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1
المؤلفون: Beth Ann McKenna, Karla Kopec, Greg A. Hostetler, Sankar Chatterjee, Derek Dunn
المصدر: Chemical Biology & Drug Design. 83:666-669
مصطلحات موضوعية: Drug Inverse Agonism, Stereochemistry, Pharmacology, Biochemistry, Benzazepine, chemistry.chemical_compound, Drug Discovery, Humans, Inverse agonist, Potency, Sulfones, Receptor, Sulfonamides, Molecular Structure, Organic Chemistry, Benzazepines, chemistry, Receptors, Serotonin, 5-HT6 receptor, Molecular Medicine, Biological Assay, Enantiomer, Chirality (chemistry), Protein Binding
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2
المؤلفون: Sankar Chatterjee, Karla Kopec, Beth Ann McKenna, Greg A. Hostetler, Derek Dunn
المصدر: Chemical Biology & Drug Design. 83:149-153
مصطلحات موضوعية: Stereochemistry, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Humans, Potency, Spiro Compounds, Structural motif, Receptor, Pharmacology, Sulfonamides, Chemistry, Organic Chemistry, Stereoisomerism, Benzazepines, Recombinant Proteins, Receptors, Serotonin, 5-HT6 receptor, Thiazolidines, Molecular Medicine, Serotonin Antagonists, Nonane, Enantiomer, Antagonism, Selectivity, Protein Binding
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3
المؤلفون: Thomas J. Connors, Jie Qian, Zeck Huang, Joanne R. Mathiasen, Edward R. Bacon, Thelma S. Angeles, Mark J. Huffman, Emir Duzic, Joseph M. Salvino, Beth Ann McKenna, Hervé Schaffhauser, Robert J. McHugh, Lily D. Lu, George C. Morton, Beverly P. Holskin, Karla Kopec, Amy DiCamillo, Gerard C. Rosse, Chrysanthe Spais, Rabindranath Tripathy, Lisa D. Aimone
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:1421-1426
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Stereoisomerism, Biochemistry, Sulfone, chemistry.chemical_compound, In vivo, Drug Discovery, 5-HT6 receptor, Molecular Medicine, Pharmacophore, Receptor, Molecular Biology, 5-HT receptor
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4
المؤلفون: Beverly P. Holskin, Karla Kopec, Joanne R. Mathiasen, Amy DiCamillo, Babu G. Sundar, Thomas J. Connors, Emir Duzic, Edward R. Bacon, Gerard C. Rosse, Chrysanthe Spais, Thomas R. Bailey, Beth Ann McKenna, Rebecca A. Brown, Jie Qian, Derek Dunn, Mark J. Huffman, Joseph M. Salvino, Huang Zeqi, Lisa D. Aimone, Hervé Schaffhauser, Deborah Galinis, Thelma S. Angeles, Lily D. Lu, George C. Morton
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:120-123
مصطلحات موضوعية: biology, Organic Chemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Pharmacology, Biochemistry, Social recognition, chemistry.chemical_compound, chemistry, Drug Discovery, biology.protein, 5-HT6 receptor, Molecular Medicine, Structure–activity relationship, Serotonin Antagonists, Penetrant (biochemical), Receptor, Molecular Biology, 5-HT receptor
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5
المؤلفون: Michael Williams, Karla Kopec, Donna Bozyczko-Coyne
المصدر: Biochemical Pharmacology. 69:1133-1139
مصطلحات موضوعية: Proteomics, Pharmacology, Two-dimensional gel electrophoresis, Proteome, Test data generation, Drug discovery, Computational Biology, Reproducibility of Results, Context (language use), Computational biology, Biology, Bioinformatics, Biochemistry, Genome, Pharmaceutical Preparations, Drug Design, Identification (biology), Forecasting, Signal Transduction
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6
