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المؤلفون: Stephanie Curry, Frederick C. Lahser, Ping Qiu, Karin Bystol, Ernest Asante-Appiah, Stuart Black, Rong Liu, Ellen Xia, Patricia McMonagle, Paul Ingravallo, Robert Chase
المصدر: Antimicrobial Agents and Chemotherapy. 63
مصطلحات موضوعية: Elbasvir, viruses, Hepatitis C virus, medicine.disease_cause, law.invention, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, law, medicine, Pharmacology (medical), NS5A, Pharmacology, chemistry.chemical_classification, 0303 health sciences, NS3, Methionine, 030306 microbiology, Chemistry, biochemical phenomena, metabolism, and nutrition, Virology, Amino acid, Infectious Diseases, Grazoprevir, Recombinant DNA, 030211 gastroenterology & hepatology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::e100148603244b2a292b9b2fdfc91b5b
https://doi.org/10.1128/aac.01269-19 -
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المؤلفون: Ernest, Asante-Appiah, Paul, Ingravallo, Patricia, McMonagle, Karin, Bystol, Ellen, Xia, Stephanie, Curry, Ping, Qiu, Stuart, Black, Robert, Chase, Rong, Liu, Fred, Lahser
المصدر: Antimicrob Agents Chemother
مصطلحات موضوعية: viruses, biochemical phenomena, metabolism, and nutrition, Antiviral Agents
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::40a831b30489de64559c83f4c7dee379
https://pubmed.ncbi.nlm.nih.gov/31527040 -
3In Vitro Antiviral Profile of Ruzasvir, a Potent and Pangenotype Inhibitor of Hepatitis C Virus NS5A
المؤلفون: Wensheng Yu, Joseph A. Kozlowski, Stuart Black, Robert Chase, Paul Ingravallo, Ling Tong, Sony Agrawal, Eric Ferrari, Patricia McMonagle, Karin Bystol, Donna Carr, Ernest Asante-Appiah, Frederick C. Lahser, Laura Rokosz, Rong Liu, Stephanie Curry
المصدر: Antimicrobial Agents and Chemotherapy. 62
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, NS3, Chemistry, viruses, Hepatitis C virus, 030106 microbiology, biochemical phenomena, metabolism, and nutrition, Prodrug, medicine.disease_cause, Antiviral Agents, Virology, digestive system diseases, 03 medical and health sciences, Infectious Diseases, Grazoprevir, medicine, Potency, Pharmacology (medical), Protease inhibitor (pharmacology), Replicon, NS5A
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::944a382870f51dc543862102d935e91a
https://doi.org/10.1128/aac.01280-18 -
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المؤلفون: Daria J. Hazuda, Robert Chase, Rong Liu, Karin Bystol, Ernest Asante-Appiah, Paul Ingravallo, Anita Y. M. Howe, Ellen Xia, Patricia McMonagle, Stephanie Curry, Frederick C. Lahser, Todd A. Black
المصدر: Antimicrobial Agents and Chemotherapy. 60:2954-2964
مصطلحات موضوعية: Cyclopropanes, 0301 basic medicine, Elbasvir, Genotype, viruses, Hepacivirus, Hepatitis C virus, 030106 microbiology, medicine.disease_cause, Antiviral Agents, 03 medical and health sciences, Quinoxalines, Ribavirin, medicine, Protease Inhibitors, Pharmacology (medical), Protease inhibitor (pharmacology), Replicon, NS5A, Benzofurans, Pharmacology, Sulfonamides, NS3, biology, Imidazoles, biology.organism_classification, Amides, Virology, Infectious Diseases, Grazoprevir, Mutation, Drug Therapy, Combination, Carbamates
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7e963f44f512925504383d93478dc2ae
