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1
المؤلفون: William J. Pitts, Alaric J. Dyckman, Scott H. Watterson, Robert V. Moquin, Kim W. McIntyre, Zheng Yang, Jagabandhu Das, Katy Van Kirk, James R. Burke, David B. Wang-Iverson, Hollie Booth-Lute, James Kempson, Laishun Chen, Charles M. Langevine, Joel C. Barrish, Guchen Yang, Xiaoxia Yang, John H. Dodd, David S. Nirschl, Murray McKinnon, Steven H. Spergel, Mark A. Pattoli, Michael Galella, Kurt R. Gregor, Junquing Guo
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:7006-7012
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Biochemistry, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Acetamides, Drug Discovery, Animals, Humans, Inhibitory concentration 50, Structure–activity relationship, Potency, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Molecular Structure, Drug discovery, Organic Chemistry, Inflammatory Bowel Diseases, In vitro, I-kappa B Kinase, Rats, Enzyme Activation, chemistry, Molecular Medicine, Heterocyclic Compounds, 3-Ring, Acetamide, Tricyclic
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2
المؤلفون: Charles M. Langevine, Joseph A. Furch, Dominique Belanger, Mark A. Pattoli, Joel C. Barrish, Alaric J. Dyckman, Marco Dodier, James Kempson, Jagabandhu Das, David S. Nirschl, Laishun Chen, Punit Marathe, Kathleen M. Gillooly, Junqing Guo, Robert V. Moquin, John H. Dodd, Murray McKinnon, Anne Marinier, Zheng Yang, Steven H. Spergel, Claude A. Quesnelle, Kim W. McIntyre, Katy Van Kirk, James R. Burke, William J. Pitts, Scott H. Watterson, Alain Martel, Patrice Gill, David B. Wang-Iverson, Tianle Li
المصدر: Journal of Medicinal Chemistry. 52:1994-2005
مصطلحات موضوعية: Lipopolysaccharides, Recombinant Fusion Proteins, IκB kinase, In Vitro Techniques, Crystallography, X-Ray, Chemical synthesis, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Animals, Humans, Thiazole, Oxazoles, Glutathione Transferase, Oxazole, chemistry.chemical_classification, Mice, Inbred BALB C, Tumor Necrosis Factor-alpha, Imidazoles, Biological activity, I-kappa B Kinase, Rats, Thiazoles, Enzyme, chemistry, Biochemistry, Leukocytes, Mononuclear, Microsomes, Liver, Molecular Medicine, Female, Signal transduction, Heterocyclic Compounds, 3-Ring, Tricyclic
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3
المؤلفون: Jacques Y. Roberge, Muthoni G. Kamau, Sam T. Chao, Arvind Mathur, Michael A. Poss, Zheming Ruan, Lalgudi S. Harikrishnan, Dora M. Schnur, Mark S. Bednarz, John K. Dickson, Roy J. Vaz, Yalei Liu, R. Michael Lawrence, Ramesh Kakarla, Leslie Leith, Ashvinikumar V. Gavai, Christopher B. Cooper, Katy Van Kirk
المصدر: Journal of Combinatorial Chemistry. 11:72-82
مصطلحات موضوعية: Polymers, Chemistry, Stereochemistry, Acetal, Antagonist, General Chemistry, Combinatorial chemistry, Receptors, G-Protein-Coupled, Propanolamines, Small Molecule Libraries, chemistry.chemical_compound, Cross-Linking Reagents, Drug Design, Combinatorial Chemistry Techniques, Humans, Amines, Linker, Polymer supported, G protein-coupled receptor
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المؤلفون: Cooper Christopher B, Katy Van Kirk, Zheming Ruan, R. Michael Lawrence
المصدر: Research Letters in Organic Chemistry. 2008:1-4
مصطلحات موضوعية: Reaction conditions, chemistry.chemical_classification, Strategy and Management, Mechanical Engineering, Carboxylic acid, Metals and Alloys, chemistry.chemical_element, One-Step, Industrial and Manufacturing Engineering, Catalysis, chemistry.chemical_compound, chemistry, Phenylsilane, Organic chemistry, Palladium
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::383403cf00f28c0edcbf0a65638087cd
https://doi.org/10.1155/2008/696090 -
5
المؤلفون: Heather Finlay, Mark E. Salvati, Leonard P. Adam, Ji Jiang, Ruth R. Wexler, Christine Huang, David S. Taylor, Xiaohong Yin, Alice Ye A. Chen, Paul G. Sleph, Yufeng Wang, Muthoni G. Kamau, Wu Yang, R. Michael Lawrence, David S. Nirschl, Lalgudi S. Harikrishnan, Katy Van Kirk, Richard Yang
المصدر: Bioorganicmedicinal chemistry letters. 24(3)
