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المؤلفون: Ronnie Maharaj, Cristina C. Clement, Weilin Sun, Yanlong Kang, Malgorzata Kokoszka, Gabriela Chiosis, Kamalika Moulick, Wenjie Luo, Joungnam Kim, Anna Rodina, Julia Aguirre, James H. Ahn, Danuta Zatorska, Jeffrey L. Brodsky
المصدر: ASSAY and Drug Development Technologies. 9:236-246
مصطلحات موضوعية: Breast Neoplasms, Biology, Gene Expression Regulation, Enzymologic, Neuroblastoma, Downregulation and upregulation, Cell Line, Tumor, Drug Discovery, medicine, Humans, HSP70 Heat-Shock Proteins, Immunoassay, Neurons, Regulation of gene expression, medicine.diagnostic_test, Original Articles, Molecular biology, Small molecule, Up-Regulation, Cell biology, Hsp70, Cell culture, Apoptosis, Drug Design, Cancer cell, Molecular Medicine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::64e8a5191cd335efa90c2a8c33209828
https://doi.org/10.1089/adt.2010.0327 -
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المؤلفون: Julia Aguirre, Gabriela Chiosis, Anna Rodina, Kamalika Moulick, Nian Wu, Joungnam Kim, Sophorn Chip, Wenjie Luo, Qi Zhao, Fei Dou, Paul Greengard
المصدر: Proceedings of the National Academy of Sciences. 104:9511-9516
مصطلحات موضوعية: Proteasome Endopeptidase Complex, Tau protein, tau Proteins, Plasma protein binding, Heat shock protein, Chlorocebus aethiops, medicine, Animals, Humans, HSP90 Heat-Shock Proteins, Phosphorylation, Protein kinase A, Multidisciplinary, biology, Phosphotransferases, Neurodegeneration, Biological Sciences, medicine.disease, Hsp90, Rats, Cell biology, Phenotype, Tauopathies, Biochemistry, Chaperone (protein), COS Cells, Mutation, biology.protein, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::91af643b3d74ae9eb8b9f17dfae5d546
https://doi.org/10.1073/pnas.0701055104 -
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المؤلفون: Laura Llauger, Julia Aguirre, Nian Wu, Gabriela Chiosis, Joungnam Kim, Huazhong He, R.M. Immormino, Danuta Zatorska, Daniel T. Gewirth, Yuhong She
المصدر: Journal of Medicinal Chemistry. 49:381-390
مصطلحات موضوعية: Purine, Molecular Structure, biology, Chemistry, Water, Hsp90, In vitro, Structure-Activity Relationship, chemistry.chemical_compound, Solubility, Biochemistry, Purines, Cell Line, Tumor, Chaperone (protein), Heat shock protein, Drug Discovery, Cancer cell, biology.protein, Humans, Molecular Medicine, Structure–activity relationship, HSP90 Heat-Shock Proteins, Drug Screening Assays, Antitumor, Signal transduction, Cell Proliferation
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المؤلفون: Gabriela Chiosis, Neal Rosen, Julia Aguirre, Joungnam Kim, Peter Davies, Laura Llauger, Huazhong He, Ulf Peters
المصدر: Journal of Medicinal Chemistry. 48:2892-2905
مصطلحات موضوعية: Purine, Antineoplastic Agents, Binding, Competitive, Cell Line, Hsp90 inhibitor, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Cell Line, Tumor, Heat shock protein, Drug Discovery, Animals, Humans, Structure–activity relationship, HSP90 Heat-Shock Proteins, Sulfones, Sulfonyl, chemistry.chemical_classification, biology, Adenine, Hsp90, chemistry, Biochemistry, Sulfoxides, Chaperone (protein), Cancer cell, biology.protein, Molecular Medicine, Drug Screening Assays, Antitumor
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المؤلفون: Gabriela Chiosis, Joungnam Kim, Ramasamy Paulmurugan, Sanjiv S. Gambhir, Olivier Gheysens, Carmel T. Chan
مصطلحات موضوعية: Cancer Research, congenital, hereditary, and neonatal diseases and abnormalities, Lactams, Macrocyclic, Alpha (ethology), Antineoplastic Agents, Biology, Article, Hsp90 inhibitor, chemistry.chemical_compound, Mice, Genes, Reporter, Heat shock protein, Cell Line, Tumor, Protein Interaction Mapping, polycyclic compounds, Benzoquinones, Bioluminescence imaging, Animals, Humans, Benzodioxoles, HSP90 Heat-Shock Proteins, skin and connective tissue diseases, Luciferases, Renilla, Prostaglandin-E Synthases, Reporter gene, Geldanamycin, Phosphoproteins, Hsp90, Molecular biology, Xenograft Model Antitumor Assays, Oncology, chemistry, Cell culture, Purines, Mutation, biology.protein, Drug Screening Assays, Antitumor, Molecular Chaperones
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7df9ebb3c8a6e631da1fb40eb21e1c02
https://europepmc.org/articles/PMC4146344/ -
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المؤلفون: Xuejun Jiang, Gabriela Chiosis, Cristina C. Clement, Yanlong Kang, Anna Rodina, Jeffrey L. Brodsky, Nian Wu, Joan Massagué, Peter Wipf, Maria Vilenchik, Yuhong She, Kamalika Moulick, Geoffrey W. Krystal, Anne C. Chiang, Joungnam Kim, Sara J. Felts, Julia Aguirre, Julie Litz
المصدر: Nature chemical biology. 3(8)
مصطلحات موضوعية: Lung Neoplasms, Time Factors, Antineoplastic Agents, Apoptosis, Inhibitor of apoptosis, Malignant transformation, Phosphatidylinositol 3-Kinases, Heat shock protein, Cell Line, Tumor, Humans, HSP90 Heat-Shock Proteins, Carcinoma, Small Cell, Molecular Biology, Inhibitor of apoptosis domain, biology, Dose-Response Relationship, Drug, Cell Biology, Hsp90, Cell biology, Gene Expression Regulation, Neoplastic, Cell Transformation, Neoplastic, Models, Chemical, Chaperone (protein), Drug Design, biology.protein, Signal transduction, Drug Screening Assays, Antitumor
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المؤلفون: Cristina C. Clement, Yanlong Kang, Kamalika Moulick, Joungnam Kim, Sara J. Felts, Julia Aguirre, Gabriela Chiosis
المصدر: Bioorganicmedicinal chemistry letters. 16(17)
مصطلحات موضوعية: Stereochemistry, Lactams, Macrocyclic, Clinical Biochemistry, Pharmaceutical Science, Color, Fluorescence Polarization, Photochemistry, Ligands, Biochemistry, Chemical synthesis, Drug Discovery, Benzoquinones, HSP90 Heat-Shock Proteins, Laser-induced fluorescence, Molecular Biology, Fluorescent Dyes, Molecular Structure, Chemistry, Organic Chemistry, Carbocyanines, Resonance fluorescence, Rifabutin, Organic dye, Molecular Medicine, Fluorescence cross-correlation spectroscopy, Fluorescence anisotropy
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المؤلفون: Maria Vilenchik, Gabriela Chiosis, David B. Solit, Joungnam Kim
المصدر: Drug discovery today. 9(20)
مصطلحات موضوعية: Pharmacology, biology, Drug discovery, HSP90 Heat-Shock Proteins, Antineoplastic Agents, Apoptosis, Hsp90, Cancer treatment, Cell biology, Biochemistry, Pharmaceutical technology, Chaperone (protein), Neoplasms, Drug Discovery, biology.protein, Animals, Humans, Chaperone activity