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1دورية أكاديمية
المؤلفون: Misato Ito, Shunji Yamazaki, Kaoru Yamagami, Masako Kuno, Yoshiaki Morita, Kenji Okuma, Koji Nakamura, Noboru Chida, Masamichi Inami, Takayuki Inoue, Shohei Shirakami, Yasuyuki Higashi
المصدر: Journal of Pharmacological Sciences, Vol 133, Iss 1, Pp 25-33 (2017)
مصطلحات موضوعية: Peficitinib, ASP015K, Janus kinase, Rheumatoid arthritis, Adjuvant-induced arthritis, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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2
المؤلفون: Hidehiko Fukahori, Kaoru Yamagami, Satoshi Kubo, Yukihito Sugano, Fumie Takahashi, Ayako Moritomo, Koji Kato, Susumu Yamaki, Koji Nakamura, Koji Yokoo, Toshihiro Hamajima, Suzuki Daisuke
المصدر: Bioorganic & Medicinal Chemistry. 27:1056-1064
مصطلحات موضوعية: Gene isoform, Scaffold, Pyrrolidines, Pyrimidine, Class I Phosphatidylinositol 3-Kinases, Clinical Biochemistry, Pharmaceutical Science, 01 natural sciences, Biochemistry, chemistry.chemical_compound, In vivo, Drug Discovery, Animals, Humans, Potency, Molecular Biology, Cells, Cultured, PI3K/AKT/mTOR pathway, Phosphoinositide-3 Kinase Inhibitors, Mice, Inbred BALB C, 010405 organic chemistry, Chemistry, Organic Chemistry, Highly selective, 0104 chemical sciences, Molecular Docking Simulation, Antibody production, 010404 medicinal & biomolecular chemistry, Molecular Medicine, Female
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3
المؤلفون: Misato Ito, Kaoru Yamagami, Takanori Marui, Koji Kato, Tatsuaki Morokata, Tomoko Kawashima, Masahiko Akamatsu, Yoko Kaneko, Fumie Takahashi, Hidehiko Fukahori
المصدر: International immunopharmacology. 87
مصطلحات موضوعية: 0301 basic medicine, Class I Phosphatidylinositol 3-Kinases, T cell, T-Lymphocytes, Immunology, Lupus nephritis, Pathogenesis, 03 medical and health sciences, 0302 clinical medicine, immune system diseases, Immunology and Allergy, Medicine, Animals, skin and connective tissue diseases, Pharmacology, Autoimmune disease, B-Lymphocytes, Mice, Inbred BALB C, Systemic lupus erythematosus, Mice, Inbred NZB, business.industry, Antibody titer, Autoantibody, medicine.disease, Lupus Nephritis, Disease Models, Animal, 030104 developmental biology, medicine.anatomical_structure, Immunoglobulin M, 030220 oncology & carcinogenesis, Female, business, Nephritis
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4
المؤلفون: Koichiro Mukoyoshi, Kaoru Yamagami, Kousei Yoshihara, Koji Yokoo, Susumu Yamaki, Fumie Takahashi, Toshihiro Hamajima, Yukihito Sugano, Koji Kato, Hidehiko Fukahori, Ayako Moritomo
المصدر: Bioorganic & Medicinal Chemistry. 26:2410-2419
مصطلحات موضوعية: 0301 basic medicine, Class I Phosphatidylinositol 3-Kinases, Pyridines, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Amide, Drug Discovery, Pyrazolopyridine, Animals, Humans, Protein Kinase Inhibitors, Molecular Biology, Phosphoinositide-3 Kinase Inhibitors, Biological evaluation, Mice, Inbred BALB C, Molecular Structure, Chemistry, Organic Chemistry, Nuclear Proteins, Stereoisomerism, Molecular Docking Simulation, 030104 developmental biology, Pyrazoles, Molecular Medicine, Female, Selectivity, Transcription Factors
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5
المؤلفون: Shohei Shirakami, Kenji Okuma, Yoshiaki Morita, Takayuki Inoue, Misato Ito, Masako Kuno, Shunji Yamazaki, Masamichi Inami, Yasuyuki Higashi, Kaoru Yamagami, Noboru Chida, Koji Nakamura
المصدر: Journal of Pharmacological Sciences, Vol 133, Iss 1, Pp 25-33 (2017)
مصطلحات موضوعية: Male, Niacinamide, 0301 basic medicine, T-Lymphocytes, medicine.medical_treatment, Administration, Oral, Arthritis, Adamantane, ASP015K, Pharmacology, 03 medical and health sciences, Immune system, Adjuvants, Immunologic, Oral administration, STAT5 Transcription Factor, Animals, Humans, Medicine, Infusions, Parenteral, Peficitinib, Phosphorylation, Rheumatoid arthritis, Receptor, STAT5, Cell Proliferation, Dose-Response Relationship, Drug, biology, business.industry, lcsh:RM1-950, Janus Kinase 3, Janus Kinase 1, medicine.disease, Arthritis, Experimental, Adjuvant-induced arthritis, Rats, lcsh:Therapeutics. Pharmacology, 030104 developmental biology, Cytokine, biology.protein, Molecular Medicine, Female, Janus kinase, business, Tyrosine kinase