مصطلحات موضوعية: Stereochemistry, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, chemistry.chemical_compound, Transactivation, Inhibitory Concentration 50, Structure-Activity Relationship, Drug Stability, Biomimetics, Heterocyclic Compounds, Drug Discovery, Cholesterylester transfer protein, Ethylamines, Humans, Urea, Molecular Biology, Pregnane X receptor, Chemotype, biology, Molecular Structure, Chemistry, Organic Chemistry, Biphenyl Compounds, Metabolic stability, Cholesterol Ester Transfer Proteins, biology.protein, Molecular Medicine
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المصدر: Solid-Phase Organic Syntheses, Volume 2
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Phenylsilane, chemistry.chemical_element, Organic chemistry, One-Step, Palladium
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::82fa37a53732461dd878613c2bea2594
https://doi.org/10.1002/9781118336953.ch3 -
7Diphenylpyridylethanamine (DPPE) derivatives as cholesteryl ester transfer protein (CETP) inhibitors
المؤلفون: Leonard P. Adam, Michael A. Poss, Mark E. Salvati, James J. Li, Muthoni G. Kamau, R. Michael Lawrence, Michael Galella, Heather Finlay, Xue-Qing Chen, Arthur V. Miller, Richard Yang, Tammy C. Wang, Doree F. Sitkoff, Xiaohong Yin, Alice Ye A. Chen, Christine Huang, David S. Taylor, Lalgudi S. Harikrishnan, Paul G. Sleph, Ji Jiang, Christopher B. Cooper, Ruth R. Wexler, David S. Nirschl, Ming Chang, Katy Van Kirk, Jennifer X. Qiao
المصدر: Journal of medicinal chemistry. 55(13)
مصطلحات موضوعية: Genetically modified mouse, Male, Pyridines, Transgene, Blood Pressure, Coronary Disease, Mice, Transgenic, Pharmacology, chemistry.chemical_compound, Inhibitory Concentration 50, Mice, Heart Rate, Amide, Cricetinae, Cholesterylester transfer protein, Drug Discovery, Stilbenes, Potency, Animals, Humans, biology, Molecular Structure, Cholesterol, Anticholesteremic Agents, Cetp inhibition, Cholesterol Ester Transfer Proteins, Rats, chemistry, Apolipoprotein B-100, biology.protein, Molecular Medicine
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8
المؤلفون: Christopher B. Cooper, Wu Yang, John K. Dickson, Ramakrishna Seethala, Jean H.M. Feyen, Katy Van Kirk, Yufeng Wang, Zhengping Ma, Zheming Ruan, Brian J. Arey
المصدر: Journal of medicinal chemistry. 52(4)
مصطلحات موضوعية: Chemistry, Drug discovery, Pyridines, Allosteric regulation, Antagonist, Small molecule, Inhibitory Concentration 50, Structure-Activity Relationship, Pyrimidines, Biochemistry, Allosteric Regulation, Solubility, In vivo, Parathyroid Hormone, Drug Discovery, Molecular Medicine, Structure–activity relationship, Humans, Osteoporosis, Calcium-sensing receptor, Receptor, Receptors, Calcium-Sensing
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المؤلفون: David S. Nirschl, Stanley R. Krystek, James C. Sutton, Daniel M. Camac, Ramakrishna Seethala, Jeffrey A. Robl, Rajasree Golla, James J. Li, Robert Zahler, Paul E. Morin, Haixia Wang, Rebecca A. Smirk, Cooper Christopher B, Mary Ellen K. Salyan, Katy Van Kirk, Zhengping Ma, Steven Sheriff, David A. Gordon, Ligaya M. Simpkins, Zheming Ruan, Robert D. Hutchins, Brian Carpenter, Akbar Nayeem, Lawrence G. Hamann, Shung C. Wu
المصدر: Bioorganicmedicinal chemistry letters. 18(11)
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Pyridines, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Carboxamide, Crystallography, X-Ray, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, Oxidoreductase, Amide, Drug Discovery, Pyridine, 11-beta-Hydroxysteroid Dehydrogenase Type 1, medicine, Combinatorial Chemistry Techniques, Humans, Molecular Biology, chemistry.chemical_classification, Molecular Structure, Aryl, Organic Chemistry, Amides, Enzyme, chemistry, Drug Design, Molecular Medicine, Selectivity
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المؤلفون: Cooper Christopher B, Michael A. Poss, Zheming Ruan, Muthoni G. Kamau, Dharmpal S. Dodd, Mark A. Hermsmeier, Katy Van Kirk, Rogelio L. Martinez, and Sarah C. Traeger
المصدر: Journal of combinatorial chemistry. 7(4)
مصطلحات موضوعية: Combinatorial Chemistry Techniques, Molecular Structure, Chemistry, Aryl, General Chemistry, Combinatorial chemistry, chemistry.chemical_compound, Solid-phase synthesis, Reagent, Organic chemistry, Molecule, Pyrazoles, Amines