المؤلفون: Rabindranath, Tripathy, Robert J, McHugh, Edward R, Bacon, Joseph M, Salvino, George C, Morton, Lisa D, Aimone, Zeck, Huang, Joanne R, Mathiasen, Amy, DiCamillo, Mark J, Huffman, Beth A, McKenna, Karla, Kopec, Lily D, Lu, Jie, Qian, Thelma S, Angeles, Thomas, Connors, Chrysanthe, Spais, Beverly, Holskin, Emir, Duzic, Hervé, Schaffhauser, Gerard C, Rossé
المصدر: Bioorganicmedicinal chemistry letters. 22(3)
مصطلحات موضوعية: Molecular Structure, Brain, Stereoisomerism, Rats, Inhibitory Concentration 50, Mice, Dogs, Receptors, Serotonin, Microsomes, Liver, Animals, Humans, Serotonin Antagonists, Sulfones, Heterocyclic Compounds, 3-Ring
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7
المؤلفون: Babu G, Sundar, Thomas R, Bailey, Derek D, Dunn, Edward R, Bacon, Joseph M, Salvino, George C, Morton, Lisa D, Aimone, Huang, Zeqi, Joanne R, Mathiasen, Amy, Dicamillo, Mark J, Huffman, Beth A, McKenna, Karla, Kopec, Lily D, Lu, Rebecca, Brown, Jie, Qian, Thelma, Angeles, Thomas, Connors, Chrysanthe, Spais, Beverly, Holskin, Deborah, Galinis, Emir, Duzic, Herve, Schaffhauser, Gerard C, Rosse
المصدر: Bioorganicmedicinal chemistry letters. 22(1)
مصطلحات موضوعية: ERG1 Potassium Channel, Brain, Ether-A-Go-Go Potassium Channels, Rats, Inhibitory Concentration 50, Kinetics, Structure-Activity Relationship, Memory, Short-Term, Models, Chemical, Piperidines, Receptors, Serotonin, Schizophrenia, Animals, Humans, Serotonin Antagonists, Benzofurans
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8
المؤلفون: Beth Ann McKenna, Karla Kopec, Daniel Pauletti
المصدر: Current Protocols in Pharmacology
مصطلحات موضوعية: Pharmacology, Gene isoform, GABA Plasma Membrane Transport Proteins, genetic structures, Cell, GABA transporter activity, Transporter, Transfection, Biology, chemistry.chemical_compound, medicine.anatomical_structure, HEK293 Cells, nervous system, chemistry, Biochemistry, Homogeneous, Cell culture, COS Cells, Chlorocebus aethiops, medicine, Animals, Humans, Neurotransmitter, gamma-Aminobutyric Acid
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9Comparison of organophosphorous acid anhydrolases from different species using monoclonal antibodies
المؤلفون: Karla Kopec-Smyth, Jennifer L. Poppino, Susan L. Futrovsky, Jeffrey R. Deschamps, Keith B. Ward
المصدر: Comparative Biochemistry and Physiology Part C: Pharmacology, Toxicology and Endocrinology. 106:765-768
مصطلحات موضوعية: Substrate Specificities, Anticorps monoclonal, medicine.drug_class, Immunology, Enzyme-Linked Immunosorbent Assay, Viper Venoms, Monoclonal antibody, Epitope, Substrate Specificity, Epitopes, Mice, medicine, Animals, Optic ganglion, Pharmacology, chemistry.chemical_classification, Mice, Inbred BALB C, biology, Aryldialkylphosphatase, Decapodiformes, Esterases, Antibodies, Monoclonal, biology.organism_classification, Molecular biology, Enzyme, chemistry, Biochemistry, Female, Hepatopancreas
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d352435290dbff404b9e48b99e97a7c2
https://doi.org/10.1016/0742-8413(93)90240-l -
10
المؤلفون: Justin Schreiber, Karla Kopec, Sheryl L. Meyer, Chrysanthe Spais, John T. Durkin
المصدر: Brain research. 1374
مصطلحات موضوعية: Gene isoform, Amino terminal, CHO Cells, Pharmacology, Biology, Glycine transporter, Cricetulus, Piperidines, Glycine Plasma Membrane Transport Proteins, Cricetinae, Potency, Animals, Humans, Protein Isoforms, Molecular Biology, Dose-Response Relationship, Drug, General Neuroscience, Sarcosine, Molecular biology, Protein Structure, Tertiary, Biochemistry, Cell culture, RNA splicing, Glycine, Benzamides, Neurology (clinical), Precursor mRNA, Developmental Biology