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1Design and synthesis of a series of glycerol-derived receptor mediated calcium entry (RMCE) blockers
المؤلفون: K Cassidy, J E Merritt, Timothy J. Rink, R. E. Dolle, Trevor J. Hallam, W. P. Armstrong, K E Moores, William Howson, BK Leigh, Riccardo Novelli, A Jaxa-Chamiec, MA Tchorzewska
المصدر: European Journal of Medicinal Chemistry. 25:595-602
مصطلحات موضوعية: Pharmacology, Chemistry, Recombinase-mediated cassette exchange, Organic Chemistry, General Medicine, Receptor-mediated endocytosis, chemistry.chemical_compound, Biochemistry, Drug Discovery, Biophysics, Glycerol, Platelet, Lead compound, Calcium entry
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2
المؤلفون: S A McCarthy, J E Merritt, K E Moores, Michael P.A. Davies
المصدر: Europe PubMed Central
مصطلحات موضوعية: Blood Platelets, Fura-2, Neutrophils, Fluorescence spectrometry, chemistry.chemical_element, Digitonin, Buffers, Calcium, Biochemistry, chemistry.chemical_compound, Cytosol, Humans, Platelet, Egtazic Acid, Molecular Biology, Benzofurans, Fluorescent Dyes, Fluo-3, Aniline Compounds, Chromatography, Probenecid, Chemistry, Thrombin, Cell Biology, Fluorescence, N-Formylmethionine Leucyl-Phenylalanine, Dissociation constant, Blood, Spectrometry, Fluorescence, Xanthenes, cardiovascular system, Research Article
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f613b6c96b8a03c9d03f232955107743
https://doi.org/10.1042/bj2690513 -
3
المؤلفون: C H, MacPhee, K E, Moores, H F, Boyd, D, Dhanak, R J, Ife, C A, Leach, D S, Leake, K J, Milliner, R A, Patterson, K E, Suckling, D G, Tew, D M, Hickey
المصدر: The Biochemical journal. 338
مصطلحات موضوعية: Aryldialkylphosphatase, Esterases, Phospholipases A, Lipoproteins, LDL, Phosphatidylcholine-Sterol O-Acyltransferase, Chemotaxis, Leukocyte, Phospholipases A2, Sulfoxides, 1-Alkyl-2-acetylglycerophosphocholine Esterase, Azetidines, Humans, lipids (amino acids, peptides, and proteins), Enzyme Inhibitors, Oxidation-Reduction, Protein Binding, Research Article
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::626460f359a74e1b15f305f443280f4d
https://pubmed.ncbi.nlm.nih.gov/10024526 -
4
المؤلفون: C H, Macphee, E R, Appelbaum, K, Johanson, K E, Moores, C S, Imburgia, J, Fornwald, T, Berkhout, M, Brawner, P H, Groot, K, O'Donnell, D, O'Shannessy, G, Scott, J R, White
المصدر: Journal of immunology (Baltimore, Md. : 1950). 161(11)
مصطلحات موضوعية: Eosinophils, Chemotaxis, Leukocyte, Chemokines, CC, Chemotactic Factors, Eosinophil, Molecular Sequence Data, Humans, Protein Isoforms, Calcium, Amino Acid Sequence, Monocytes, Recombinant Proteins, Monocyte Chemoattractant Proteins
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::5f4cc6014e97c593c660b01f0e6617a5
https://pubmed.ncbi.nlm.nih.gov/9834116 -
5
المؤلفون: K E, Moores, J E, Merritt
المصدر: Eicosanoids. 4(2)
مصطلحات موضوعية: Lipoxins, N-Formylmethionine Leucyl-Phenylalanine, Cytosol, Dose-Response Relationship, Drug, Neutrophils, Hydroxyeicosatetraenoic Acids, Humans, Calcium
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::d46619fd81d8fa2c64e1c58c8b720471
https://pubmed.ncbi.nlm.nih.gov/1910866 -
6
المؤلفون: Paul J. England, Trevor J. Hallam, K E Moores, Alec W. M. Simpson, Martin L. Reeves, Joanne Maguire, Timothy J. Rink, Kenneth J. Murray
المصدر: British journal of pharmacology. 99(3)
مصطلحات موضوعية: Blood Platelets, medicine.medical_specialty, Platelet Aggregation, Platelet Function Tests, Siguazodan, Phosphodiesterase Inhibitors, chemistry.chemical_element, Calcium, In Vitro Techniques, Guanidines, chemistry.chemical_compound, Internal medicine, medicine, Cyclic AMP, Humans, Platelet, Phosphodiesterase inhibitor, Pharmacology, biology, Aspirin, Phosphodiesterase, Chromatography, Ion Exchange, Prostaglandin Endoperoxides, Synthetic, Adenosine Diphosphate, Pyridazines, Adenosine diphosphate, Endocrinology, chemistry, Enzyme inhibitor, 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid, biology.protein, Platelet aggregation inhibitor, Collagen, Platelet Aggregation Inhibitors, Research Article
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7
المؤلفون: K E Moores, J E Merritt, Michael P.A. Davies
المصدر: Biochemical Society Transactions. 17:123-123
مصطلحات موضوعية: Cytoplasmic calcium, Neutrophil adhesion, Chemistry, Stimulation, Biochemistry, Cell biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::f2c51dbaef7acc952baee23edc6b2634
https://doi.org/10.1042/bst0170123