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1دورية أكاديمية
المؤلفون: Eva S. Istvan, Jeremy P. Mallari, Victoria C. Corey, Neekesh V. Dharia, Garland R. Marshall, Elizabeth A. Winzeler, Daniel E. Goldberg
المصدر: Nature Communications, Vol 8, Iss 1, Pp 1-8 (2017)
مصطلحات موضوعية: Science
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2041-1723
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2
المؤلفون: Emmett Pompa, Scott Eagon, Michael Heying, Jeremy P. Mallari, Emma Callant, Nimrat Brar, McClane Howland
المصدر: Bioorganic & Medicinal Chemistry Letters. 52:128394
مصطلحات موضوعية: Models, Molecular, Molecular Structure, biology, Chemistry, Plasmodium falciparum, Organic Chemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Protozoan Proteins, Metalloendopeptidases, Pharmaceutical Science, Computational biology, biology.organism_classification, Biochemistry, Antimalarials, Drug Discovery, Virtual screen, Humans, Molecular Medicine, Identification (biology), Enzyme Inhibitors, Molecular Biology
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3
المؤلفون: Marc O. Anderson, Gulbag Kahlon, Jeremy P. Mallari, Jeff P. Chance, Ngoc Huynh, Nohemy Celis, Emmett Pompa, Paulina Rodriguez, Aaron Keniston, Scott Eagon, Nimrat Brar, Rogelio Lira, Brian Vidal, Nikolay Masvlov, Armann Andaya, Hannah Fejzic, Nicholas Trieu
المصدر: Bioorganic & Medicinal Chemistry Letters. 37:127836
مصطلحات موضوعية: chemistry.chemical_compound, Piperazine, Hydroxamic acid, chemistry, Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Molecular Biology, Biochemistry, Combinatorial chemistry
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4
المؤلفون: Rogelio Lira, Marc O. Anderson, Paulina Rodriguez, Armann Andaya, Nohemy Celis, Nicholas Trieu, Nimrat Brar, Ngoc Huynh, Aaron Keniston, Brian Vidal, Hannah Fejzic, Emmett Pompa, Nikolay Masvlov, Gulbag Kahlon, Jeremy P. Mallari, Jeff P. Chance, Scott Eagon
المصدر: Bioorganic & Medicinal Chemistry Letters. 32:127683
مصطلحات موضوعية: Proteases, medicine.medical_treatment, Plasmodium falciparum, Clinical Biochemistry, Protozoan Proteins, Pharmaceutical Science, Hydroxamic Acids, 01 natural sciences, Biochemistry, Antimalarials, Structure-Activity Relationship, chemistry.chemical_compound, parasitic diseases, Drug Discovery, medicine, Parasite hosting, Piperazine, Molecular Biology, Binding Sites, Hydroxamic acid, Protease, biology, 010405 organic chemistry, Organic Chemistry, Metalloendopeptidases, biology.organism_classification, 0104 chemical sciences, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, chemistry, Molecular Medicine, Lead compound, Function (biology)
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5
المؤلفون: Teodulo Crisanto, Hannah Fejzic, Brian Vidal, Armann Andaya, Jeremy P. Mallari, Jeffrey P. Chance, Bradley Kuwahara, Daniel E. Goldberg, Ruby Aispuro, Nikolay S. Maslov, Eva S. Istvan, Obiel Hernandez, Corey Pugne Andanado, Whitney Serrano, Huyen Nguyen
المصدر: Bioorganicmedicinal chemistry letters. 28(10)
مصطلحات موضوعية: 0301 basic medicine, medicine.medical_treatment, Clinical Biochemistry, Plasmodium falciparum, Druggability, Protozoan Proteins, Pharmaceutical Science, Hydroxamic Acids, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, Antimalarials, Inhibitory Concentration 50, Structure-Activity Relationship, Drug Discovery, medicine, Protease Inhibitors, Molecular Biology, Piperazine, Metalloproteinase, Hydroxamic acid, Protease, biology, Organic Chemistry, Metalloendopeptidases, biology.organism_classification, 030104 developmental biology, chemistry, Human parasite, Molecular Medicine, Function (biology)
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6
المؤلفون: Anna Oksman, Jeremy P. Mallari, Barbara A. Vaupel, Daniel E. Goldberg
المصدر: Journal of Biological Chemistry. 289:30025-30039
