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1دورية أكاديمية
المؤلفون: Ricardo A García, Debra J Search, John A Lupisella, Jacek Ostrowski, Bo Guan, Jian Chen, Wen-Pin Yang, Amy Truong, Aiqing He, Rongan Zhang, Mujing Yan, Samuel E Hellings, Peter S Gargalovic, Carol S Ryan, Linda M Watson, Robert A Langish, Petia A Shipkova, Nancy L Carson, Joseph R Taylor, Richard Yang, George C Psaltis, Thomas W Harrity, Jeffrey A Robl, David A Gordon
المصدر: PLoS ONE, Vol 8, Iss 2, p e53192 (2013)
وصف الملف: electronic resource
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2
المؤلفون: Yan Shi, Ying Wang, Wei Meng, Robert P. Brigance, Denis E. Ryono, Scott Bolton, Hao Zhang, Sean Chen, Rebecca Smirk, Shiwei Tao, Joseph A. Tino, Kristin N. Williams, Richard Sulsky, Laura Nielsen, Bruce Ellsworth, Michael K. Y. Wong, Jung-Hui Sun, Leslie W. Leith, Dawn Sun, Dauh-Rurng Wu, Anuradha Gupta, Richard Rampulla, Arvind Mathur, Bang-Chi Chen, Aiying Wang, Helen G. Fuentes-Catanio, Lori Kunselman, Michael Cap, Jacob Zalaznick, Xiaohui Ma, Heng Liu, Joseph R. Taylor, Rachel Zebo, Beverly Jones, Stephen Kalinowski, Joann Swartz, Ada Staal, Kevin O’Malley, Lisa Kopcho, Jodi K. Muckelbauer, Stanley R. Krystek, Steven A. Spronk, Jovita Marcinkeviciene, Gerry Everlof, Xue-Qing Chen, Carrie Xu, Yi-Xin Li, Robert A. Langish, Yanou Yang, Qi Wang, Kamelia Behnia, Aberra Fura, Evan B. Janovitz, Nicola Pannacciulli, Steven Griffen, Bradley A. Zinker, John Krupinski, Mark Kirby, Jean Whaley, Robert Zahler, Joel C. Barrish, Jeffrey A. Robl, Peter T. W. Cheng
المصدر: Journal of Medicinal Chemistry. 65:4291-4317
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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3
المؤلفون: Brian J. Murphy, Daniel Smith, Julia Sapuppo, Giridhar S. Tirucherai, Lawrence J. Kennedy, Ching-Hsuen Chu, Anthony V. Azzara, Shiwei Tao, Glenn D. Rosen, Subramaniam Krishnananthan, Jun Li, Victor R. Guarino, Lisa Burns, Joseph R. Taylor, Milinda Ziegler, Lakshmi Sivaraman, Bruce A. Ellsworth, Selvakumar Kumaravel, Hao Zhang, Tao Wang, Jun Shi, Atsu Apedo, Dhanusu Suresh, Kathy Mosure, Gerry Everlof, David A. Gordon, Lisa Zhang, Michael Gill, Chen-Pin Hung, Jianqing Li, Peter T. W. Cheng, Robert F. Kaltenbach, Sutjano Jusuf, Ying Wang, Stephanie Boehm, Mary Ellen Cvijic, Matthew G. Soars, Chi Shing Sum, Yan Shi, Jeffrey A. Robl, Reddigunta Ramesh Babu, Bradley A. Zinker, Yanou Yang, Stephen S. Kalinowski, Carrie Xu, Steven J. Walker, Sarah C. Traeger, Rebekah Heiry, Kimberley A. Lentz, Qian Ruan
المصدر: Journal of Medicinal Chemistry. 64:15549-15581
مصطلحات موضوعية: Clinical trial, Pharmacokinetics, In vivo, Chemistry, Drug Discovery, Antagonist, Molecular Medicine, Phases of clinical research, Distribution (pharmacology), Pharmacology, In vitro, ADME
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4
المؤلفون: Carl G. Jones, Vikash Tatayah, Ken Norris, Caroline M. Wainwright, Malcolm A. C. Nicoll, Emily Black, Joseph R. Taylor, Pier Luigi Vidale
المصدر: Climatic Change. 164
مصطلحات موضوعية: 0106 biological sciences, Atmospheric Science, Global and Planetary Change, education.field_of_study, Phenotypic plasticity, Extinction, 010504 meteorology & atmospheric sciences, Phenology, Ecology, Population, Climate change, Biology, 010603 evolutionary biology, 01 natural sciences, Population bottleneck, Temperate climate, Adaptation, education, 0105 earth and related environmental sciences
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المؤلفون: Michael Gill, Matt Soars, Robert F. Kaltenbach, Mosure Kathy, Peter T. W. Cheng, Anthony V. Azzara, Stephen S. Kalinowski, Shiwei Tao, Chen-Pin Hung, Larry Kennedy, Yan Shi, Lisa Burns, Julia Sapuppo, Tao Wang, David A. Gordon, Roble Jeffrey, Cvijic Mary-Ellen, Hao Zhang, Ching-Hsuen Chu, Reddigunta Ramesh Babu, Jun Shi, Bruce A. Ellsworth, Jun Li, Bradley A. Zinker, Brian J. Murphy, Dhanusu Suresh, Joseph R. Taylor, Ying Wang, Chi-Shing Sum, Ziegler Milinda, Rebekah Heiry, Steve Walker, Stephanie Boehm
المصدر: Idiopathic interstitial pneumonias.
