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1
المؤلفون: Jeffrey J Barlow, Lynn Scarlett, Keith Hopkinson Gibson, Susan Ashton, Walter Grundy, Lianne Henthorn, Laura Richards, Brenda Curry, Mark P Healy, Barker Andrew John, J. R. Woodburn, Godfrey Andrew Aydon
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:1911-1914
مصطلحات موضوعية: Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Antineoplastic Agents, Sensitivity and Specificity, Biochemistry, KB Cells, Gefitinib, Growth factor receptor, Epidermal growth factor, Drug Discovery, Tumor Cells, Cultured, medicine, Humans, Growth factor receptor inhibitor, Molecular Biology, biology, Chemistry, Organic Chemistry, Cancer, medicine.disease, ErbB Receptors, Enzyme inhibitor, Carcinoma, Squamous Cell, Quinazolines, biology.protein, Cancer research, Molecular Medicine, Signal transduction, Tyrosine kinase, medicine.drug
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2
المؤلفون: Brian G. Main, Michael H. Block, Jethro L. Longridge, Stuart Nicholson, Alison Leach, Jeffrey J. Barlow, Julian A. Hudson
المصدر: The Journal of Organic Chemistry. 57:5158-5162
مصطلحات موضوعية: chemistry.chemical_classification, Hydrolysis, chemistry.chemical_compound, Acid catalysis, chemistry, Heterocyclic compound, Acid catalyzed, Organic Chemistry, Acetal, Kinetics, Organic chemistry, Racemization
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3
المؤلفون: H. Michael Snow, Jeffrey J. Barlow, Brian G. Main
المصدر: Journal of Medicinal Chemistry. 24:315-322
مصطلحات موضوعية: Agonist, medicine.drug_class, Stereochemistry, Aryl, medicine.medical_treatment, Adrenergic beta-Agonists, Beta adrenoceptor, Partial agonist, Cardiac stimulant, Propanolamines, Stimulant, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, chemistry, Ethanolamines, Heart Rate, Amide, Receptors, Adrenergic, beta, Drug Discovery, medicine, Animals, Molecular Medicine, Selectivity
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4
المصدر: European journal of pharmacology. 151(3)
مصطلحات موضوعية: Agonist, Narcotics, Pyrrolidines, Ratón, medicine.drug_class, Guinea Pigs, Ileum, Pharmacology, In Vitro Techniques, Guinea pig, Mice, medicine, Potency, Animals, Receptor, Chemistry, Naloxone, Receptors, Opioid, kappa, Vas deferens, 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer, Muscle, Smooth, Electric Stimulation, Benzomorphans, medicine.anatomical_structure, Opioid, Morphinans, Receptors, Opioid, medicine.drug, Muscle Contraction