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1دورية أكاديمية
المؤلفون: Sven Ruf, Sridharan Rajagopal, Sanjay Venkatachalapathi Kadnur, Mahanandeesha S. Hallur, Shilpa Rani, Rajendra Kristam, Srinivasan Swaminathan, Bharat Ravindra Zope, Pavan Kumar Gondrala, Indu Swamy, V. P. Rama Kishore Putta, Saravanan Kandan, Gernot Zech, Herman Schreuder, Christine Rudolph, Ralf Elvert, Joerg Czech, Swarnakumari Birudukota, M. Amir Siddiqui, Niranjan Naranapura Anand, Vishal Subhash Mane, Sreekanth Dittakavi, Juluri Suresh, Ramachandraiah Gosu, Mullangi Ramesh, Takeshi Yura, Saravanakumar Dhakshinamoorthy, Aimo Kannt
المصدر: Scientific Reports, Vol 12, Iss 1, Pp 1-18 (2022)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2045-2322
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2دورية أكاديمية
المؤلفون: Aimo Kannt, Sridharan Rajagopal, Mahanandeesha S. Hallur, Indu Swamy, Rajendra Kristam, Saravanakumar Dhakshinamoorthy, Joerg Czech, Gernot Zech, Herman Schreuder, Sven Ruf
المصدر: Molecules, Vol 26, Iss 4, p 991 (2021)
مصطلحات موضوعية: nicotinamide-N-methyltransferase, small molecule inhibitor, nicotinamide, metabolic disease, X-ray, Organic chemistry, QD241-441
وصف الملف: electronic resource
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3
المؤلفون: Patrick Shum, Thomas Licher, John L. Kane, Carolin Gerbeth-Kreul, Gerhard Hessler, Antje Pommereau, Sven Ruf, Christian Engel, Linli Wei, Joerg Czech, Theresa A Kuntzweiler
المصدر: SLAS Discovery. 26:783-797
مصطلحات موضوعية: 0301 basic medicine, Chemistry, Biological membrane, Transporter, Biochemistry, Small molecule, Analytical Chemistry, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Membrane, Direct assay, Biological target, Biophysics, Molecular Medicine, Amino acid transporter, Patch clamp, 030217 neurology & neurosurgery, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::44e4fb083c4e35d492c537df0250e79a
https://doi.org/10.1177/24725552211011180 -
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المؤلفون: Carolin, Gerbeth-Kreul, Antje, Pommereau, Sven, Ruf, John L, Kane, Theresa, Kuntzweiler, Gerhard, Hessler, Christian K, Engel, Patrick, Shum, LinLi, Wei, Joerg, Czech, Thomas, Licher
المصدر: SLAS discovery : advancing life sciences RD. 26(6)
مصطلحات موضوعية: Patch-Clamp Techniques, Cell Membrane, Reproducibility of Results, Biological Transport, CHO Cells, Electrophysiological Phenomena, High-Throughput Screening Assays, Small Molecule Libraries, Mice, Amino Acid Transport Systems, Neutral, Cricetulus, Animals, Humans, Biological Assay
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::b9160baf68ccf7faf0016023ba5f4dc1
https://pubmed.ncbi.nlm.nih.gov/33955247 -
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المؤلفون: Indu N. Swamy, Mahanandeesha S. Hallur, Saravanakumar Dhakshinamoorthy, Rajendra Kristam, Sven Ruf, Aimo Kannt, Sridharan Rajagopal, Gernot Zech, Herman Schreuder, Joerg Czech
المساهمون: Publica
المصدر: Molecules
Volume 26
Issue 4
Molecules, Vol 26, Iss 991, p 991 (2021)مصطلحات موضوعية: Models, Molecular, Niacinamide, Pharmaceutical Science, Adipose tissue, nicotinamide, Nicotinamide N-methyltransferase, Ligands, Article, Analytical Chemistry, Substrate Specificity, lcsh:QD241-441, X-ray, 03 medical and health sciences, chemistry.chemical_compound, Mice, 0302 clinical medicine, lcsh:Organic chemistry, Metabolic Diseases, Drug Discovery, medicine, Nicotinamide N-Methyltransferase, Animals, Humans, nicotinamide-N-methyltransferase, Physical and Theoretical Chemistry, Enzyme Inhibitors, 030304 developmental biology, chemistry.chemical_classification, 0303 health sciences, Binding Sites, Nicotinamide, Organic Chemistry, Skeletal muscle, small molecule inhibitor, metabolic disease, Small molecule, High-Throughput Screening Assays, Rats, Cytosol, medicine.anatomical_structure, Enzyme, chemistry, Biochemistry, Chemistry (miscellaneous), 030220 oncology & carcinogenesis, Microsomes, Liver, Molecular Medicine, Cancer cell lines
