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المؤلفون: Philip G. Humphreys, Niall A. Anderson, Paul Bamborough, Andrew Baxter, Chun-wa Chung, Rosa Cookson, Peter D. Craggs, Toryn Dalton, Julie C. L. Fournier, Laurie J. Gordon, Heather F. Gray, Matthew W. Gray, Richard Gregory, David J. Hirst, Craig Jamieson, Katherine L. Jones, Hripsimee Kessedjian, David Lugo, Grant McGonagle, Vipulkumar K. Patel, Christopher Patten, Darren L. Poole, Rab K. Prinjha, Cesar Ramirez-Molina, Inmaculada Rioja, Gail Seal, Kayleigh A. J. Stafford, Rishi R. Shah, Daniel Tape, Natalie H. Theodoulou, Laura Tomlinson, Sabri Ukuser, Ian D. Wall, Natalie Wellaway, Gemma White
المصدر: Journal of Medicinal Chemistry. 65:15174-15207
مصطلحات موضوعية: Histones, Protein Domains, Lysine, Drug Discovery, Humans, Molecular Medicine, Ligands, Transcription Factors
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المؤلفون: Sebastien Andre Campos, Gemma V. White, Francesca Zappacosta, Daniel Thomas, John P. Evans, Vipulkumar Kantibhai Patel, Nicholas C. O. Tomkinson, Julie C. L. Fournier
مصطلحات موضوعية: Class I Phosphatidylinositol 3-Kinases, Protein Conformation, Lysine, Afatinib, Biochemistry, Catalysis, Mass Spectrometry, Substrate Specificity, Acylation, Piperidines, Catalytic Domain, Humans, QD, Amino Acid Sequence, Kinase activity, Phosphoinositide-3 Kinase Inhibitors, chemistry.chemical_classification, Acrylamides, Aniline Compounds, Chemistry, Adenine, Ligand binding assay, Acetylation, General Medicine, Small molecule, Molecular Docking Simulation, Enzyme, Covalent bond, Molecular Medicine, Protein Binding
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