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المؤلفون: Alfred P. Spada, Robert J. Leadley, Jonathan S. Mason, Dennis J. Colussi, Ewing William R, Mark H. Perrone, Karen D. Brown, Michael R. Becker, Don D. Cha, Daniel M. Green, Ross Bentley, Henry W. Pauls, Christopher T. Dunwiddie, Jean-Pierre Guilloteau, Y.M. Choi-Sledeski, Sebastien Maignan, Mason Helen J, Vincent E. Manetta, Charles Kasiewski, Valeria Chu, Roderick S. Davis, Suzanne Morgan, Daniel L. Cheney, Jeff Bostwick
المصدر: Journal of Medicinal Chemistry. 42:3557-3571
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, medicine.drug_class, Factor Xa Inhibitor, Thiophenes, Crystallography, X-Ray, Amidine, Structure-Activity Relationship, chemistry.chemical_compound, Thrombin, In vivo, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Sulfonamides, Molecular Structure, biology, Chemistry, Anticoagulant, Anticoagulants, Stereoisomerism, Thrombosis, Trypsin, Pyrrolidinones, Rats, Biochemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Rabbits, Factor Xa Inhibitors, medicine.drug
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2
المؤلفون: Charles Kasiewski, Suzanne Morgan, Roderick S. Davis, Robert J. Leadley, Jeff Bostwick, Valeria Chu, Henry W. Pauls, Ewing William R, Karen D. Brown, Cuong Ly, Michael R. Becker, Mason Helen J, Ross Bentley, Y.M. Choi-Sledeski, Dennis J. Colussi, Alfred P. Spada, Aiwen Li
المصدر: Bioorganicmedicinal chemistry letters. 9(18)
مصطلحات موضوعية: Thienopyridine, medicine.drug_mechanism_of_action, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Pharmaceutical Science, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Dogs, In vivo, Drug Discovery, medicine, Structure–activity relationship, Animals, Pyrrolidinones, Molecular Biology, chemistry.chemical_classification, biology, Organic Chemistry, Thrombosis, Sulfonamide, Rats, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Factor Xa Inhibitors