وصف الملف: application/pdf
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6
المؤلفون: Nisha K. Anchan, Thomas Langer, Vishal Subhash Mane, Raghunadha Reddy Burri, Christine Rudolph, Herman Schreuder, Joerg Czech, Ramachandraiah Gosu, Rajendra Kristam, Saravanakumar Dhakshinamoorthy, Ramesh Mullangi, Juluri Suresh, Mahanandeesha S. Hallur, Sridharan Rajagopal, Takeshi Yura, Manvi Singh, Aimo Kannt, Devaraj Venkatapura Chandrasekar, Shama Shaik, Sanjay Venkatachalapathi Kadnur, V.P. Rama Kishore Putta, Lokesh Kananti Narasimhulu, Karthikai Raj Murugesan, Ravi Kanth Bhamidipati, Sven Ruf, Indu N. Swamy, Alexander Marker, Sayantani Sarkar
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:922-925
مصطلحات موضوعية: Niacinamide, 0301 basic medicine, Clinical Biochemistry, Pharmaceutical Science, Nicotinamide N-methyltransferase, Pharmacology, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Diabetes mellitus, Drug Discovery, Nicotinamide N-Methyltransferase, medicine, Humans, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, Nicotinamide, Organic Chemistry, Primary metabolite, medicine.disease, 030104 developmental biology, Enzyme, chemistry, 030220 oncology & carcinogenesis, Molecular Medicine
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7كتاب إلكتروني
المؤلفون: Hans-Jörg Czech, Kareen Kümpel, Rita Müller
نوع المادة: eBook.
تصنيفات: ART / Museum Studies, ART / Art & Politics
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8
المؤلفون: Martin Lorenz, Hans Peter Nestler, Otmar Klingler, Monica Donghi, Manfred Schudok, Herman Schreuder, Hauke Szillat, Joerg Czech, Hans Matter
المصدر: Bioorganicmedicinal chemistry letters. 14(14)
مصطلحات موضوعية: Molecular model, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Factor VIIa, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Fibrinolytic Agents, Drug Discovery, Binding site, Molecular Biology, Serine protease, Binding Sites, biology, Molecular Structure, Chemistry, Protease binding, Phenylurea Compounds, Organic Chemistry, Docking (molecular), Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Fibrinolytic agent, Peptide Hydrolases
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9
المؤلفون: Hans Matter, Manfred Schudok, Martin Lorenz, Peter Wildgoose, Hans Peter Nestler, Otmar Klingler, S. Paul Bajaj, Joerg Czech, Herman Schreuder
المصدر: ChemInform. 34
مصطلحات موضوعية: Models, Molecular, Molecular model, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Factor VIIa, Selective inhibition, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Amidine, chemistry.chemical_compound, Structure-Activity Relationship, Antithrombotic treatment, Drug Discovery, medicine, otorhinolaryngologic diseases, Humans, Structure–activity relationship, Molecular Biology, biology, Chemistry, Phenylurea Compounds, Organic Chemistry, Coagulation factor VIIa, General Medicine, Combinatorial chemistry, Design synthesis, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, sense organs
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10
المؤلفون: Sofia Mitaku, Jean-Claude Jacquesy, Jean-Pierre Gesson, Xia Dong, Manfred Gerken, Klaus Bosslet, François Tillequin, Claude Monneret, Brigitte Renoux, Joerg Czech, Jean-Claude Florent, Sylvie Michel, Rainer Straub, Michel Koch, Martine Mondon, Solo Andrianomenjanahary, Gilbert Gaudel
المصدر: Journal of medicinal chemistry. 41(19)
مصطلحات موضوعية: Daunorubicin, Recombinant Fusion Proteins, Glucuronates, Immunoglobulin Fab Fragments, Mice, Structure-Activity Relationship, Drug Stability, Drug Discovery, medicine, Escherichia coli, Tumor Cells, Cultured, Structure–activity relationship, Animals, Humans, Doxorubicin, Prodrugs, Cytotoxicity, Leukemia L1210, Glucuronidase, chemistry.chemical_classification, Antibiotics, Antineoplastic, Hydrolysis, Antibodies, Monoclonal, Adept, Prodrug, In vitro, Carcinoembryonic Antigen, Rats, Kinetics, Enzyme, chemistry, Biochemistry, Molecular Medicine, Drug Screening Assays, Antitumor, Cell Division, medicine.drug