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1
المؤلفون: Karen A. Maegley, Kephart Susan Elizabeth, Christopher P. Dillon, Manli Shi, Kristen Jensen-Pergakes, Prakash B. Palde, Ya-Li Deng, Chi-Yeh Chung, Natalie Miller, John Sherrill, Wei Liu, Ryan L. Patman, Shinji Yamazaki, Tao Xie, Fen Wang, Hieu Lam, Eleanore Hendrickson, John F. Braganza, Yuli Wang, Robert Arnold Kumpf, Shannon Karlicek Bryant, Thomas A Paul, Noah Spiegel, Martin James Wythes, Amy Nemeth, Stephanie Scales, Elizabeth A. McMillan, Michelle Tran-Dubé, Alexei Brooun, Vesta Goshtasbi, Eugene Rui, Michele McTigue, Indrawan James Mcalpine, Tatlock John H
المصدر: Molecular Cancer Therapeutics. 21:3-15
مصطلحات موضوعية: Protein-Arginine N-Methyltransferases, S-Adenosylmethionine, Cancer Research, Cell signaling, Spliceosome, Lung Neoplasms, Chemistry, Cellular differentiation, Protein arginine methyltransferase 5, Alternative splicing, Drug Resistance, Apoptosis, Cell cycle, Mice, Oncology, Carcinoma, Non-Small-Cell Lung, Cell Line, Tumor, RNA splicing, Cancer cell, Cancer research, Animals, Humans, Female, Cell Proliferation
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::621805778a73d6732ba64af7ea279a54
https://doi.org/10.1158/1535-7163.mct-21-0620 -
2
المؤلفون: Eleanore Hendrickson, Martin James Wythes, Indrawan James Mcalpine, Karen A. Maegley, Christopher P. Dillon, Fen Wang, Kephart Susan Elizabeth, Amy Nemeth, Prakash B. Palde, Manli Shi, Kristen Jensen-Pergakes, Shinji Yamazaki, Tao Xie, Chi-Yeh Chung, Michelle Tran-Dubé, Tatlock John H, Stephanie Scales, Hieu Lam, Eugene Rui, Thomas A Paul, Elizabeth A. McMillan, Robert Arnold Kumpf, Ryan L. Patman, Michele McTigue, Natalie Miller, Ya-Li Deng, Yuli Wang, Noah Spiegel, Alexei Brooun, John Sherrill, Wei Liu, John F. Braganza
المصدر: Cancer Research. 81:1160-1160
مصطلحات موضوعية: Antitumor activity, Cancer Research, Oncology, Chemistry, Protein arginine methyltransferase 5, RNA splicing, Cancer research, Drug resistance
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ffac773af19496024ab15b63ff654a26
https://doi.org/10.1158/1538-7445.am2021-1160 -
3
المؤلفون: Huiling Shao, Jose M. Medina, Ryan T. Helsel, Peng Liu, Joseph Derosa, Indrawan James Mcalpine, John F. Braganza, Tuğçe G. Erbay, Christopher P. Ashcroft, Gary M. Gallego, Shouliang Yang, Paul F. Richardson, Ryan L. Patman, Keary M. Engle, Fen Wang, Taeho Kang, Michelle Tran-Dubé
المصدر: ACS Catal
مصطلحات موضوعية: Reaction conditions, Steric effects, Scope (project management), 010405 organic chemistry, Aryl, General Chemistry, 010402 general chemistry, 01 natural sciences, Combinatorial chemistry, Article, Catalysis, 0104 chemical sciences, Cyclopropane, chemistry.chemical_compound, Hydroboration, chemistry, Selectivity, Derivatization, Phosphine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3c4e3f4d66a75d1c1eab647eda2e78b1
https://doi.org/10.26434/chemrxiv.8341016.v1 -
4
المؤلفون: Michael R. Collins, Louise Bernier, Michelle Tran-Dubé, Botrous Iriny, Shijian Ren, Qingbin Zeng, Sacha Ninkovic, Neal W. Sach, John F. Braganza, Baojiang Zheng, Indrawan James Mcalpine, Baohua Li
المصدر: Tetrahedron Letters. 56:5757-5760
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Organic Chemistry, Drug Discovery, Intramolecular cyclization, Organic chemistry, Hydroamination, Biochemistry, Medicinal chemistry, Fluoride, Stoichiometry, Catalysis
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5
المؤلفون: Michelle Tran-Dubé, Bruce M. Bechle, Michelle Kraus, Ciarán N. Cronin, Kim James, Joseph S. Warmus, Fen Wang, Jianmin Sun, Indrawan James Mcalpine, Sacha Ninkovic, Jianwei Bian, Samantha Elizabeth Greasley, Neil J. Flanagan, Matthew Corbett, Rebecca Dias, Andrews Mark David, Asako Nagata, John F. Braganza, Linda Kitching, David C. Blakemore, Eric Johnson, Sarah Elizabeth Skerratt, Kiyoyuki Omoto, Sharan K. Bagal, Jingrong Jean Cui, James Bilsland, Peter J. Bungay, Rachel L. Grimley, Stephanie Scales, Gareth Waldron
المصدر: Journal of medicinal chemistry. 61(15)