مصطلحات موضوعية: Lung, business.industry, Antagonist, Pharmacology, Bleomycin, medicine.disease, Pathogenesis, 03 medical and health sciences, FEV1/FVC ratio, chemistry.chemical_compound, Idiopathic pulmonary fibrosis, 0302 clinical medicine, medicine.anatomical_structure, 030228 respiratory system, chemistry, In vivo, Lysophosphatidic acid, Medicine, 030212 general & internal medicine, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::8b54aea41cff0b233b97a0c88ca4d9ae
https://doi.org/10.1183/13993003.congress-2019.pa5383 -
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المؤلفون: Paul E. Morin, Haixia Wang, Lawrence J. Kennedy, Stephen P. O'connor, James J. Li, Akbar Nayeem, Vidhyashankar Ramamurthy, Steven Sheriff, Nathan Morgan, Steven J. Walker, Xiang-Yang Ye, Frederick Moulin, Brad D. Maxwell, Thomas Harrity, Jeffrey A. Robl, Stephanie Y. Chen, Timothy W. Harper, Rachel Zebo, Jun Li, Zhenqiu Hong, Shung Wu, Mengmeng Wang, Randolph P. Ponticiello, David A. Gordon, Rajasree Golla, Ramakrishna Seethala, Daniel M. Camac, Joseph R. Taylor, David S. Yoon
مصطلحات موضوعية: 0301 basic medicine, biology, Chemistry, Organic Chemistry, Adipose tissue, Dehydrogenase, Pharmacology, Biochemistry, Bioavailability, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Pharmacokinetics, 11β-hydroxysteroid dehydrogenase type 1, 030220 oncology & carcinogenesis, Pharmacodynamics, Drug Discovery, biology.protein, IC50, Ex vivo
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::537bf023154f9aff48423a9bc7df61b2
https://europepmc.org/articles/PMC6295842/ -
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المؤلفون: Steven J. Walker, Vidyhashankar Ramamurthy, Jun Li, Shung Wu, David K. Leahy, John D. Dimarco, Brad D. Maxwell, Daniel M. Camac, Joseph R. Taylor, Akbar Nayeem, Zhiwei Guo, James J. Li, Xiang-Yang Ye, Frederick Moulin, Paul E. Morin, Stepen P O’Connor, Haixia Wang, Jeffrey A. Robl, Rachel Zebo, Mark S. Kirby, Thomas Harrity, Joel C. Barrish, Timothy W. Harper, Lawrence L Kennedy, Rajasree Golla, Atsu Apedo, Bogdan Sleczka, Yi-Xin Li, David S. Yoon, Bin He, Steven Sheriff, Ramakrishna Seethala, Nathan Morgan, Mengmeng Wang, Randolph P. Ponticiello, Raymond P. Scaringe, Stephanie Y. Chen, Jianqing Li, Zhenqiu Hong, Ronald L. Hanson, David A. Gordon
المصدر: Journal of medicinal chemistry. 60(12)
مصطلحات موضوعية: 0301 basic medicine, Male, Hypothalamo-Hypophyseal System, Administration, Oral, Biological Availability, Mice, Obese, Dehydrogenase, Adamantane, Pharmacology, Crystallography, X-Ray, 03 medical and health sciences, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, Dogs, Pharmacokinetics, 11β-hydroxysteroid dehydrogenase type 1, Drug Discovery, 11-beta-Hydroxysteroid Dehydrogenase Type 1, Animals, Humans, Enzyme Inhibitors, IC50, ED50, ADME, chemistry.chemical_classification, biology, Chemistry, Actins, Rats, Macaca fascicularis, 030104 developmental biology, Enzyme, biology.protein, Molecular Medicine, Azetidines, Female, Acetamide, Half-Life
