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1
المؤلفون: Frances Lu, Bryan G. Johnson, Daniel Ursu, Joan H. Carter, Lisa M. Broad, Kofi Adragni, Shane Atwell, Jing Wang, David K. Clawson, Beverly A. Heinz, Steven P. Swanson, James A. Monn, Qi Chen, Helene E. Sanger, David B. Shaw, Steven Marc Massey, Xushan Wang, Marijane Russell, Steven S. Henry, Junliang Hao, Rajni M. Bhardwaj, Diseroad Benjamin Alan, David L. McKinzie, Brian G. Getman, John T. Catlow
المصدر: Journal of Medicinal Chemistry. 61:2303-2328
مصطلحات موضوعية: 0301 basic medicine, chemistry.chemical_classification, Agonist, Bicyclic molecule, Stereochemistry, medicine.drug_class, Glutamate binding, Ligand (biochemistry), Small molecule, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Metabotropic receptor, Dicarboxylic acid, chemistry, Drug Discovery, medicine, Molecular Medicine, Receptor, 030217 neurology & neurosurgery
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2
المؤلفون: Chuanxi Xiang, Steven Swanson, Joan H. Carter, Paul L. Ornstein, Lisa M. Broad, Charles H. Mitch, Xu Shan Wang, Wesley H. Anderson, Helen E. Sanger, Renhua Li, Jeffrey M. Witkin, Stephon C. Smith, Stephen M. Fitzjohn, Francesca Pasqui, Xia Li, Jodi L. Smith, James A. Monn, Beverly A. Heinz, John T. Catlow
المصدر: Neuropharmacology. 115:100-114
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, medicine.drug_class, Metabotropic glutamate receptor 5, Metabotropic glutamate receptor 7, Metabotropic glutamate receptor 6, Biology, Receptor antagonist, 03 medical and health sciences, Cellular and Molecular Neuroscience, 030104 developmental biology, 0302 clinical medicine, Metabotropic receptor, Metabotropic glutamate receptor, medicine, Metabotropic glutamate receptor 1, Long-term depression, 030217 neurology & neurosurgery
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3
المؤلفون: Junliang Hao, Robert F. Bruns, Beverly A. Heinz, Joan H. Carter, James P. Beck, Kjell A. Svensson, Yue-Wei Qian, Sheila P. Little, Robert Alan Gadski, John Mehnert Schaus, Xushan Wang, Charles R. Yang, Lisa Selsam Beavers
المصدر: Molecular pharmacology. 94(4)
مصطلحات موضوعية: 0301 basic medicine, Allosteric modulator, Dopamine, Allosteric regulation, Cell Line, 03 medical and health sciences, 0302 clinical medicine, Dopamine receptor D1, Allosteric Regulation, Animals, Humans, Homology modeling, Binding site, Amino Acids, Receptor, Conserved Sequence, Pharmacology, Alanine, Chemistry, Receptors, Dopamine D1, Isoquinolines, Molecular biology, Rats, Transmembrane domain, 030104 developmental biology, HEK293 Cells, Molecular Medicine, 030217 neurology & neurosurgery, Allosteric Site
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dfb145a6374970273781446aa5024dd7
https://pubmed.ncbi.nlm.nih.gov/30111649 -
4
المؤلفون: James A, Monn, Steven S, Henry, Steven M, Massey, David K, Clawson, Qi, Chen, Benjamin A, Diseroad, Rajni M, Bhardwaj, Shane, Atwell, Frances, Lu, Jing, Wang, Marijane, Russell, Beverly A, Heinz, Xu-Shan, Wang, Joan H, Carter, Brian G, Getman, Kofi, Adragni, Lisa M, Broad, Helene E, Sanger, Daniel, Ursu, John T, Catlow, Steven, Swanson, Bryan G, Johnson, David B, Shaw, David L, McKinzie, Junliang, Hao
المصدر: Journal of medicinal chemistry. 61(6)
مصطلحات موضوعية: Male, Models, Molecular, Neurons, Molecular Structure, Phencyclidine, Motor Activity, Crystallography, X-Ray, Receptors, Metabotropic Glutamate, Rats, Molecular Docking Simulation, Rats, Sprague-Dawley, Bridged Bicyclo Compounds, Cyclic AMP, Excitatory Amino Acid Agonists, Animals, Humans, Excitatory Amino Acid Antagonists, Protein Binding
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5
المؤلفون: Mark G. Bures, David Edward Tupper, Joan H. Carter, James A. Monn, David L. McKinzie, Marijane Russell, Lourdes Prieto, Steven S. Henry, Reinhard Matthew Robert, Alicia Marcos, Lesley Walton, Christopher David Beadle, Bryan G. Johnson, Brian G. Getman, John T. Catlow, Frances Lu, Xushan Wang, Lorena Taboada, S. Richard Baker, Beverly A. Heinz, Helene Rudyk, David B. Shaw, Jaime Blanco, Carlos Lamas, Steven Swanson, David K. Clawson, Junliang Hao, Carlos Montero, Teresa Man, Shane Atwell, Barry Peter Clark, Jing Wang
المصدر: Journal of Medicinal Chemistry. 58:7526-7548
مصطلحات موضوعية: Agonist, chemistry.chemical_classification, Bicyclic molecule, medicine.drug_class, Stereochemistry, Allosteric regulation, Stereoisomerism, Partial agonist, Dicarboxylic acid, Protein structure, chemistry, Biochemistry, Drug Discovery, medicine, Molecular Medicine, Receptor
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6
