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1
المؤلفون: Kurt R. Gregor, Kim W. McIntyre, Carl Ouellet, Francis Beaulieu, Ruediger Edward H, Xuejie Yang, Yuping Qiu, Alain Martel, Dolatrai M. Vyas, Jacques Banville, F. Christopher Zusi, James R. Burke, Makonen Belema, John F. MacMaster, Mark A. Pattoli
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:1233-1237
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Heterocyclic Compounds, 4 or More Rings, environment and public health, Biochemistry, Chemical synthesis, Cell Line, Substrate Specificity, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Quinoxaline, In vivo, Quinoxalines, Drug Discovery, Humans, skin and connective tissue diseases, Protein kinase A, Molecular Biology, chemistry.chemical_classification, biology, Organic Chemistry, In vitro, I-kappa B Kinase, enzymes and coenzymes (carbohydrates), Enzyme, chemistry, Enzyme inhibitor, Quinazolines, Quinolines, biology.protein, Molecular Medicine, Benzimidazoles, biological phenomena, cell phenomena, and immunity, Tricyclic
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2
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:3591-3594
مصطلحات موضوعية: Paclitaxel, Stereochemistry, Clinical Biochemistry, Mice, Nude, Pharmaceutical Science, Biochemistry, Chemical synthesis, Dithiothreitol, Terpene, Inhibitory Concentration 50, Mice, chemistry.chemical_compound, In vivo, Drug Discovery, Tumor Cells, Cultured, medicine, Animals, Humans, Prodrugs, Disulfides, Cytotoxicity, Molecular Biology, Chemistry, Organic Chemistry, Disulfide bond, Captopril, General Medicine, Neoplasms, Experimental, Prodrug, Combinatorial chemistry, In vitro, Treatment Outcome, Molecular Medicine, Oxidation-Reduction, Cell Division, Half-Life, medicine.drug
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3
المؤلفون: T G Murali, Dhar, Zhongqi, Shen, Junqing, Guo, Chunjian, Liu, Scott H, Watterson, Henry H, Gu, William J, Pitts, Catherine A, Fleener, Katherine A, Rouleau, N Z, Sherbina, Kim W, McIntyre, David J, Shuster, Mark R, Witmer, Jeffrey A, Tredup, Bang-Chi, Chen, Rulin, Zhao, Mark S, Bednarz, Daniel L, Cheney, John F, MacMaster, Laura M, Miller, Karen K, Berry, Timothy W, Harper, Joel C, Barrish, Diane L, Hollenbaugh, Edwin J, Iwanowicz
المصدر: Journal of Medicinal Chemistry. 45:2127-2130
مصطلحات موضوعية: Male, Purine, Stereochemistry, Morpholines, Enzyme-Linked Immunosorbent Assay, Chemical synthesis, Mice, Structure-Activity Relationship, chemistry.chemical_compound, IMP Dehydrogenase, In vivo, IMP dehydrogenase, Drug Discovery, Animals, Structure–activity relationship, Nucleotide, Enzyme Inhibitors, Oxazoles, chemistry.chemical_classification, Mice, Inbred BALB C, biology, Mycophenolic Acid, Arthritis, Experimental, Rats, De novo synthesis, Biochemistry, chemistry, Rats, Inbred Lew, Enzyme inhibitor, Antibody Formation, biology.protein, Molecular Medicine
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4
المؤلفون: Philip M. Wallace, John F. MacMaster, Katherine A. Rouleau, T. Joseph Brown, James K. Loy, Karen L. Donaldson, Alan F. Wahl
المصدر: The Journal of Immunology. 162:5547-5555
مصطلحات موضوعية: Immunology, Immunology and Allergy
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::73dcb1d36adf8f331b20e5ab7a9fa889
https://doi.org/10.4049/jimmunol.162.9.5547 -
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المؤلفون: Philip M. Wallace, Jill Rillema, Jingpeng Peng, Samuel A. Burstein, Mohammed Shoyab, John F. MacMaster
المصدر: Blood. 86:1310-1315
مصطلحات موضوعية: medicine.medical_specialty, Immunology, Oncostatin M, Cell Biology, Hematology, Biology, Biochemistry, Blood cell, Haematopoiesis, Animal data, Endocrinology, medicine.anatomical_structure, Megakaryocyte, In vivo, Internal medicine, medicine, biology.protein, Platelet, Thrombopoiesis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::9de95c50075ea28ae5f57cefeac8d341
https://doi.org/10.1182/blood.v86.4.1310.bloodjournal8641310 -
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المؤلفون: Paul Gladstone, Jennifer S. Johnson, John F. MacMaster, Karen A. Kennedy, Peter S. Linsley, Philip M. Wallace
المصدر: Transplantation. 58:602-610