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المؤلفون: Ramakrishna Seethala, Steven J. Walker, Jun Li, Stephen P. O'connor, Lawrence J. Kennedy, Steven Sheriff, Rachel Zebo, Daniel M. Camac, Paul E. Morin, Jeffrey A. Robl, Joseph R. Taylor, James J. Li, Haixia Wang, Thomas Harrity, David A. Gordon, Akbar Nayeem, Timothy W. Harper, Zhenqiu Hong, Mengmeng Wang, Randolph P. Ponticiello, Rajasree Golla, Nathan Morgan
المصدر: ACS Medicinal Chemistry Letters. 5:803-808
مصطلحات موضوعية: chemistry.chemical_classification, Pregnane X receptor, Stereochemistry, Organic Chemistry, Pregnane, Biology, Biochemistry, chemistry.chemical_compound, Transactivation, Enzyme, chemistry, 11β-hydroxysteroid dehydrogenase type 1, Drug Discovery, Pyridine, biology.protein, Receptor, Alkyl
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9
المؤلفون: Claudio Mapelli, Ramakrishna Seethala, Songping Han, Ellen Sieber-McMaster, William R. Ewing, Ashish Khanna, Keith L. Constantine, Douglas James Riexinger, Daniel Longhi, John Krupinski, Zhengping Ma, Constance Smith-Monroy, Bastos Margarita M, Dan Shi, Michael S. Bernatowicz, Joseph R. Taylor, Christine Huang, Rajasree Golla, Gordon William Robinson, Jelka Pluscec, Jean M. Whaley, Sesha Natarajan, Jean-Philippe Meyer, Robert H. Stoffel, Li Xin, Ving G. Lee, Barry Koplowitz, Cecilia L Chi, Ildiko Antal-Zimanyi
المصدر: Journal of Medicinal Chemistry. 52:7788-7799
مصطلحات موضوعية: Male, Models, Molecular, endocrine system, Protein Conformation, Molecular Sequence Data, Peptide, CHO Cells, Glucagon-Like Peptide-1 Receptor, Mice, chemistry.chemical_compound, Cricetulus, Dogs, Cricetinae, Drug Discovery, Receptors, Glucagon, Peptide synthesis, Animals, Humans, Hypoglycemic Agents, Glucose homeostasis, Amino Acid Sequence, Receptor, Peptide sequence, Glucagon-like peptide 1 receptor, chemistry.chemical_classification, Dipeptide, Dose-Response Relationship, Drug, digestive, oral, and skin physiology, Amino acid, chemistry, Biochemistry, Molecular Medicine, Oligopeptides
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10Dapagliflozin, a Selective SGLT2 Inhibitor, Improves Glucose Homeostasis in Normal and Diabetic Rats
المؤلفون: John R. Wetterau, Deborah Hagan, William N. Washburn, Wei Meng, Joseph R. Taylor, Songping Han, Scott A. Biller, Jean M. Whaley, Li Xin
المصدر: Diabetes. 57:1723-1729
مصطلحات موضوعية: Blood Glucose, medicine.medical_specialty, Endocrinology, Diabetes and Metabolism, Carbohydrate metabolism, Sodium-Glucose Transport Proteins, Cell Line, chemistry.chemical_compound, Sodium-Glucose Transporter 1, Glucosides, Sodium-Glucose Transporter 2, Reference Values, Internal medicine, Diabetes mellitus, Adipocytes, Internal Medicine, Animals, Humans, Medicine, Glucose homeostasis, Benzhydryl Compounds, Cloning, Molecular, Dapagliflozin, Sodium-Glucose Transporter 2 Inhibitors, business.industry, Glucose transporter, Glucose analog, medicine.disease, Rats, Rats, Zucker, Renal glucose reabsorption, Glucose, Endocrinology, chemistry, SGLT2 Inhibitor, business