المؤلفون: Junliang Hao, Matt R. Reinhard, Barry Peter Clark, Jaime Blanco, Concepción Pedregal, Shane Atwell, Michael P. Johnson, Paul Goldsmith, Carlos Montero, Rosa Maria A. Simmons, James A. Monn, Steven Swanson, Chuanxi Xiang, Bryan G. Johnson, Frances Lu, Lorena Taboada, Teresa Man, David K. Clawson, Marijane Russell, Lesley Walton, Steven S. Henry, Jing Wang, Beverly A. Heinz, S. Richard Baker, Helen E. Sanger, Xushan Wang, David B. Shaw, Lourdes Prieto, Mark G. Bures, Joan H. Carter, Lisa M. Broad, Kelly L. Knopp, Helene Rudyk, David L. McKinzie, David Edward Tupper, Christopher David Beadle, John T. Catlow, Carlos Lamas, Alicia Marcos
المصدر: Journal of Medicinal Chemistry. 58:1776-1794
مصطلحات موضوعية: Agonist, Chemistry, medicine.drug_class, Stereochemistry, Metabotropic glutamate receptor 5, Receptor agonist activity, Biochemistry, Metabotropic glutamate receptor, Drug Discovery, medicine, Molecular Medicine, Metabotropic glutamate receptor 1, Inverse agonist, Metabotropic glutamate receptor 2, Endogenous agonist
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7
المؤلفون: Reinhard Matthew Robert, James A. Monn, Bryan G. Johnson, Xushan Wang, Matthew John Valli, Beverly A. Heinz, Mark G. Bures, Steven S. Henry, Brian G. Getman, Joan H. Carter, John T. Catlow, Junliang Hao, David L. McKinzie, Steven Marc Massey, Marc Herin, Steven Swanson, Gregory A. Stephenson
المصدر: Journal of Medicinal Chemistry. 56:4442-4455
مصطلحات موضوعية: Male, Models, Molecular, Agonist, medicine.drug_class, Stereochemistry, Administration, Oral, Motor Activity, Pharmacology, Receptors, Metabotropic Glutamate, Rats, Sprague-Dawley, Bridged Bicyclo Compounds, Structure-Activity Relationship, Cyclohexanes, Drug Discovery, medicine, Animals, Humans, Receptor, Metabotropic glutamate receptor 5, Chemistry, Glutamate receptor, Stereoisomerism, Amino Acids, Dicarboxylic, Rats, HYDIA, Metabotropic receptor, Psychotic Disorders, Molecular Medicine, Metabotropic glutamate receptor 1, Receptor antagonist activity, Antipsychotic Agents
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8
المؤلفون: Jeffrey M, Witkin, Paul L, Ornstein, Charles H, Mitch, Renhua, Li, Stephon C, Smith, Beverly A, Heinz, Xu-Shan, Wang, Chuanxi, Xiang, Joan H, Carter, Wesley H, Anderson, Xia, Li, Lisa M, Broad, Francesca, Pasqui, Stephen M, Fitzjohn, Helen E, Sanger, Jodi L, Smith, John, Catlow, Steven, Swanson, James A, Monn
المصدر: Neuropharmacology. 115
مصطلحات موضوعية: Cerebral Cortex, Male, Rats, Sprague-Dawley, Dose-Response Relationship, Drug, Cyclohexanes, Animals, Humans, Receptors, Metabotropic Glutamate, Excitatory Amino Acid Antagonists, Cell Line, Rats
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9
المؤلفون: James A, Monn, Lourdes, Prieto, Lorena, Taboada, Junliang, Hao, Matthew R, Reinhard, Steven S, Henry, Christopher D, Beadle, Lesley, Walton, Teresa, Man, Helene, Rudyk, Barry, Clark, David, Tupper, S Richard, Baker, Carlos, Lamas, Carlos, Montero, Alicia, Marcos, Jaime, Blanco, Mark, Bures, David K, Clawson, Shane, Atwell, Frances, Lu, Jing, Wang, Marijane, Russell, Beverly A, Heinz, Xushan, Wang, Joan H, Carter, Brian G, Getman, John T, Catlow, Steven, Swanson, Bryan G, Johnson, David B, Shaw, David L, McKinzie
المصدر: Journal of medicinal chemistry. 58(18)
مصطلحات موضوعية: Male, Models, Molecular, Stereoisomerism, Motor Activity, Triazoles, Receptors, Metabotropic Glutamate, Binding, Competitive, Protein Structure, Tertiary, Drug Partial Agonism, Rats, Sprague-Dawley, Bridged Bicyclo Compounds, Mice, Dogs, Allosteric Regulation, Cyclic AMP, Mutagenesis, Site-Directed, Animals, Humans, Calcium
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10
المؤلفون: James A, Monn, Lourdes, Prieto, Lorena, Taboada, Concepcion, Pedregal, Junliang, Hao, Matt R, Reinhard, Steven S, Henry, Paul J, Goldsmith, Christopher D, Beadle, Lesley, Walton, Teresa, Man, Helene, Rudyk, Barry, Clark, David, Tupper, S Richard, Baker, Carlos, Lamas, Carlos, Montero, Alicia, Marcos, Jaime, Blanco, Mark, Bures, David K, Clawson, Shane, Atwell, Frances, Lu, Jing, Wang, Marijane, Russell, Beverly A, Heinz, Xushan, Wang, Joan H, Carter, Chuanxi, Xiang, John T, Catlow, Steven, Swanson, Helen, Sanger, Lisa M, Broad, Michael P, Johnson, Kelly L, Knopp, Rosa M A, Simmons, Bryan G, Johnson, David B, Shaw, David L, McKinzie
المصدر: Journal of medicinal chemistry. 58(4)
مصطلحات موضوعية: Male, Models, Molecular, Rats, Sprague-Dawley, Bridged Bicyclo Compounds, Animals, Humans, Spiro Compounds, Crystallography, X-Ray, Receptors, Metabotropic Glutamate, Protein Structure, Tertiary, Rats