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1دورية أكاديمية
المؤلفون: Chihiro Nakamoto, Yuhei Goto, Yoko Tomizawa, Yuko Fukata, Masaki Fukata, Kasper Harpsøe, David E. Gloriam, Kazuhiro Aoki, Tomonori Takeuchi
المصدر: Molecular Brain, Vol 14, Iss 1, Pp 1-14 (2021)
مصطلحات موضوعية: GPCR, Dopamine, Norepinephrine, Fluorescence probe, Hippocampal neuron, Neurology. Diseases of the nervous system, RC346-429
وصف الملف: electronic resource
Relation: https://doaj.org/toc/1756-6606
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2
المؤلفون: Jimmy Caroli, Alibek Mamyrbekov, Kasper Harpsøe, Sahar Gardizi, Linda Dörries, Eshan Ghosh, Alexander S. Hauser, Albert J. Kooistra, David E. Gloriam
المصدر: Nature Chemical Biology. 19:531-535
مصطلحات موضوعية: Cell Biology, Molecular Biology
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3
المؤلفون: Emil Marcher-Rørsted, Jitka Nykodemová, Kasper Harpsøe, Anders A. Jensen, Jesper L. Kristensen
المصدر: ACS Medicinal Chemistry Letters. 14:319-325
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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4
المؤلفون: Christian R. O. Bartling, Flora Alexopoulou, Sarah Kuschert, Yanni K.-Y. Chin, Xinying Jia, Vita Sereikaite, Dennis Özcelik, Thomas M. Jensen, Palash Jain, Mads M. Nygaard, Kasper Harpsøe, David E. Gloriam, Mehdi Mobli, Kristian Strømgaard
المصدر: Journal of Medicinal Chemistry. 66:3045-3057
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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5
المؤلفون: Yali Zhou, Henrik Daver, Boris Trapkov, Lijie Wu, Meng Wu, Kasper Harpsøe, Patrick R. Gentry, Kaiwen Liu, Marina Larionova, Junlin Liu, Na Chen, Hans Bräuner-Osborne, David E. Gloriam, Tian Hua, Zhi-Jie Liu
المصدر: Cell Research
Zhou, Y, Daver, H, Trapkov, B, Wu, L, Wu, M, Harpsøe, K, Gentry, P R, Liu, K, Larionova, M, Liu, J, Chen, N, Bräuner-Osborne, H, Gloriam, D E, Hua, T & Liu, Z J 2022, ' Molecular insights into ligand recognition and G protein coupling of the neuromodulatory orphan receptor GPR139 ', Cell Research, vol. 32, no. 2, pp. 210-213 . https://doi.org/10.1038/s41422-021-00591-wمصطلحات موضوعية: Cryoelectron microscopy, GTP-Binding Proteins, Extracellular signalling molecules, Nerve Tissue Proteins, Cell Biology, Ligands, Molecular Biology, Letter to the Editor, Receptors, G-Protein-Coupled
وصف الملف: application/pdf
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6
المؤلفون: Jimmy Caroli, Alibek Mamyrbekov, Kasper Harpsøe, Sahar Gardizi, Linda Dörries, Eshan Ghosh, Alexander Hauser, Albert Kooistra, David Gloriam
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::63a11ac73dbd339303f540d89d777140
https://doi.org/10.21203/rs.3.rs-2155951/v1 -
7
المؤلفون: Christian B M, Poulie, Eline, Pottie, Icaro A, Simon, Kasper, Harpsøe, Laura, D'Andrea, Igor V, Komarov, David E, Gloriam, Anders A, Jensen, Christophe P, Stove, Jesper L, Kristensen
المصدر: Journal of medicinal chemistry. 65(18)
مصطلحات موضوعية: Lysergic Acid Diethylamide, Serotonin, Hallucinogens, Receptor, Serotonin, 5-HT2A, Serotonin 5-HT2 Receptor Agonists, beta-Arrestins
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8
المؤلفون: Sijie Huang, Peiyu Xu, Dan-Dan Shen, Icaro A. Simon, Chunyou Mao, Yangxia Tan, Huibing Zhang, Kasper Harpsøe, Huadong Li, Yumu Zhang, Chongzhao You, Xuekui Yu, Yi Jiang, Yan Zhang, David E. Gloriam, H. Eric Xu
المساهمون: Medicinal chemistry, AIMMS
المصدر: Huang, S, Xu, P, Shen, D D, Simon, I A, Mao, C, Tan, Y, Zhang, H, Harpsøe, K, Li, H, Zhang, Y, You, C, Yu, X, Jiang, Y, Zhang, Y, Gloriam, D E & Xu, H E 2022, ' GPCRs steer G i and G s selectivity via TM5-TM6 switches as revealed by structures of serotonin receptors ', Molecular cell, vol. 82, no. 14, pp. 2681-2695.e6 . https://doi.org/10.1016/j.molcel.2022.05.031
Molecular cell, 82(14), 2681-2695.e6. Cell Pressمصطلحات موضوعية: ligand selectivity, serotonin receptor, GPCR, 5-HT, cryo-EM structure, Cell Biology, G protein selectivity, Molecular Biology, 5-HT receptor, signaling complex
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::54c14e6f3505ee05c519a1463efa9c29
https://hdl.handle.net/1871.1/713d857a-269d-42a6-a385-466fed3a7d58 -
9
المؤلفون: Lisa Pallareti, Tine F. Rath, Boris Trapkov, Tsonko Tsonkov, Anders Thorup Nielsen, Kasper Harpsøe, Patrick R. Gentry, Hans Bräuner-Osborne, David E. Gloriam, Simon R. Foster
المصدر: Pallareti, L, Rath, T F, Trapkov, B, Tsonkov, T, Nielsen, A T, Harpsøe, K, Gentry, P R, Bräuner-Osborne, H, Gloriam, D E & Foster, S R 2023, ' Pharmacological characterization of novel small molecule agonists and antagonists for the orphan receptor GPR139 ', European Journal of Pharmacology, vol. 943, 175553 . https://doi.org/10.1016/j.ejphar.2023.175553
مصطلحات موضوعية: Pharmacology
وصف الملف: application/pdf
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10
المؤلفون: David E. Gloriam, Rebekka Löffler, Frederik Rostrup, Petrine Wellendorph, Bente Frølund, Christina Birkedahl Falk-Petersen, Kasper Harpsøe, Stine Buchleithner
المصدر: Molecular Pharmacology. 100:46-56
مصطلحات موضوعية: Pharmacology, Diazepam binding, GABAA receptor, Chemistry, Docking (molecular), Stereochemistry, Allosteric regulation, Functional selectivity, Molecular Medicine, Ligand-gated ion channel, Binding site, Receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b61e1339ce2ac4e170729ea407919188
https://doi.org/10.1124/molpharm.121.000266