مصطلحات موضوعية: 0301 basic medicine, animal structures, Protein Conformation, Pyridines, Pain, Tropomyosin receptor kinase B, Neurotrophin-3, Pharmacology, Tropomyosin receptor kinase A, Ligands, 030226 pharmacology & pharmacy, Tropomyosin receptor kinase C, 03 medical and health sciences, Structure-Activity Relationship, 0302 clinical medicine, Drug Discovery, Animals, Humans, Tissue Distribution, Protein Kinase Inhibitors, Brain-derived neurotrophic factor, biology, Chemistry, Receptor Protein-Tyrosine Kinases, Rats, Molecular Docking Simulation, 030104 developmental biology, Nerve growth factor, nervous system, Solubility, Trk receptor, biology.protein, Molecular Medicine, Neurotrophin
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المؤلفون: Hovhannes J. Gukasyan, Michael R. Collins, Sutton Scott Channing, Kephart Susan Elizabeth, Shinji Yamazaki, Sacha Ninkovic, Simon Bergqvist, Fen Wang, Robert Arnold Kumpf, Michael Ryskin, Patrick Bingham, Pei-Pei Kung, Dominique Verhelle, Brian Yip, Karen A. Maegley, Robert A. Rollins, Peter A. Wells, Martha A. Ornelas, Buwen Huang, Valeria Fantin, Xiu Yu, Stephanie Scales, Wade Diehl, Indrawan James Mcalpine, Cody Krivacic, Mei Cui, Lisa Nguyen, Wenyue Hu, Tatlock John H, Dac M. Dinh, Martin James Wythes, Connie Fan, Gary Li, Martin Paul Edwards, Rui Eugene Yuanjin, John F. Braganza, Zehnder Luke Raymond, Wei-Guo Zhang
المصدر: Journal of medicinal chemistry. 59(18)
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, Lactams, Stereochemistry, Pyridones, Antineoplastic Agents, Mice, SCID, 03 medical and health sciences, chemistry.chemical_compound, Mice, In vivo, Amide, Cell Line, Tumor, Neoplasms, Drug Discovery, Potency, Moiety, Animals, Humans, Enhancer of Zeste Homolog 2 Protein, Ligand efficiency, Isoquinolines, 030104 developmental biology, chemistry, Lipophilic efficiency, Cyclization, Drug Design, Lactam, Molecular Medicine, Female, Linker
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المؤلفون: John F. Braganza, null et al.
المصدر: ChemInform. 47
مصطلحات موضوعية: Chemistry, Organic chemistry, General Medicine, Catalysis
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المؤلفون: Michael R. Collins, Sacha Ninkovic, Benjamin F. Johnson, Michelle Tran-Dubé, Qinhua Huang, John F. Braganza, Neal W. Sach
المصدر: Tetrahedron Letters. 53:4372-4375
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, chemistry, Yield (chemistry), Organic Chemistry, Drug Discovery, Pyridine, Enol ether, Biochemistry, Combinatorial chemistry, Cycloaddition
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المؤلفون: Tanya Michelle Jewell, Robert Steven Kania, Anand Sistla, Bennett Michael John, Michael R. Gehring, Evan Smith, Zehnder Luke Raymond, Shinji Yamazaki, Karen A. Maegley, Elena Z. Dovalsantos, Ben Burke, Fen Wang, Sacha Ninkovic, Jeff Wang, Joe Zhongxiang Zhou, Pei-Pei Kung, Min-Jean Yin, Michael J. Hickey, Martin James Wythes, Jerry Meng, Buwen Huang, Ping Kang, John F. Braganza, Ketan S. Gajiwala, Tatlock John H, Pramod P. Mehta
المصدر: Journal of Medicinal Chemistry. 54:3368-3385
مصطلحات موضوعية: Pyrimidine, biology, Chemistry, Stereochemistry, medicine.drug_class, Carboxamide, Metabolic stability, Combinatorial chemistry, Hsp90, Bioavailability, chemistry.chemical_compound, Heat shock protein, Drug Discovery, Alkoxy group, biology.protein, medicine, Molecular Medicine, Potency
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المؤلفون: Indrawan James Mcalpine, Shinji Yamazaki, Wei Liu, Zhenxiong Wang, Michelle Tran-Dubé, Deng Ya-Li, Kristen Jensen-Pergakes, Brad Hirakawa, Ryan L. Patman, Karen A. Maegley, Joseph Billitti, Martin James Wythes, Tatlock John H, Fen Wang, Robert Arnold Kumpf, Tao Zhang, Stephanie Scales, Noah Spiegel, Rui Eugene Yuanjin, John F. Braganza, Michele McTigue, Alexei Brooun
المصدر: Cancer Research. 78:4857-4857
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Arginine, Chemistry, Protein arginine methyltransferase 5, Ligand (biochemistry), In vitro, 03 medical and health sciences, 030104 developmental biology, Protein structure, Oncology, Biochemistry, RNA splicing, Transcriptional regulation, Nucleoside
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::2b8092ccb21304e98d228226d2d47f11
https://doi.org/10.1158/1538-7445.am2018-4857