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المؤلفون: Nicola G. Wallis, Alison J.-A. Woolford, Nicola E. Wilsher, Neil T. Thompson, Lukas Stanczuk, Alpesh D. Shah, Caroline J. Richardson, Sharna J. Rich, David C. Rees, Michael Reader, Marc O'Reilly, David Norton, Christopher W. Murray, Sandra Muench, Vanessa Martins, John F. Lyons, Justyna Kucia-Tran, Christopher J. Hindley, Tom D. Heightman, Roberta Ferraldeschi, Charlotte East, Aurélie Courtin, Juan Castro, Jessica L. Brothwood, Luke Bevan, Valerio Berdini, Joanne M. Munck
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::45c83a97aa3dd2ed35fbdc9ef36e9bb5
https://doi.org/10.1158/1535-7163.22521489.v1 -
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المؤلفون: Nicola G. Wallis, Alison J.-A. Woolford, Nicola E. Wilsher, Neil T. Thompson, Lukas Stanczuk, Alpesh D. Shah, Caroline J. Richardson, Sharna J. Rich, David C. Rees, Michael Reader, Marc O'Reilly, David Norton, Christopher W. Murray, Sandra Muench, Vanessa Martins, John F. Lyons, Justyna Kucia-Tran, Christopher J. Hindley, Tom D. Heightman, Roberta Ferraldeschi, Charlotte East, Aurélie Courtin, Juan Castro, Jessica L. Brothwood, Luke Bevan, Valerio Berdini, Joanne M. Munck
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::185aef78c19fca4a606a8b2c178f1341
https://doi.org/10.1158/1535-7163.22521498.v1 -
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المؤلفون: Neil T. Thompson, Nicola G. Wallis, Michael Reader, Christopher J. Hindley, Juan Castro, John Lyons, David C. Rees, Nicola E. Wilsher, Caroline Richardson, Tom D. Heightman, Lukas Stanczuk, Alpesh Shah, Sharna J. Rich, Charlotte East, Valerio Berdini, Marc O'Reilly, Justyna Kucia-Tran, Jessica L. Brothwood, Joanne M. Munck, Alison Jo-Anne Woolford, Sandra Muench, Christopher William Murray, David Norton, Luke Bevan, Aurélie Courtin, Roberta Ferraldeschi, Vanessa Martins
المصدر: Molecular Cancer Therapeutics. 20:1757-1768
مصطلحات موضوعية: Male, MAPK/ERK pathway, Cancer Research, Indoles, Mice, Nude, Apoptosis, Ribosomal s6 kinase, Mice, Downregulation and upregulation, Cell Movement, In vivo, Tumor Cells, Cultured, Animals, Humans, Phosphorylation, Extracellular Signal-Regulated MAP Kinases, Protein Kinase Inhibitors, Cell Proliferation, Mice, Inbred BALB C, biology, Chemistry, Effector, Cell Cycle, Xenograft Model Antitumor Assays, In vitro, Gene Expression Regulation, Neoplastic, Pyrimidines, Oncology, Drug Resistance, Neoplasm, Cell culture, Colonic Neoplasms, Cancer research, biology.protein
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6856599564530823950e091fd6e69a67
https://doi.org/10.1158/1535-7163.mct-20-0909 -
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المؤلفون: Michael Reader, Aurélie Courtin, Steven Howard, Nicola G. Wallis, Jonathan Shannon, Hugh Walton, Christopher William Murray, Joseph E. Coyle, Joanne M. Munck, Alison Jo-Anne Woolford, Torren M. Peakman, David C. Rees, James Edward Harvey Day, Charlotte Mary Griffiths-Jones, Marc O'Reilly, Alpesh Shah, David Norton, Valerio Berdini, Lynsey Fazal, Maria Grazia Carr, Charlotte East, Tom D. Heightman, Nicola E. Wilsher, Ildiko Maria Buck, Luke Bevan, Stuart Thomas Onions, Michael Cooke, Justyna Kucia-Tran, Sandra Muench, Nick Palmer, Sharna J. Rich, Vanessa Martins, David Cousin, Puja Pathuri, John P. Watts
المصدر: Journal of medicinal chemistry. 64(16)
مصطلحات موضوعية: Male, Indoles, Antineoplastic Agents, Crystallography, X-Ray, Proto-Oncogene Mas, Rats, Sprague-Dawley, Structure-Activity Relationship, Dogs, Pharmacokinetics, Neoplasms, Drug Discovery, Animals, Humans, In patient, Tumor growth, Phosphorylation, Rats, Wistar, Protein kinase A, Protein Kinase Inhibitors, Mitogen-Activated Protein Kinase 1, Mice, Inbred BALB C, Molecular Structure, Chemistry, Kinase, Xenograft Model Antitumor Assays, Clinical trial, Pyrimidines, Cancer research, Molecular Medicine, Once daily dosing, Protein Binding
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المؤلفون: Stephen R. Wedge, Justyna Kucia-Tran, N. Ferrari, Steven Howard, Lynsey Fazal, Luke Bevan, M. Ahn, Gianni Chessari, G. Ward, E. Willmore, Juan Castro, M. Sims
المصدر: HemaSphere. 3:443-444
مصطلحات موضوعية: biology, Apoptosis, Chemistry, Wild type, biology.protein, Antagonist, Mdm2, Hematology, Small molecule, Molecular biology
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المؤلفون: John Lyons, Aurélie Courtin, Tom D. Heightman, Nicola E. Wilsher, Luke Bevan, Justyna Kucia-Tran, Sandra Muench, Birikiti Kidane, Nicola G. Wallis, Lukas Stanczuk, Alpesh Shah, Joanne M. Munck, Neil Thompson
المصدر: Cancer Research. 78:5781-5781
مصطلحات موضوعية: MAPK/ERK pathway, Cancer Research, education.field_of_study, Kinase, business.industry, Population, medicine.disease, medicine.disease_cause, respiratory tract diseases, Oncology, In vivo, Cell culture, Cancer cell, medicine, Cancer research, KRAS, Lung cancer, education, business, neoplasms
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::c67a56f2b6c67597d7decefa3a9f43b6
https://doi.org/10.1158/1538-7445.am2018-5781 -
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المؤلفون: Luke Bevan, John Lyons, Caroline Richardson, Charlotte Mary Griffiths-Jones, Juan Castro, Lukas Stanczuk, Alpesh Shah, Hugh Walton, Neil T. Thompson, Harpreet K Saini, Nicola G. Wallis, Joanne M. Munck, Alison Jo-Anne Woolford, David Norton, Tom D. Heightman, Lynsey Fazal, Christopher J. Hindley, Christopher W. Murray, Hannah Braithwaite, Mike Reader, Vanessa Martins, Charlotte East, Puja Pathuri, Birikiti Kidane, Marc O'Reilly, David C. Rees, Aurélie Courtin, Megan Cassidy, Justyna Kucia-Tran, James Edward Harvey Day, Sandra Muench, Nicola E. Wilsher, Ildiko Maria Buck, Nick Palmer, Sharna J. Rich, Valerio Berdini, Brent Graham
المصدر: Molecular Cancer Therapeutics. 17:B154-B154
مصطلحات موضوعية: MAPK/ERK pathway, Cancer Research, Cell signaling, biology, Chemistry, Receptor tyrosine kinase, Substrate-level phosphorylation, Oncology, Downregulation and upregulation, In vivo, Cell culture, biology.protein, Cancer research, Phosphorylation
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::9fb0f164a64005dde16a1115a0571fd2
https://doi.org/10.1158/1535-7163.targ-17-b154