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1
المصدر: Medicinal chemistry (Shariqah (United Arab Emirates)). 12(6)
مصطلحات موضوعية: Models, Molecular, Quinuclidines, Stereochemistry, 02 engineering and technology, Ligands, 01 natural sciences, Partial agonist, PC12 Cells, Nicotine, Rats, Sprague-Dawley, Drug Discovery, medicine, Animals, Humans, Drug Partial Agonism, Nicotinic Agonists, Receptor, Neurotransmitter Agents, 010405 organic chemistry, Ligand, Chemistry, 021001 nanoscience & nanotechnology, Acetylcholine, 0104 chemical sciences, Rats, Nicotinic agonist, Biochemistry, Female, Carbamates, Alpha-4 beta-2 nicotinic receptor, 0210 nano-technology, medicine.drug, Ethers, Synaptosomes
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::865cc7f21f3745aae5b9989fbcc0f67a
https://pubmed.ncbi.nlm.nih.gov/26833074 -
2
المؤلفون: William M. Mitchell, Yashwant M. Deo, Miroslaw K. Gorny, Constance Williams, Tibor Keler, Jerome L. Gabriel, Sherri Burda, Susan Zolla-Pazner
مصطلحات موضوعية: Bispecific antibody, business.industry, Immunology, Human immunodeficiency virus (HIV), medicine, Functional studies, Receptor type, medicine.disease_cause, business, Virology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::51ea08f871221ba08eb69241d2226dfd
https://doi.org/10.1159/000425174 -
3Biososteric Replacement in the Design and Synthesis of Ligands for Nicotinic Acetylcholine Receptors
المؤلفون: Weilin Sun, Jerome L. Gabriel, Michael P. Blanton, Daniel J. Canney
المصدر: Medicinal Chemistry Research. 14:241-259
مصطلحات موضوعية: chemistry.chemical_compound, Nicotinic agonist, Ganglion type nicotinic receptor, Chemistry, Organic Chemistry, Muscarinic acetylcholine receptor, Pyridine, Muscarinic acetylcholine receptor M3, General Pharmacology, Toxicology and Pharmaceutics, Alpha-4 beta-2 nicotinic receptor, Medicinal chemistry, Pyrrolidine, Acetylcholine receptor
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4
المصدر: Bioconjugate Chemistry. 15:1068-1075
مصطلحات موضوعية: Male, Models, Molecular, Molecular model, Stereochemistry, Embolism, Molecular Sequence Data, Biomedical Engineering, Pharmaceutical Science, Bioengineering, Peptide, Plasma protein binding, Mice, chemistry.chemical_compound, Dogs, Animals, Humans, Amino Acid Sequence, Binding site, Radionuclide Imaging, Peptide sequence, Pharmacology, chemistry.chemical_classification, Tricine, Chemistry, Organic Chemistry, Thrombosis, In vitro, Biochemistry, Drug Design, Platelet aggregation inhibitor, Peptides, Platelet Aggregation Inhibitors, Protein Binding, Snake Venoms, Biotechnology
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5
المؤلفون: Richard L. Beard, Kenneth J. Soprano, Jerome L. Gabriel, Juliet M. Hutcheson, Carlo J. Gambone, Dianne Robert Soprano, Roshantha A.S. Chandraratna
المصدر: Molecular Pharmacology. 61:334-342
مصطلحات موضوعية: Transcriptional Activation, Aryl hydrocarbon receptor nuclear translocator, Protein Conformation, medicine.drug_class, Blotting, Western, Retinoic acid, Adamantane, Naphthalenes, Retinoid X receptor, Binding, Competitive, Retinoids, chemistry.chemical_compound, Cytochrome P-450 CYP1A1, Tumor Cells, Cultured, medicine, Humans, Retinoid, Promoter Regions, Genetic, Transcription factor, Pharmacology, biology, DNA, respiratory system, Aryl hydrocarbon receptor, Enzyme Activation, Retinoic acid receptor, Receptors, Aryl Hydrocarbon, chemistry, Biochemistry, Nuclear receptor, biology.protein, Molecular Medicine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fee75fb1bb979a5453cd5aa4e9eaf2e9
https://doi.org/10.1124/mol.61.2.334 -
6
