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المؤلفون: Franciszek Sączewski, Maria Gdaniec, Jarosław Sączewski, Mariusz Belka, Alan L. Hudson, Anita Kornicka, Apolonia Rybczyńska, Tomasz Bączek, Aleksandra Wasilewska, Karol Gzella, Konrad Boblewski, Artur Lehmann
المصدر: Chemical Biology & Drug Design. 89:400-410
مصطلحات موضوعية: Male, 0301 basic medicine, Indoles, Stereochemistry, In silico, Drug Evaluation, Preclinical, Imidazoline receptor, Blood Pressure, Chemistry Techniques, Synthetic, Imidazolidines, 01 natural sciences, Biochemistry, Rats, Sprague-Dawley, Radioligand Assay, Structure-Activity Relationship, 03 medical and health sciences, Drug Stability, Heart Rate, In vivo, Drug Discovery, Animals, Rats, Wistar, Binding site, Receptor, Antihypertensive Agents, Pharmacology, Indole test, Dose-Response Relationship, Drug, 010405 organic chemistry, Chemistry, Organic Chemistry, Receptors, Adrenergic, alpha, In vitro, 0104 chemical sciences, 030104 developmental biology, Molecular Medicine, Selectivity
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المؤلفون: Ordyszewska, Anita Kornicka, Karol Gzella, Katarzyna Garbacz, Małgorzata Jarosiewicz, Maria Gdaniec, Joanna Fedorowicz, Łukasz Balewski, Jakub Kokoszka, Anna
المصدر: Pharmaceuticals; Volume 16; Issue 7; Pages: 918
مصطلحات موضوعية: indole-acrylonitrile derivatives, cell growth inhibition, antimicrobial activity, molecular docking, ADME
وصف الملف: application/pdf
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المصدر: Molbank, Vol 2019, Iss 4, p M1093 (2019)
مصطلحات موضوعية: Reaction mechanism, Carboxylic acid, [1,3]-h shift, isoxazolo[3,4-b]quinolin-3(1h)-one, 010402 general chemistry, Mass spectrometry, 01 natural sciences, Biochemistry, Medicinal chemistry, dft calculations, chemistry.chemical_compound, dimethyl acetylenedicarboxylate, aza-michael addition, lcsh:Inorganic chemistry, Physical and Theoretical Chemistry, Dimethyl acetylenedicarboxylate, chemistry.chemical_classification, 010405 organic chemistry, Organic Chemistry, Quinoline, Nuclear magnetic resonance spectroscopy, lcsh:QD146-197, 0104 chemical sciences, chemistry, Elemental analysis, Density functional theory
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4دورية أكاديمية
المؤلفون: Anita Kornicka, Karol Gzella, Katarzyna Garbacz, Małgorzata Jarosiewicz, Maria Gdaniec, Joanna Fedorowicz, Łukasz Balewski, Jakub Kokoszka, Anna Ordyszewska
المصدر: Pharmaceuticals, Vol 16, Iss 7, p 918 (2023)
مصطلحات موضوعية: indole-acrylonitrile derivatives, cell growth inhibition, antimicrobial activity, molecular docking, ADME, Medicine, Pharmacy and materia medica, RS1-441
وصف الملف: electronic resource
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5دورية أكاديمية
المصدر: Molbank, Vol 2019, Iss 4, p M1093 (2019)
مصطلحات موضوعية: [1,3]-h shift, aza-michael addition, dft calculations, dimethyl acetylenedicarboxylate, isoxazolo[3,4-b]quinolin-3(1h)-one, Inorganic chemistry, QD146-197
وصف الملف: electronic resource