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1CP-154,526: a potent and selective nonpeptide antagonist of corticotropin releasing factor receptors
المؤلفون: J P Braselton, Michael L. Corman, Judith L. Collins, A W Schmidt, J Heym, Patricia A. Seymour, David W. Schulz, F. D. Tingley, A. Dunaiskis, S Faraci, E N Winston, Robert S. Mansbach, T Seeger, Yuhpyng L. Chen, J Sprouse
المصدر: Proceedings of the National Academy of Sciences. 93:10477-10482
مصطلحات موضوعية: Male, Reflex, Startle, endocrine system, medicine.medical_specialty, Startle response, Corticotropin-Releasing Hormone, Guinea Pigs, Context (language use), Binding, Competitive, Receptors, Corticotropin-Releasing Hormone, Cell Line, Cerebral Ventricles, Rats, Sprague-Dawley, Dogs, Adrenocorticotropic Hormone, Internal medicine, medicine, Animals, Humans, Pyrroles, Receptor, Injections, Intraventricular, Cerebral Cortex, Neurons, Multidisciplinary, medicine.diagnostic_test, Chemistry, CP-154,526, Cell Membrane, Antagonist, Corticotropin-Releasing Factor Receptor 1, Callithrix, Rats, Kinetics, Pyrimidines, Endocrinology, Acoustic Stimulation, Pituitary Gland, Locus coeruleus, Locus Coeruleus, Cyclase activity, hormones, hormone substitutes, and hormone antagonists, Adenylyl Cyclases, Research Article, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::42a0f15e8489903459ee8036cf4d276e
https://doi.org/10.1073/pnas.93.19.10477 -
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المؤلفون: G.W. Antognoli, J.T. Shirley, A. Marfat, C.F. Wright, Thomas J. Carty, Frank W. Rusek, J. W. Watson, J. Delehunt, B. A. Naclerio, James F. Eggler, J.S. Pillar, Herbert Sherman, E.G. Andrews, Francis J. Sweeney, K. W. Freiert, R. Breslow, C. J. Mularski, V. L. Cohan, C J Pazoles, Lawrence S. Melvin, L.A. Rappach, John B. Cheng, David B. Damon, Jeanene E. Tickner, Judith L. Collins, P. Reiche, Hiroko Masamune, M. P. Carta, James D. Eskra, Hada William Andrew, R. J. Chambers
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:1365-1370
مصطلحات موضوعية: LTD4 receptor, Chemistry, Organic Chemistry, Clinical Biochemistry, Drug Discovery, Antagonist, Pharmaceutical Science, Molecular Medicine, Pharmacology, Receptor, Molecular Biology, Biochemistry, First generation
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المصدر: Bioorganic & Medicinal Chemistry Letters. 2:915-918
مصطلحات موضوعية: endocrine system, medicine.medical_specialty, Chemistry, digestive, oral, and skin physiology, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Biochemistry, Non peptide, Endocrinology, Competitive antagonist, Internal medicine, Drug Discovery, medicine, Enzyme-linked receptor, Molecular Medicine, Receptor, Molecular Biology, Glucagon receptor family, Glucagon receptor, hormones, hormone substitutes, and hormone antagonists, Glucagon-like peptide 1 receptor
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المؤلفون: Sanner Mark Allen, Desai Kishor A, Celeste Johnson, Jae S. Lee, Judith L. Collins, Audrey R. Dunaiskis, W. Stephen Faraci, Cecilia C. Di Prete, Angela Trozzi, Thomas Allen Chappie, Patricia A. Seymour, Jean Morrone, David B. Duignan, Stevin H. Zorn, Mark J. Majchrzak, Jackson Elisa Rose, Fliri Anton F J
المصدر: Bioorganicmedicinal chemistry letters. 8(7)
مصطلحات موضوعية: Pyrazine, Apomorphine, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Motor Activity, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, In vivo, Dopamine, Drug Discovery, medicine, Animals, Receptor, Molecular Biology, Molecular Structure, Chemistry, Organic Chemistry, Receptors, Dopamine D4, Antagonist, Receptor antagonist, In vitro, Rats, Dopamine D2 Receptor Antagonists, Pyrimidines, Drug Design, Pyrazines, Molecular Medicine, Dopamine Antagonists, Haloperidol, Indicators and Reagents, medicine.drug
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المؤلفون: Faraci Ws, Brooks E, Robert S. Mansbach, Anne W. Schmidt, Randall James Gallaschun, A. Dunaiskis, David W. Schulz, Michael L. Corman, Yuhpyng L. Chen, Winter Sm, Judith L. Collins
المصدر: Journal of medicinal chemistry. 40(11)
مصطلحات موضوعية: Male, medicine.medical_specialty, Reflex, Startle, medicine.drug_class, Chemical synthesis, Receptors, Corticotropin-Releasing Hormone, Rats, Sprague-Dawley, Structure-Activity Relationship, In vivo, Oral administration, Internal medicine, Drug Discovery, medicine, Structure–activity relationship, Animals, Pyrroles, Bicyclic molecule, Molecular Structure, Chemistry, Antagonist, Fear, Receptor antagonist, Startle reaction, Rats, Endocrinology, Pyrimidines, Anti-Anxiety Agents, Molecular Medicine