Acta. 77:1673-1688
مصطلحات موضوعية: chemistry.chemical_classification, Chemistry, Aryl, Organic Chemistry, Dispersity, Branching (polymer chemistry), Biochemistry, Catalysis, Inorganic Chemistry, chemistry.chemical_compound, Bromide, Dendrimer, Drug Discovery, Polymer chemistry, Molecule, Hydroxymethyl, Physical and Theoretical Chemistry, Alkyl
-
8
المؤلفون: Guy Greiveldinger, Dieter Seebach, Jean-Marc Lapierre, Markus Gautschi
المصدر: Chemische Berichte. 126:2739-2746
مصطلحات موضوعية: Inorganic Chemistry, chemistry.chemical_classification, chemistry.chemical_compound, chemistry, Aldol reaction, Acetal, Molecule, Aldol condensation, Crystal structure, Aldehyde, Medicinal chemistry, Isobutyraldehyde, Lactone
-
9
المؤلفون: Dieter Seebach, Jean-Marc Lapierre, Konstantinos Skobridis
المصدر: Helvetica Chimica Acta. 76:2419-2432
مصطلحات موضوعية: Tris, Aryl, Organic Chemistry, Biochemistry, Medicinal chemistry, Catalysis, Inorganic Chemistry, chemistry.chemical_compound, Acetic acid, chemistry, Bromide, Dendrimer, Drug Discovery, Functional group, Organic chemistry, Hydroxymethyl, Triol, Physical and Theoretical Chemistry
-
10
المؤلفون: Dieter Seebach, Jean-Marc Lapierre, Paul Seiler, Wilfried Jaworek
المصدر: Helvetica Chimica Acta. 76:459-475
مصطلحات موضوعية: chemistry.chemical_classification, Chemistry, Organic Chemistry, Diastereomer, Enantioselective synthesis, Biochemistry, Catalysis, Inorganic Chemistry, Acylation, chemistry.chemical_compound, Aldol reaction, Drug Discovery, Organic chemistry, Triol, Hydroxymethyl, Aldol condensation, Physical and Theoretical Chemistry, Lactone