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1دورية أكاديمية
المؤلفون: Dries Bauters, Mathias Cobbaut, Lotte Geys, Johan Van Lint, Bianca Hemmeryckx, H. Roger Lijnen
المصدر: Molecular Metabolism, Vol 6, Iss 7, Pp 715-724 (2017)
مصطلحات موضوعية: ADAMTS5, Brown adipose tissue, Browning, Beige, Thermogenesis, Obesity, Internal medicine, RC31-1245
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Mathias Cobbaut, Rita Derua, Heike Döppler, Hua Jane Lou, Sandy Vandoninck, Peter Storz, Benjamin E. Turk, Thomas Seufferlein, Etienne Waelkens, Veerle Janssens, Johan Van Lint
المصدر: Scientific Reports, Vol 7, Iss 1, Pp 1-17 (2017)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2045-2322
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المؤلفون: Thomas Seufferlein, Claudia Scholl, Stefan Fröhling, John Koren, Gabriela Chiosis, Johan van Lint, Hans Kestler, Alexander Becher, Felicitas Genze, Arefeh Rouhi, Cornelia Brunner, Kristina Diepold, Ninel Azoitei
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::45e7472c2655a483e5d4463c06336d14
https://doi.org/10.1158/0008-5472.22405673 -
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المؤلفون: Thomas Seufferlein, Claudia Scholl, Stefan Fröhling, John Koren, Gabriela Chiosis, Johan van Lint, Hans Kestler, Alexander Becher, Felicitas Genze, Arefeh Rouhi, Cornelia Brunner, Kristina Diepold, Ninel Azoitei
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2e158f575db770e38a67cfab73a0bb07
https://doi.org/10.1158/0008-5472.22405685.v1 -
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المؤلفون: Wim M. De Borggraeve, Lauren Voets, Philippe Gilles, Johan Van Lint
المصدر: ChemMedChem. 16:2158-2171
مصطلحات موضوعية: Gene isoform, Computational biology, Biology, 01 natural sciences, Biochemistry, Serine, Structure-Activity Relationship, Drug Development, Drug Discovery, Animals, Humans, Kinome, General Pharmacology, Toxicology and Pharmaceutics, Protein kinase A, Protein Kinase Inhibitors, Protein Kinase C, Pharmacology, Dose-Response Relationship, Drug, Molecular Structure, PKD1, 010405 organic chemistry, Kinase, Organic Chemistry, musculoskeletal system, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Cardiac hypertrophy, cardiovascular system, Molecular Medicine, PROTEIN KINASE D
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6
المؤلفون: Maria João Freitas, Steven De Jonghe, Sam Ceusters, Arnout Voet, Mathias Cobbaut, Dirk Daelemans, Koen Van Asch, Johan Van Lint, Rudra Kashyap, Anke Janssens, Philippe Gilles, Leentje Persoons, Wim M. De Borggraeve
مصطلحات موضوعية: Pyrimidine, Chemistry Techniques, Synthetic, macromolecular substances, 01 natural sciences, Inhibitory Concentration 50, 03 medical and health sciences, chemistry.chemical_compound, 3-IN-PP1, Cell Line, Tumor, Drug Discovery, medicine, Humans, Phosphorylation, Protein Kinase Inhibitors, Protein Kinase C, Cell Proliferation, 030304 developmental biology, Biological evaluation, Pharmacology, 0303 health sciences, Protein kinase D inhibitor, biology, 010405 organic chemistry, Chemistry, Organic Chemistry, 1-NM-PP1, Cancer, Biological activity, General Medicine, medicine.disease, musculoskeletal system, 0104 chemical sciences, Pyrimidines, Pyrazolo[3,4-d]pyrimidines, Design synthesis, Biochemistry, Drug Design, Anticancer agents, biology.protein, cardiovascular system, Pyrazoles, PROTEIN KINASE D, Cortactin
وصف الملف: Print-Electronic
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d10f8fc9d70fc54d72e8ca4755001d2a
https://lirias.kuleuven.be/handle/123456789/659296 -
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المؤلفون: Peter J. Parker, Johan Van Lint, Mathias Cobbaut, Veerle Janssens, Rita Derua, Etienne Waelkens
المصدر: Febs Letters