المؤلفون: Kenneth J. Soprano, Roshantha A.S. Chandraratna, Jerome L. Gabriel, Sabina N. Sheikh, Carlo J. Gambone, Dianne Robert Soprano, D. M. Kochhar
المصدر: Toxicology and Applied Pharmacology. 174:153-159
مصطلحات موضوعية: Male, medicine.medical_specialty, Aryl hydrocarbon receptor nuclear translocator, Receptors, Retinoic Acid, medicine.drug_class, Retinoic acid, Tretinoin, Naphthalenes, Biology, Retinoid X receptor, Toxicology, Mice, chemistry.chemical_compound, Internal medicine, Cytochrome P-450 CYP1A1, medicine, Animals, RNA, Messenger, Retinoid, Receptor, Cells, Cultured, Pharmacology, Differential display, Aryl Hydrocarbon Receptor Nuclear Translocator, respiratory system, Embryo, Mammalian, Aryl hydrocarbon receptor, DNA-Binding Proteins, Retinoic acid receptor, Endocrinology, Receptors, Aryl Hydrocarbon, chemistry, embryonic structures, biology.protein, Female, Transcription Factors
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7
المؤلفون: Jerome L. Gabriel, Zeng-Ping Zhang, Kenneth J. Soprano, Dianne Robert Soprano, Muna Shukri, Carlo J. Gambone
المصدر: Archives of Biochemistry and Biophysics. 380:339-346
مصطلحات موضوعية: Transcriptional Activation, Receptors, Retinoic Acid, medicine.drug_class, Biophysics, Retinoic acid, Tretinoin, In Vitro Techniques, Biochemistry, Mice, chemistry.chemical_compound, Transactivation, Serine, Homologous chromosome, medicine, Animals, Retinoid, Amino acid residue, Receptor, Molecular Biology, DNA Primers, Binding Sites, Base Sequence, Retinoic Acid Receptor alpha, Ligand binding domain, Recombinant Proteins, Protein Structure, Tertiary, Cell biology, Kinetics, chemistry, Mutagenesis, Site-Directed
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8
المصدر: Journal of Biological Chemistry. 275:13558-13563
مصطلحات موضوعية: Protein Conformation, Molecular Sequence Data, Autoimmunity, Biochemistry, Epitope, Histones, Mice, Antigen, Antibody Specificity, Histone H2B, Animals, Amino Acid Sequence, Molecular Biology, Autoantibodies, Genes, Immunoglobulin, biology, Autoantibody, Antibodies, Monoclonal, Cell Biology, Molecular biology, Primary and secondary antibodies, Chromatin, Histone, Immunoglobulin G, biology.protein, Antibody
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::16e311ad1001f9065509585b937e20ed
https://doi.org/10.1074/jbc.275.18.13558 -
9
المؤلفون: Parkson Lee-Gau Chong, Jerome L. Gabriel
المصدر: Chemistry and Physics of Lipids. 105:193-200
مصطلحات موضوعية: Sulfolobus acidocaldarius, Lipid Bilayers, Biophysics, Glyceryl Ethers, Cyclopentanes, Biochemistry, Biophysical Phenomena, Diglycerides, Membrane Lipids, chemistry.chemical_compound, Molecular dynamics, Organic chemistry, Computer Simulation, Electrochemical gradient, Cyclopentane, Molecular Biology, Chemistry, Organic Chemistry, Cell Biology, Interaction energy, Hydrogen-Ion Concentration, Crystallography, Membrane, Dipalmitoylphosphatidylcholine, Methyl group
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10
المؤلفون: William F. Wade, Doug Demian, Jerome L. Gabriel, B. George Barisas, Thomas Nydam, Shyam Yadati, Terri K. Wade
المصدر: Immunology Letters. 67:47-55
مصطلحات موضوعية: Molecular model, Stereochemistry, Dimer, Immunology, Mutant, Antigen presentation, medicine.disease_cause, Epitope, Mice, chemistry.chemical_compound, Image Processing, Computer-Assisted, medicine, Animals, Humans, Immunology and Allergy, chemistry.chemical_classification, Antigen Presentation, Mutation, Chemistry, Adenine, HLA-DR1 Antigen, Histocompatibility Antigens Class II, Inosine, Amino acid, Biochemistry, Pyrimidine Dimers, Salt bridge