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1
المؤلفون: Strang Ross Sinclair, Markus Streiff, Daniel J. McKay, Johannes Ottl, Andreas Billich, Claudia Betschart, Stephanie Harlfinger, Eloísa Jiménez-Núñez, Nigel Graham Cooke, Christine Guntermann, Markus Voegtle, Janet Dawson, Samuel Hintermann, Klemens Kaupmann, Rowan Stringer, Christian Beerli, Nathalie Gobeau, Juergen Wagner, Klemens Hoegenauer, Joerg Kallen, Peter Ertl
المصدر: Journal of Medicinal Chemistry. 62:10816-10832
مصطلحات موضوعية: chemistry.chemical_classification, Orphan receptor, 0303 health sciences, Chemistry, Carboxylic acid, Retinoic acid, 01 natural sciences, Combinatorial chemistry, 0104 chemical sciences, Proinflammatory cytokine, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, In vivo, Lipophilic efficiency, RAR-related orphan receptor gamma, Drug Discovery, Molecular Medicine, 030304 developmental biology, ADME
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2
المؤلفون: Klemens, Hoegenauer, Joerg, Kallen, Eloísa, Jiménez-Núñez, Ross, Strang, Peter, Ertl, Nigel G, Cooke, Samuel, Hintermann, Markus, Voegtle, Claudia, Betschart, Daniel J J, McKay, Juergen, Wagner, Johannes, Ottl, Christian, Beerli, Andreas, Billich, Janet, Dawson, Klemens, Kaupmann, Markus, Streiff, Nathalie, Gobeau, Stephanie, Harlfinger, Rowan, Stringer, Christine, Guntermann
المصدر: Journal of medicinal chemistry. 62(23)
مصطلحات موضوعية: Male, Models, Molecular, Dose-Response Relationship, Drug, Molecular Structure, Imidazoles, Administration, Oral, Nuclear Receptor Subfamily 1, Group F, Member 3, Rats, Drug Design, Fluorescence Resonance Energy Transfer, Animals, Female, Hypersensitivity, Delayed, Half-Life
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3
المؤلفون: Christine Guntermann, Janet Dawson, Anna Vulpetti, Andreas Billich, Rowan Stringer, Johannes Ottl, Samuel Hintermann, Henri Mattes, Eric Vangrevelinghe, Nigel Graham Cooke, Klemens Kaupmann, Romain M. Wolf, Juergen Wagner, Klemens Hoegenauer, Joerg Kallen, David Orain, David Carcache
المصدر: Journal of Medicinal Chemistry. 61:6724-6735
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Drug Inverse Agonism, Inflammation, 01 natural sciences, 03 medical and health sciences, Transcription (biology), In vivo, RAR-related orphan receptor gamma, Catalytic Domain, Drug Discovery, medicine, Animals, Inverse agonist, Transcription factor, 010405 organic chemistry, Drug discovery, Chemistry, Nuclear Receptor Subfamily 1, Group F, Member 3, Rats, 0104 chemical sciences, Cell biology, Disease Models, Animal, 030104 developmental biology, Molecular Medicine, Female, medicine.symptom
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4كتاب إلكتروني
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5
المؤلفون: Christine Guntermann, Juergen Wagner, David Orain, Andreas Billich, Joerg Kallen, Samuel Hintermann, Janet Dawson, Rowan Stringer, Henri Mattes, Klemens Kaupmann, David Carcache, Anna Vulpetti
المصدر: ChemMedChem. 11:2640-2648
مصطلحات موضوعية: 0301 basic medicine, Imidazopyridine, Drug Inverse Agonism, Pyridines, Receptors, Retinoic Acid, Stereochemistry, medicine.medical_treatment, Plasma protein binding, Pharmacology, Crystallography, X-Ray, Biochemistry, Inhibitory Concentration 50, 03 medical and health sciences, Pharmacokinetics, RAR-related orphan receptor gamma, Drug Discovery, medicine, Animals, Humans, Potency, Inverse agonist, General Pharmacology, Toxicology and Pharmaceutics, Transcription factor, Cells, Cultured, Binding Sites, Molecular Structure, Chemistry, Interleukin-17, Organic Chemistry, Imidazoles, Nuclear Receptor Subfamily 1, Group F, Member 3, Triazoles, Rats, 030104 developmental biology, Cytokine, Molecular Medicine, Protein Binding
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6
المؤلفون: Thomas Kilger, Juergen Wagner, Dominic Maier, Thomas Fischer, Ulf Bartl, Stephan Helbig, Johannes Lodermeyer, Ulrich Krumbein, Waechter Claus, Franz-Xaver Muehlbauer, A. Dehe, Alfred Sigl, Horst Theuss, Matthias Vobl, Bernd Goller, Matthias Herrmann, Christian Geissler
المصدر: 2019 IEEE 69th Electronic Components and Technology Conference (ECTC).
