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1دورية أكاديمية
المؤلفون: Fernando Orden Rueda, Michal Bista, Matthew D. Newton, Anne U. Goeppert, M. Emanuela Cuomo, Euan Gordon, Felix Kröner, Jon A. Read, Jonathan D. Wrigley, David Rueda, Benjamin J. M. Taylor
المصدر: Nature Communications, Vol 8, Iss 1, Pp 1-11 (2017)
مصطلحات موضوعية: Science
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2041-1723
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المؤلفون: John Brognard, Owen J. Sansom, Tony Hunter, Crispin J. Miller, Ewelina Testoni, Matthew Collier, Ross Overman, Isabelle Green, Chris Phillips, Hannah K. Pollard, Claire Brassington, Jon A. Read, Lorena A. Puto, Phil Chapman, Susan Mason, Karen Blyth, Yaoyong Li, Eleanor W. Trotter, Hayeon Baik, Natalie L. Stephenson, Anna A. Marusiak
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8d0722c76c95b7bbc4901db1e2b3ae68
https://doi.org/10.1158/0008-5472.22409912 -
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المؤلفون: David Longmire, Haley Woods, Phillip B Rawlins, Jessie Hao-Ru Hsu, Daniel H O' Donovan, Alexandra Borodovsky, Peng Wang, Sharan K Bagal, Shaun M Fillery, Peter Barton, Clare Gregson, Beth Williamson, Samuel C Nash, Andrew Pike, Jon A Read, Kurt Gordon Pike, Andrew Bloecher, Erin Code, Minhui Shen, Sameer Kawatkar, Youfeng Nai, Jia Tang, Chengzhi Li, James C. Robinson
المصدر: Journal of Medicinal Chemistry. 64:17146-17183
مصطلحات موضوعية: Methyltransferase, Protein subunit, Allosteric regulation, macromolecular substances, Ligands, Cell Line, Structure-Activity Relationship, Allosteric Regulation, Heterocyclic Compounds, Catalytic Domain, Drug Discovery, Animals, Humans, Enhancer of Zeste Homolog 2 Protein, Enzyme Inhibitors, Enhancer, Cell Proliferation, biology, Chemistry, EZH2, Polycomb Repressive Complex 2, Small molecule, Rats, Histone methyltransferase, biology.protein, Cancer research, Molecular Medicine, PRC2
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المؤلفون: Qibin, Su, Erica, Banks, Geraldine, Bebernitz, Kirsten, Bell, Cassandra F, Borenstein, Huawei, Chen, Claudio E, Chuaqui, Nanhua, Deng, Andrew D, Ferguson, Sameer, Kawatkar, Neil P, Grimster, Linette, Ruston, Paul D, Lyne, Jon A, Read, Xianyou, Peng, Xiaohui, Pei, Stephen, Fawell, Zhanlei, Tang, Scott, Throner, Melissa M, Vasbinder, Haoyu, Wang, Jon, Winter-Holt, Richard, Woessner, Allan, Wu, Wenzhan, Yang, Michael, Zinda, Jason G, Kettle
المصدر: Journal of medicinal chemistry. 63(9)
مصطلحات موضوعية: Acrylamides, Aniline Compounds, Indoles, Molecular Structure, Mice, Nude, Drug Synergism, Janus Kinase 1, Xenograft Model Antitumor Assays, ErbB Receptors, Structure-Activity Relationship, Cell Line, Tumor, Drug Design, Drug Discovery, Animals, Humans, Female, Drug Screening Assays, Antitumor, Protein Kinase Inhibitors