مصطلحات موضوعية: TRNA modification, Protein family, Immunoprecipitation, Molecular Sequence Data, Plasmodium falciparum, Protozoan Proteins, Apicoplasts, Biochemistry, Ribosome, Mass Spectrometry, Conserved sequence, Cytosol, Nucleic Acids, Animals, Cluster Analysis, Humans, Parasites, Amino Acid Sequence, Protein Interaction Maps, Molecular Biology, Alleles, Conserved Sequence, Phylogeny, Life Cycle Stages, Apicoplast, biology, Molecular Sequence Annotation, Cell Biology, DNA, Protozoan, biology.organism_classification, Recombinant Proteins, Cell Compartmentation, Cell biology, Transport protein, Protein Transport, RNA, Ribosomal, Ribosomes, Sequence Alignment, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d48231f9d83ee88de6035fbb48485e67
https://doi.org/10.1074/jbc.m114.586735 -
7
المؤلفون: Neekesh V. Dharia, Victoria C. Corey, Daniel E. Goldberg, Eva S. Istvan, Elizabeth A. Winzeler, Garland R. Marshall, Jeremy P. Mallari
المصدر: Nature Communications
Nature Communications, Vol 8, Iss 1, Pp 1-8 (2017)مصطلحات موضوعية: 0301 basic medicine, Science, 030106 microbiology, Mutant, Plasmodium falciparum, Drug Resistance, Protozoan Proteins, General Physics and Astronomy, Drug resistance, medicine.disease_cause, Esterase, General Biochemistry, Genetics and Molecular Biology, Article, law.invention, 03 medical and health sciences, chemistry.chemical_compound, Antimalarials, law, Pepstatins, medicine, Prodrugs, Mutation, Multidisciplinary, biology, Esterases, General Chemistry, Prodrug, biology.organism_classification, Molecular biology, 3. Good health, 030104 developmental biology, Biochemistry, chemistry, Recombinant DNA, Pepstatin
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8
المؤلفون: Reto Brun, Marcel Kaiser, Fangyi Zhu, Andrew Lemoff, Jeremy P. Mallari, Min Lu, R. Kiplin Guy
المصدر: Bioorganic & Medicinal Chemistry. 18:8302-8309
مصطلحات موضوعية: medicine.medical_treatment, Trypanosoma brucei brucei, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Trypanosoma brucei, Pharmacology, Biochemistry, Mice, In vivo, Nitriles, parasitic diseases, Drug Discovery, medicine, Animals, Humans, Protease Inhibitors, Protease inhibitor (pharmacology), African trypanosomiasis, Molecular Biology, Protease, biology, Organic Chemistry, Trypanosoma brucei rhodesiense, biology.organism_classification, medicine.disease, Trypanocidal Agents, Cysteine Endopeptidases, Disease Models, Animal, Trypanosomiasis, African, Purines, Enzyme inhibitor, biology.protein, Molecular Medicine, Ex vivo
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9
المؤلفون: Aaron Kosinski, R. Kiplin Guy, James H. McKerrow, Fangyi Zhu, Conor R. Caffrey, Michele Connelly, Anang A. Shelat, Jeremy P. Mallari
المصدر: Journal of Medicinal Chemistry. 52:6489-6493
مصطلحات موضوعية: Models, Molecular, Protein Conformation, Cathepsin L, Trypanosoma brucei brucei, Article, Cathepsin B, Cell Line, Substrate Specificity, Drug Discovery, Animals, Humans, Protease Inhibitors, Cytotoxicity, Trypanocidal agent, Cathepsin, biology, Drug discovery, Chemistry, Biological activity, Trypanocidal Agents, Cysteine Endopeptidases, Biochemistry, Purines, Enzyme inhibitor, biology.protein, Molecular Medicine
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10
المؤلفون: Jeremy P. Mallari, Guiguemde Wendyam Armand, R. Kiplin Guy
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:3546-3549
مصطلحات موضوعية: Thiosemicarbazones, Purine, Proteases, Plasmodium falciparum, Clinical Biochemistry, Pharmaceutical Science, Cysteine Proteinase Inhibitors, Biochemistry, Article, Antimalarials, chemistry.chemical_compound, Chloroquine, Nitriles, Drug Discovery, medicine, Animals, Protease inhibitor (pharmacology), Molecular Biology, biology, Chemistry, Organic Chemistry, biology.organism_classification, Cysteine protease, Purines, Enzyme inhibitor, biology.protein, Molecular Medicine, medicine.drug