مصطلحات موضوعية: Microelectromechanical systems, Materials science, Microphone, 010401 analytical chemistry, Mechanical engineering, Fan-out, 02 engineering and technology, 021001 nanoscience & nanotechnology, 01 natural sciences, 0104 chemical sciences, Embedded Wafer Level Ball Grid Array, Wafer fabrication, Wafer, 0210 nano-technology, Wafer-level packaging, Decoupling (electronics)
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::be3ad265cbb3320d11b7363814c73c55
https://doi.org/10.1109/ectc.2019.00134 -
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المؤلفون: Juergen Wagner, Eric Vangrevelinghe, Gerhard Zenke, Maurice Van Eis, Peter von Matt, Walter Schuler, Jean-Pierre Evenou
المصدر: Bioorganicmedicinal chemistry letters. 27(4)
مصطلحات موضوعية: 0301 basic medicine, Indoles, Protein Kinase C-alpha, T-Lymphocytes, Clinical Biochemistry, Pharmaceutical Science, Naphthols, Lymphocyte Activation, Biochemistry, Maleimides, 03 medical and health sciences, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, 0302 clinical medicine, Drug Discovery, Protein Kinase C beta, Humans, Molecular Biology, Maleimide, Protein Kinase Inhibitors, Protein kinase C, B-cell activation, Cell Proliferation, B-Lymphocytes, Binding Sites, Kinase, Organic Chemistry, Protein Structure, Tertiary, Isoenzymes, Molecular Docking Simulation, 030104 developmental biology, chemistry, Molecular Medicine, Selectivity, 030215 immunology, Protein Binding
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8
المؤلفون: Thierry T. Diagana, Suresh B. Lakshminarayana, Susan Noh, Francesca Blasco, Carrie F. Brooks, Jennifer A. Zambriski, Laura B. Goodman, Gu Feng, Sumiti Vinayak, Gillian T. Herbert, Peter Gedeck, Lijun Zhang, Jayesh Tandel, Siau H. Lim, Christian G. Noble, F. Joel Leong, Alex Chao, Juergen Wagner, Bin Zou, Boris Striepen, Tracy Sy, Ravinder Reddy Kondreddi, Christophe Bodenreider, Ujjini H. Manjunatha, Ghislain M. C. Bonamy, Adam Sateriale
المصدر: Nature
مصطلحات موضوعية: 0301 basic medicine, Male, Pyridines, Cryptosporidiosis, Cryptosporidium, Communicable Diseases, Article, Microbiology, 03 medical and health sciences, Immunocompromised Host, Interferon-gamma, Mice, Cell Line, Tumor, parasitic diseases, Pyrazolopyridine, medicine, Animals, Humans, Interferon gamma, Rats, Wistar, 1-Phosphatidylinositol 4-Kinase, Mice, Knockout, Multidisciplinary, biology, Kinase, Drug discovery, business.industry, biology.organism_classification, Antiparasitic agent, Virology, 3. Good health, Rats, Disease Models, Animal, 030104 developmental biology, Cryptosporidium parvum, Animals, Newborn, Pyrazoles, Cattle, Female, business, Cryptosporidium hominis, medicine.drug
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9
المؤلفون: Chetan Pandit, Christine E. Gee, Daniel Hoyer, Vinod D. Chaudhari, Grit Laue, Juergen Wagner, Laura H. Jacobson, Dirk Behnke, Claudia Betschart, Simona Cotesta, Sangamesh Badiger, Samuel Hintermann, Markus Fendt, Silvio Ofner
المصدر: Journal of Medicinal Chemistry. 56:7590-7607
مصطلحات موضوعية: Male, Indoles, Sleep induction, Primary Insomnia, Motor Activity, Pharmacology, Doras, Non-rapid eye movement sleep, Mice, Structure-Activity Relationship, Quinoxalines, Sleep Initiation and Maintenance Disorders, mental disorders, Drug Discovery, medicine, Animals, Spiro Compounds, Sleep Stages, biology, Electromyography, Chemistry, Suvorexant, Electroencephalography, Stereoisomerism, Azepines, Triazoles, biology.organism_classification, Orexin receptor, Mice, Inbred C57BL, Pyrimidines, Molecular Medicine, Orexin Receptor Antagonists, Almorexant, Sleep, medicine.drug
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10كتاب إلكتروني
المؤلفون: Gotthard Breit, Ulf von Krause, Steffen Lehndorf, Krzysztof Malinowski, Almut Möller, Jürgen Stark, Roland Sturm, Hans-Jürgen Urban, Henrik Uterwedde, Manuel Wäschle, Jürgen Wagner, Hans-Jürgen Bieling, Johannes Varwick
نوع المادة: eBook.
تصنيفات: POLITICAL SCIENCE / Reference