مصطلحات موضوعية: Immunoconjugates, T cell, Graft vs Host Disease, chemical and pharmacologic phenomena, CHO Cells, Major histocompatibility complex, Abatacept, Major Histocompatibility Complex, Mice, CD28 Antigens, Antigens, CD, T-Lymphocyte Subsets, immune system diseases, Cricetinae, Minor histocompatibility antigen, Animals, Humans, Medicine, CTLA-4 Antigen, Bone Marrow Transplantation, B-Lymphocytes, Transplantation, biology, business.industry, CD28, medicine.disease, Antigens, Differentiation, Mice, Inbred C57BL, Disease Models, Animal, surgical procedures, operative, medicine.anatomical_structure, Graft-versus-host disease, Immunology, biology.protein, Female, Bone marrow, business, CD80, Signal Transduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1b6eea3a00abc45aa8f25c1fb6163192
https://doi.org/10.1097/00007890-199409150-00013 -
7
المؤلفون: James R. Burke, Kurt R. Gregor, John F. MacMaster, Mark A. Pattoli
المصدر: The Journal of pharmacology and experimental therapeutics. 315(1)
مصطلحات موضوعية: IκB kinase, Cartilage metabolism, Matrix metalloproteinase, Gene Expression Regulation, Enzymologic, Chondrocytes, Quinoxalines, Animals, Humans, Lectins, C-Type, Aggrecans, Phosphorylation, Protein Kinase Inhibitors, Aggrecan, Pharmacology, Metalloproteinase, Thrombospondin, Extracellular Matrix Proteins, Chemistry, Imidazoles, ADAMTS4 Protein, Bovine Cartilage, Cell biology, ADAM Proteins, Cartilage, Biochemistry, Metalloproteases, Molecular Medicine, Cattle, Proteoglycans, ADAMTS5 Protein, Collagen, Procollagen N-Endopeptidase, Interleukin-1
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a8b11a2bc5ba15091c0f011454cc9dd0
https://pubmed.ncbi.nlm.nih.gov/16009742 -
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المؤلفون: Fred Christopher Zusi, Donna M. Dambach, James R. Burke, Yuping Qiu, K. K. Berry, D. B. Lee, John F. MacMaster
المصدر: Inflammation research : official journal of the European Histamine Research Society ... [et al.]. 52(12)
مصطلحات موضوعية: Immunology, Vascular Cell Adhesion Molecule-1, IκB kinase, Protein Serine-Threonine Kinases, Inflammatory bowel disease, Pathogenesis, chemistry.chemical_compound, Mice, Quinoxalines, medicine, Animals, Humans, BMS-345541, Colitis, Cells, Cultured, Pharmacology, Crohn's disease, business.industry, Tumor Necrosis Factor-alpha, Dextran Sulfate, Imidazoles, Endothelial Cells, medicine.disease, Intercellular Adhesion Molecule-1, Ulcerative colitis, digestive system diseases, I-kappa B Kinase, Sulfasalazine, Disease Models, Animal, chemistry, Gene Expression Regulation, Cancer research, Tumor necrosis factor alpha, business, Cell Adhesion Molecules
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المؤلفون: Kim W. McIntyre, Mark A. Pattoli, James R. Burke, Violetta Iotzova, Joann Strnad, Qiu Yuping, Patrick J. Brassil, Kurt R. Gregor, F. Christopher Zusi, Wendy Clarke, Xiaoxia Yang, John F. MacMaster
المصدر: The Journal of biological chemistry. 278(3)
مصطلحات موضوعية: Transcription, Genetic, Allosteric regulation, IκB kinase, Biology, Protein Serine-Threonine Kinases, environment and public health, Biochemistry, chemistry.chemical_compound, Mice, Catalytic Domain, Quinoxalines, Animals, BMS-345541, Enzyme Inhibitors, CHUK, Protein kinase A, Molecular Biology, Mice, Inbred BALB C, Kinase, Imidazoles, NF-kappa B, Cell Biology, Molecular biology, I-kappa B Kinase, enzymes and coenzymes (carbohydrates), IκBα, Kinetics, chemistry, Phosphorylation, Female, Allosteric Site
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::16f62b87cf59cb6cd6bac92c557bca08
https://pubmed.ncbi.nlm.nih.gov/12403772 -
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المؤلفون: Karen K. Berry, Davidson Thomas J, John F. MacMaster, Bharat Danle, James Loy, Stephen K. Durham
المصدر: Toxicologic pathology. 27(2)
مصطلحات موضوعية: medicine.medical_specialty, Lipopolysaccharide, 040301 veterinary sciences, medicine.medical_treatment, Anti-Inflammatory Agents, Antineoplastic Agents, Oncostatin M, Toxicology, 030226 pharmacology & pharmacy, Pathology and Forensic Medicine, 0403 veterinary science, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Internal medicine, medicine, Animals, Humans, Serum amyloid A, Interleukin 6, Molecular Biology, Inflammation, biology, business.industry, Experimental autoimmune encephalomyelitis, 04 agricultural and veterinary sciences, Cell Biology, medicine.disease, Disease Models, Animal, Cytokine, Endocrinology, chemistry, Toxicity, biology.protein, Cytokines, Tumor necrosis factor alpha, business, Peptides
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::19064cc5e90fe7668f9ec6508ba885ed
https://pubmed.ncbi.nlm.nih.gov/10207978