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1
المؤلفون: Nicola J. Curtin, Graeme C.M. Smith, David R. Newell, Niall M.B. Martin, Pia Thommes, Andrew Slade, Keith Menear, Roger J. Griffin, Liam Cornell, Julia Bardos, Jody Barbeau, Michele Tavecchio, Celine Cano, Caroline J. Richardson, Helen Jenkins, Yan Zhao, Michael A. Batey, Joanne M. Munck
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::33c9f0d0e3e98828130b4f41f16e3e80
https://doi.org/10.1158/1535-7163.c.6535653.v1 -
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المؤلفون: Nicola J. Curtin, Graeme C.M. Smith, David R. Newell, Niall M.B. Martin, Pia Thommes, Andrew Slade, Keith Menear, Roger J. Griffin, Liam Cornell, Julia Bardos, Jody Barbeau, Michele Tavecchio, Celine Cano, Caroline J. Richardson, Helen Jenkins, Yan Zhao, Michael A. Batey, Joanne M. Munck
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3174dc79b3c750b99d9eff50af83dd73
https://doi.org/10.1158/1535-7163.22497552 -
3
المؤلفون: Nicola J. Curtin, Graeme C.M. Smith, David R. Newell, Niall M.B. Martin, Pia Thommes, Andrew Slade, Keith Menear, Roger J. Griffin, Liam Cornell, Julia Bardos, Jody Barbeau, Michele Tavecchio, Celine Cano, Caroline J. Richardson, Helen Jenkins, Yan Zhao, Michael A. Batey, Joanne M. Munck
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2593b57508ee0ef2270374929c03d884
https://doi.org/10.1158/1535-7163.22497549 -
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المؤلفون: Celine Cano, Pia Thommes, Niall M. B. Martin, Yan Zhao, Liam Cornell, Michael A. Batey, Helen Jenkins, Jody Barbeau, Keith Allan Menear, Julia Bardos, Nicola J. Curtin, Michele Tavecchio, David R. Newell, Roger J. Griffin, Caroline Richardson, Graeme C. M. Smith, Andrew Slade, Joanne M. Munck
المصدر: Molecular Cancer Therapeutics. 11:1789-1798
مصطلحات موضوعية: Cancer Research, Antineoplastic Agents, DNA-Activated Protein Kinase, Thiophenes, Article, Mice, Chemosensitization, Cell Line, Tumor, Neoplasms, medicine, Animals, Humans, Cytotoxic T cell, Enzyme Inhibitors, Cytotoxicity, Etoposide, Phosphoinositide-3 Kinase Inhibitors, biology, Chemistry, Cell growth, Topoisomerase, fungi, Xenograft Model Antitumor Assays, Molecular biology, Tumor Burden, Enzyme Activation, enzymes and coenzymes (carbohydrates), Oncology, Chromones, Drug Resistance, Neoplasm, Cell culture, Cancer cell, Immunology, MCF-7 Cells, biology.protein, Female, biological phenomena, cell phenomena, and immunity, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::79970d5d09b4bd6b730644af5e24957f
https://doi.org/10.1158/1535-7163.mct-11-0535 -
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المؤلفون: Keith Allan Menear, Ian R. Hardcastle, Edward Jolyon Griffen, M. Raymond V. Finlay, Roger J. Griffin, Kate M. Clapham, Bernard T. Golding, Celine Cano, Attilla Ting, Turner Paul, Julia Bardos, Gail L. Young
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:966-970
مصطلحات موضوعية: DNA repair, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, DNA-Activated Protein Kinase, Plasma protein binding, Biochemistry, Phosphatidylinositol 3-Kinases, Structure-Activity Relationship, chemistry.chemical_compound, Adenosine Triphosphate, Protein structure, Drug Discovery, Humans, Structure–activity relationship, Protein kinase A, Protein Kinase Inhibitors, Molecular Biology, Phosphoinositide-3 Kinase Inhibitors, Organic Chemistry, Protein Structure, Tertiary, chemistry, Chromones, Molecular Medicine, Pharmacophore, DNA, Protein Binding, Binding domain
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المؤلفون: Celine Cano, Bernard T. Golding, Sonsoles Rodriguez-Aristegui, Roger J. Griffin, Sara L. Payne, Ian R. Hardcastle, Nahida Parveen, Julia Bardos, Marcus Peacock
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:3649-3653
مصطلحات موضوعية: Stereochemistry, DNA repair, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, DNA-Activated Protein Kinase, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Adenosine Triphosphate, Coumarins, Drug Discovery, Humans, Binding site, Molecular Biology, chemistry.chemical_classification, Binding Sites, Organic Chemistry, Coumarin, Isocoumarin, Enzyme, Isocoumarins, chemistry, Chromones, Molecular Medicine, DNA, Lactone, Binding domain
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المؤلفون: Roger J. Griffin, Celine Cano, Bernard T. Golding, Attilla Ting, Mark Frigerio, Keith Allan Menear, Julia Bardos, Christopher M. Bailey, Marc Geoffrey Hummersone, Kappusamy Saravanan, Kerry Shea, Ian R. Hardcastle, Caroline Richardson, Nicola J. Curtin, Pia Thommes, Graeme C. M. Smith, David R. Newell
المصدر: Journal of medicinal chemistry. 56(16)
مصطلحات موضوعية: Chemistry, Stereochemistry, Morpholines, DNA-Activated Protein Kinase, In vitro, chemistry.chemical_compound, In vivo, Morpholine, Drug Discovery, Molecular Medicine, Moiety, Humans, Phosphatidylinositol, Protein kinase A, Cytotoxicity, Protein Kinase Inhibitors, Acetamide, HeLa Cells, Phosphoinositide-3 Kinase Inhibitors
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المؤلفون: Derek Manas, Newell, Nicola J. Curtin, Joanne M. Munck, Julia Bardos, F Budhisetiawan, Liam Cornell, Helen L. Reeves
المصدر: Hepatology. 52
مصطلحات موضوعية: chemistry.chemical_compound, Hepatology, chemistry, Cell culture, medicine, Synthetic lethality, Liver cancer, medicine.disease, Molecular biology, DNA, Double Strand Break Repair
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المؤلفون: Zora Sulekova, Julia Bardos, Wolfgang G. Ballhausen
المصدر: International journal of cancer. 73(1)
مصطلحات موضوعية: Genetics, Cancer Research, Genes, APC, biology, Adenomatous polyposis coli, Sequence analysis, Alternative splicing, Intron, Brain, Exons, Exon shuffling, Molecular biology, Polymerase Chain Reaction, Cell Line, Exon, Exon trapping, Oncology, biology.protein, Humans, Tandem exon duplication, RNA, Messenger
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المؤلفون: Faye Craven, Julia Bardos, Bernard T. Golding, Gavin Jones, Ian R. Hardcastle, Karen Haggerty, Celine Cano, Attilla Ting, Roger J. Griffin, Pia Thommes, Kate M. Clapham, Tommy Rennison
المصدر: Organic & Biomolecular Chemistry. 10:6747
مصطلحات موضوعية: Models, Molecular, Atropisomer, Binding Sites, Swine, Stereochemistry, Chemistry, Morpholines, Organic Chemistry, Stereoisomerism, Biological activity, DNA-Activated Protein Kinase, Biochemistry, Chiral column chromatography, Structure-Activity Relationship, Chromones, Animals, Humans, Structure–activity relationship, Physical and Theoretical Chemistry, Enantiomer, Pharmacophore, Protein kinase A, Protein Kinase Inhibitors
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::24b2d6f5c46d63b3169c87e4923677fa
https://doi.org/10.1039/c2ob26035b