https://doi.org/10.1128/aac.00051-16 -
5
المؤلفون: Shiying Chen, Mark Cartwright, Joseph A. Kozlowski, Lei Chen, Tao Ji, Ling Tong, Patricia McMonagle, Wensheng Yu, Frederick C. Lahser, Laura L. Rokosz, Rong Liu, Kung-I Feng, Bin Hu, Jingjun Yin, Jinglai Hao, Shuai Zan, Oleg Selyutin, Sony Agrawal, Paul Ingravallo, Rebecca T. Ruck, Bin Zhong, Karin Bystol, Donna Carr, Ernest Asante-Appiah, Stephanie Curry
المصدر: Journal of medicinal chemistry. 61(9)
مصطلحات موضوعية: Male, Elbasvir, Genotype, Drug resistance, Hepacivirus, Viral Nonstructural Proteins, 01 natural sciences, Antiviral Agents, chemistry.chemical_compound, Dogs, Pharmacokinetics, Valine, Drug Discovery, Drug Resistance, Viral, Potency, Animals, Tissue Distribution, 010405 organic chemistry, Chemistry, Drug discovery, Virology, 0104 chemical sciences, Rats, 010404 medicinal & biomolecular chemistry, Aminal, Molecular Medicine
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المؤلفون: Sony Agrawal, Bin Hu, Deyou Sha, Rebecca T. Ruck, Tao Ji, Rong Liu, Bin Zhong, Wensheng Yu, Ian W. Davies, Kung-I Feng, Patricia McMonagle, Shuai Zan, Lei Chen, Ellen Xia, Laura L. Rokosz, Robert Mazzola, Frederick C. Lahser, Jingjun Yin, Stephanie Curry, Karin Bystol, Donna Carr, Ernest Asante-Appiah, Oleg Selyutin, Shiying Chen, Anilkumar G. Nair, Mark Cartwright, Jae-Hun Kim, Jinglai Hao, Paul Ingravallo, Ling Tong, Joseph A. Kozlowski, Michael P. Dwyer
المصدر: Journal of medicinal chemistry. 60(1)
مصطلحات موضوعية: 0301 basic medicine, Pyrrolidines, viruses, Mutant, Hepacivirus, Pharmacology, Viral Nonstructural Proteins, Bioinformatics, Antiviral Agents, Heterocyclic Compounds, 4 or More Rings, Cell Line, 03 medical and health sciences, Structure-Activity Relationship, 0302 clinical medicine, Dogs, Drug Discovery, Genotype, Animals, Humans, HCV NS5A Inhibitor, NS5A, Indole test, Polymorphism, Genetic, Chemistry, virus diseases, Haplorhini, biochemical phenomena, metabolism, and nutrition, digestive system diseases, Rats, Regimen, Thiazoles, 030104 developmental biology, Molecular Medicine, 030211 gastroenterology & hepatology
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المؤلفون: Bin Hu, Ling Tong, Sony Agrawal, Craig A. Coburn, Bandarpalle B. Shankar, Michael P. Dwyer, Bin Zhong, Lei Chen, Shiying Chen, Seong Heon Kim, Stuart B. Rosenblum, Shuai Zan, Karin Bystol, Ian W. Davies, Donna Carr, Ernest Asante-Appiah, Wensheng Yu, Joseph A. Kozlowski, Rebecca T. Ruck, Patricia McMonagle, Anilkumar G. Nair, Rong Liu, Oleg Selyutin, De-Yi Yang, Paul Ingravallo, Tao Ji, Qingbei Zeng, Jinglai Hao, Stephanie Curry, Frederick C. Lahser
المصدر: Bioorganicmedicinal chemistry letters. 26(21)
مصطلحات موضوعية: 0301 basic medicine, Indoles, Proline, Stereochemistry, viruses, Clinical Biochemistry, Pharmaceutical Science, Viral Nonstructural Proteins, 01 natural sciences, Biochemistry, Antiviral Agents, 03 medical and health sciences, Structure-Activity Relationship, Drug Discovery, HCV NS5A Inhibitor, Replicon, NS5A, Molecular Biology, Benzofurans, Indole test, Chemistry, Organic Chemistry, Imidazoles, virus diseases, biochemical phenomena, metabolism, and nutrition, digestive system diseases, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 030104 developmental biology, Molecular Medicine