مصطلحات موضوعية: 0301 basic medicine, kinase, Biophysics, Inhibitory postsynaptic potential, Biochemistry, 03 medical and health sciences, Residue (chemistry), Structural Biology, In vivo, Chlorocebus aethiops, Research Letter, Genetics, Animals, Homeostasis, Humans, Amino Acid Sequence, Phosphorylation, Molecular Biology, Cells, Cultured, Protein Kinase C, dual‐specificity, PKD1, Mechanism (biology), Chemistry, Autophosphorylation, Cell Biology, musculoskeletal system, Research Letters, In vitro, Cell biology, Enzyme Activation, HEK293 Cells, 030104 developmental biology, COS Cells, Enzymology, Mutagenesis, Site-Directed, cardiovascular system, Tyrosine, Drosophila, autophosphorylation, protein kinase D
وصف الملف: Print-Electronic
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8
المؤلفون: Rudra Kashyap, Johan Van Lint, Olivia Appelmans, Arnout Voet, Wim M. De Borggraeve, Philippe Gilles
المصدر: Analytical Biochemistry. 630:114313
مصطلحات موضوعية: Paper, Biochemistry & Molecular Biology, Cation exchange paper, Biophysics, Biochemistry, Biochemical Research Methods, Protein kinase, Research community, Alternative paper, Luciferase, Kinase activity, Cellulose, Radiometry, Protein kinase A, Molecular Biology, Science & Technology, Kinase, Chemistry, Chemistry, Analytical, Cell Biology, Radiometric kinase assay, Physical Sciences, Phosphocellulose paper, Life Sciences & Biomedicine, Protein Kinases
وصف الملف: Print-Electronic
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المؤلفون: Johan Van Lint, Lotte Geys, Mathias Cobbaut, Dries Bauters, H. Roger Lijnen, Bianca Hemmeryckx
المصدر: Molecular Metabolism, Vol 6, Iss 7, Pp 715-724 (2017)
Molecular Metabolismمصطلحات موضوعية: 0301 basic medicine, Male, HFD, high-fat diet, ADAMTS, A disintesgrin and metalloproteinase with a thrombospondin type-1 motif, Adipose tissue, White adipose tissue, Brown adipose tissue, %ID/g, percentage injected dose per gram, chemistry.chemical_compound, Mice, 0302 clinical medicine, Adipose Tissue, Brown, Adipocyte, Cyclic AMP Response Element-Binding Protein, Cells, Cultured, WAT, white adipose tissue, Thermogenesis, Thermogenin, ECM, extracellular matrix, medicine.anatomical_structure, 030220 oncology & carcinogenesis, ADAMTS5, GON, gonadal, Original Article, β3-AR, beta-3 adrenergic receptor, Beta-3 adrenergic receptor, CAMP Responsive Element Binding Protein, medicine.medical_specialty, lcsh:Internal medicine, Adipose Tissue, White, SUV, standardized uptake value, Adrenergic beta-3 Receptor Agonists, Dioxoles, Biology, TLG, total lesion glycolysis, 03 medical and health sciences, Internal medicine, CREB, cAMP responsive element-binding protein, AT, adipose tissue, UCP1, uncoupling protein 1, medicine, Animals, Obesity, lcsh:RC31-1245, Molecular Biology, Beige, Cell Biology, BAT, brown adipose tissue, SC, subcutaneous, Mice, Inbred C57BL, 030104 developmental biology, Endocrinology, chemistry, ADAMTS5 Protein, Browning, Energy Metabolism
وصف الملف: Electronic-eCollection; application/pdf
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المؤلفون: Wim M. De Borggraeve, Lina Saadah, Johan Van Lint, Mathias Cobbaut, Arnout Voet, Klaas Verschueren, Joachim Demaerel
المصدر: MedChemComm. 8:640-646
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Specific protein, Pyrimidine, Stereochemistry, Kinase, Organic Chemistry, Pharmaceutical Science, Ligand (biochemistry), Biochemistry, Combinatorial chemistry, 3. Good health, 03 medical and health sciences, chemistry.chemical_compound, Pyrimidine analogue, 030104 developmental biology, chemistry, Drug Discovery, Molecular Medicine, PROTEIN KINASE D, Lead compound
وصف الملف: Print-Electronic; application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4c2c31f72905cc507c48809f53a82c24
https://doi.org/10.1039/c6md00675b