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6
المؤلفون: Kaoru Yamagami, Saki Oaku, Shinji Yamada
المصدر: Tetrahedron Letters. 57:2451-2454
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Organic Chemistry, Inorganic chemistry, Cation π, 010402 general chemistry, Photochemistry, 01 natural sciences, Biochemistry, 0104 chemical sciences, Drug Discovery, Solid phases, Molecule, Irradiation, Selectivity
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7
المؤلفون: Toshihiro Hamajima, Fumie Takahashi, Yukihito Sugano, Susumu Yamaki, Satoshi Kubo, Kaoru Yamagami, Koji Kato, Koji Nakamura, Nozomu Hamakawa, Koji Yokoo, Hidehiko Fukahori, Ayako Moritomo
المصدر: Bioorganicmedicinal chemistry. 26(14)
مصطلحات موضوعية: 0301 basic medicine, Gene isoform, Models, Molecular, Class I Phosphatidylinositol 3-Kinases, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, 03 medical and health sciences, Mice, Phosphatidylinositol 3-Kinases, Structure-Activity Relationship, 0302 clinical medicine, Pharmacokinetics, In vivo, Drug Discovery, Pyrazolopyridine, Potency, Animals, Humans, Molecular Biology, Protein Kinase Inhibitors, Cell Proliferation, Phosphoinositide-3 Kinase Inhibitors, Mice, Inbred BALB C, biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Computational Biology, 030104 developmental biology, 030220 oncology & carcinogenesis, biology.protein, Microsome, Molecular Medicine, Pyrazoles, Female, Antibody, Selectivity
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8
المؤلفون: Tomoko Masunaga, Junko Imanishi, Katsuya Nakamura, Eiji Yoshimi, Kanae Kuroda, Fumie Takahashi, Kaoru Yamagami, Seitaro Mutoh, Emi Hamachi, Masako Kuno, Susumu Miyata, Yoshitaka Ohkubo, Yoshiaki Morita, Satoshi Aoki
المصدر: Biochemical Pharmacology. 82:746-754
مصطلحات موضوعية: Male, Analgesic, Pain, CHO Cells, Osteoarthritis, In Vitro Techniques, Pharmacology, Carrageenan, Biochemistry, Rats, Sprague-Dawley, Mice, Cricetulus, Diclofenac, Cricetinae, medicine, Animals, Edema, Humans, Cyclooxygenase Inhibitors, Stomach Ulcer, Antipyretic, Rofecoxib, ED50, Acetic Acid, Cyclooxygenase 2 Inhibitors, biology, business.industry, Triazoles, medicine.disease, Arthritis, Experimental, Recombinant Proteins, Rats, Cyclooxygenase 2, Hyperalgesia, Rats, Inbred Lew, Rheumatoid arthritis, Cyclooxygenase 1, biology.protein, Female, Cyclooxygenase, business, medicine.drug
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9Effect of FK3657, a non-peptide bradykinin B2 receptor antagonist, on allergic airway disease models
المؤلفون: Seitaro Mutoh, Kikuo Miyayasu, Yoshitaka Ohkubo, Takumi Imai, Yoshitaka Hirayama, Kaoru Yamagami
المصدر: European Journal of Pharmacology. 467:197-203
مصطلحات موضوعية: Male, Ovalbumin, Bronchoconstriction, Guinea Pigs, Bradykinin, Bronchi, Mucous membrane of nose, Pharmacology, Bronchoconstrictor Agents, Capillary Permeability, Plasma, chemistry.chemical_compound, Bradykinin B2 Receptor Antagonists, medicine, Animals, ED50, Asthma, Activator (genetics), business.industry, medicine.disease, Extravasation, Trachea, Nasal Mucosa, chemistry, Acrylamide, Immunology, Quinolines, Toluene 2,4-Diisocyanate, medicine.symptom, business, Bronchoalveolar Lavage Fluid
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10
المؤلفون: N. Seki, Yasutomo Fujii, Kaori Hanaoka, Kenji Okuma, Kaoru Yamagami, Masamichi Inami, Misato Ito, Shohei Shirakami, S. Miyata, Yoshiaki Morita, Takayuki Inoue, Shunji Yamazaki, Yasuyuki Higashi, Hiroki Morio
المصدر: Annals of the Rheumatic Diseases. 72:A197.1-A197
مصطلحات موضوعية: business.industry, medicine.medical_treatment, Immunology, Ankle bone, Pharmacology, medicine.disease, General Biochemistry, Genetics and Molecular Biology, Cytokine, Rheumatology, Erythropoietin, Tyrosine kinase 2, Oral administration, Rheumatoid arthritis, medicine, Immunology and Allergy, medicine.bone, Janus kinase, business, medicine.drug, Whole blood