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1
المؤلفون: Dennis A. Holt, Gatto Gregory J, Joanne Philp, Sharon Sweitzer, Marlys Hammond, Guofeng Zhang, Mui Cheung, Rachel D. Totoritis, Lisa M. Shewchuk, Liping Wang, Huizhen Zhao, Benjamin Schwartz, Joshua E. Cottom, Harvey E. Fries, Brian G. Lawhorn, Hu Li, Alan P. Graves, Hongwei Qi, Yongdong Zhao, Lara S. Kallander, Christopher Louer
المصدر: Journal of Medicinal Chemistry. 58:7431-7448
مصطلحات موضوعية: Male, Purine, Protein Conformation, Administration, Oral, Protein Serine-Threonine Kinases, Crystallography, X-Ray, Cell Line, Rats, Sprague-Dawley, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, Troponin I, Animals, Humans, Structure–activity relationship, Purine metabolism, Sulfonamides, MAP kinase kinase kinase, Kinase, MAP Kinase Kinase Kinases, In vitro, chemistry, Biochemistry, Purines, Molecular Medicine, Protein Binding
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2
المؤلفون: James J. Foley, John G. Emery, Nicholas J. Laping, Jeffrey M. Axten, Miriam Burman, Jeffrey Guss, Demartino Michael P, Joshua E. Cottom, Sanjay Kumar, Allen Oliff, Mui Cheung
مصطلحات موضوعية: 0301 basic medicine, Chemotherapy, Innate immune system, Cyclophosphamide, Immunobiology and Immunotherapy, business.industry, medicine.medical_treatment, Lipopeptide, Hematology, Granulocyte, Pharmacology, Neutropenia, medicine.disease, Peripheral blood mononuclear cell, 03 medical and health sciences, TLR2, chemistry.chemical_compound, 030104 developmental biology, medicine.anatomical_structure, chemistry, medicine, business, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9418230308829ed6c3c1b3795a98ece6
https://europepmc.org/articles/PMC5728636/ -
3
المؤلفون: Charles William Mann, Lloyd M. Garrick, Matthew D. Vera, Linda Shanno, Jeffrey C. Pelletier, John F. Rogers, Diane B. Hauze, Jay E. Wrobel, Daniel M. Green, Irene Feingold, Murty Chengalvala, John F. Mehlmann, Joseph T. Lundquist, Joshua E. Cottom
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:2512-2515
مصطلحات موضوعية: Male, medicine.medical_specialty, Benzimidazole, medicine.drug_class, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Gonadotropin-releasing hormone, Pharmacology, Biochemistry, Piperazines, Gonadotropin-releasing hormone antagonist, Rats, Sprague-Dawley, chemistry.chemical_compound, Heterocyclic Compounds, Internal medicine, Drug Discovery, medicine, Animals, Humans, Receptor, Molecular Biology, Cells, Cultured, G protein-coupled receptor, Chemistry, Organic Chemistry, Biological activity, In vitro, Rats, Endocrinology, Molecular Medicine, Antagonism, Receptors, LHRH, Half-Life
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4
المؤلفون: Lloyd M. Garrick, John F. Mehlmann, Diane B. Hauze, Joshua E. Cottom, Daniel M. Green, Jeffrey C. Pelletier, Murty Chengalvala, Irene Feingold, Joseph T. Lundquist, John F. Rogers, Charles William Mann, Linda Shanno, Jay E. Wrobel, Christine Huselton, Wenling Kao, Kees Kenneth L
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:1986-1990
مصطلحات موضوعية: medicine.medical_specialty, Benzimidazole, Time Factors, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Gonadotropin-releasing hormone, Peptide hormone, Biochemistry, Piperazines, Structure-Activity Relationship, chemistry.chemical_compound, Heterocyclic Compounds, Oral administration, Internal medicine, Drug Discovery, medicine, Animals, Receptor, Molecular Biology, Volume of distribution, Chemistry, Organic Chemistry, Antagonist, Luteinizing Hormone, Rats, Bioavailability, Endocrinology, Models, Animal, Molecular Medicine, Benzimidazoles, Receptors, LHRH
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5
المؤلفون: William R. Adams, Irene Feingold, John F. Mehlmann, Cesario O Tio, Joshua E. Cottom, Jay E. Wrobel, Jeffrey C. Pelletier, Daniel M. Green, John F. Rogers, James W. Jetter, Murty Chengalvala, Joseph T. Lundquist, Charles William Mann, Linda Shanno, Ronald L. Magolda, Diane B. Hauze, Gregory S. Kopf, Christine Huselton
المصدر: Journal of Medicinal Chemistry. 52:2148-2152
مصطلحات موضوعية: Male, Stereochemistry, Administration, Oral, Biological Availability, In Vitro Techniques, Binding, Competitive, Chemical synthesis, Radioligand Assay, Structure-Activity Relationship, chemistry.chemical_compound, Quinoxaline, Oral administration, Quinoxalines, Drug Discovery, Animals, Humans, Structure–activity relationship, Receptor, Antagonist, Luteinizing Hormone, Rats, chemistry, Pituitary Gland, Microsomes, Liver, Molecular Medicine, Benzimidazoles, Pharmacophore, Orchiectomy, Receptors, LHRH, Gonadotropin-releasing hormone receptor, Half-Life
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6
المؤلفون: Joshua E. Cottom, Murty V. Chengalvala, Linda Shanno, Gregory S. Kopf
المصدر: Drug Design Reviews - Online. 2:35-46
مصطلحات موضوعية: Drug, Drug discovery, business.industry, media_common.quotation_subject, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Medicine, Computational biology, business, media_common
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::d40760d1dafbdee9c46e045491f49fe0
https://doi.org/10.2174/1567269053390301 -
7
المؤلفون: Daniel W. CARR, Richard E. CUTLER, Joshua E. COTTOM, Lisa M. SALVADOR, Iain D. C. FRASER, John D. SCOTT, Mary HUNZICKER-DUNN
المصدر: Biochemical Journal. 344:613-623
مصطلحات موضوعية: endocrine system, Cell Biology, Molecular Biology, Biochemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::8f2ca078b8192c09c230e49ee62009b9
https://doi.org/10.1042/bj3440613 -
8
المؤلفون: Joshua E. Cottom, Edwin H. Meade, Gregory S. Kopf, William H. Hoffman, Murty V. Chengalvala, Linda Shanno, May M. Wu, Emily S. Shen
المصدر: Current Pharmaceutical Design. 12
مصطلحات موضوعية: Infertility, medicine.drug_class, media_common.quotation_subject, Transgenic technology, Population, Fertility, Bioinformatics, Drug Delivery Systems, Drug Discovery, Contraceptive Agents, Female, Humans, Medicine, education, media_common, Pharmacology, education.field_of_study, business.industry, medicine.disease, Contraceptives, Oral, Combined, Safety profile, Estrogen, Family planning, Immunology, Female, Identification (biology), business, Infertility, Female
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9دورية أكاديمية
المؤلفون: Jeffrey C. Pelletier, Murty V. Chengalvala, Joshua E. Cottom, Irene B. Feingold, Daniel M. Green, Diane B. Hauze, Christine A. Huselton, James W. Jetter, Gregory S. Kopf, Joseph T. Lundquist, Ronald L. Magolda, Charles W. Mann, John F. Mehlmann, John F. Rogers, Linda K. Shanno, William R. Adams, Cesario O. Tio, Jay E. Wrobel
المصدر: Journal of Medicinal Chemistry; Apr2009, Vol. 52 Issue 7, p2148-2152, 5p