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1دورية أكاديمية
المؤلفون: Montalvo, Geronda, Zhang, Yao, Young, Trevor, Costanzo, Michael, Freeman, Katie, Wang, Jun, Clements, Dylan, Magavern, Emma, Kavash, Robert, Scott, Richard, Liu, Dahui, Degrado, William
المصدر: ACS Chemical Biology. 9(4)
مصطلحات موضوعية: Circular Dichroism, Dose-Response Relationship, Drug, Drug Design, Fibrinolytic Agents, Heparin, Inhibitory Concentration 50, Models, Biological, Molecular Structure, Protein Binding, Protein Conformation
وصف الملف: application/pdf
URL الوصول: https://escholarship.org/uc/item/32f3w1x1
https://escholarship.org/content/qt32f3w1x1/qt32f3w1x1.pdf -
2دورية أكاديمية
المؤلفون: Love, Melissa S, Millholland, Melanie G, Mishra, Satish, Kulkarni, Swapnil, Freeman, Katie B, Pan, Wenxi, Kavash, Robert W, Costanzo, Michael J, Jo, Hyunil, Daly, Thomas M, Williams, Dewight R, Kowalska, M Anna, Bergman, Lawrence W, Poncz, Mortimer, DeGrado, William F, Sinnis, Photini, Scott, Richard W, Greenbaum, Doron C
المصدر: Cell Host & Microbe. 12(6)
مصطلحات موضوعية: Medical Microbiology, Biomedical and Clinical Sciences, Clinical Sciences, Infectious Diseases, Rare Diseases, HIV/AIDS, Malaria, Vector-Borne Diseases, Hematology, Aetiology, 2.1 Biological and endogenous factors, 2.2 Factors relating to the physical environment, Infection, Good Health and Well Being, Animals, Antimalarials, Cell Survival, Disease Models, Animal, Erythrocytes, Mice, Parasite Load, Parasitemia, Plasmodium falciparum, Platelet Factor 4, Microbiology, Immunology, Biochemistry and cell biology, Medical microbiology
وصف الملف: application/pdf
URL الوصول: https://escholarship.org/uc/item/7mx657d1
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3دورية أكاديمية
المؤلفون: Lewis, Paul J., de Jonge, Marc, Daeyaert, Frits, Koymans, Luc, Vinkers, Maarten, Heeres, Jan, Janssen, Paul A.J., Arnold, Eddy, Das, Kalyan, Clark, Jr., Art D., Hughes, Stephen H., Boyer, Paul L., de Béthune, Marie-Pierre, Pauwels, Rudi, Andries, Koen, Kukla, Mike, Ludovici, Donald, De Corte, Bart, Kavash, Robert, Ho, Chih
المصدر: Journal of Computer-Aided Molecular Design. February 2003 17(2-4):129-134
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4دورية أكاديمية
المؤلفون: Winter, Hans De *, Breslin, Henry, Miskowski, Tamara, Kavash, Robert, Somers, Marijke
المصدر: In Journal of Molecular Graphics and Modelling 2005 23(5):409-418
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5
المؤلفون: Chaozhong Cai, Alexey B. Dyatkin, Paul R. Wade, Kavash Robert W, Sui-Po Zhang, Henry J. Breslin, Craig J. Diamond, Wei He, Tamara A. Miskowski, Pamela J. Hornby
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:4869-4872
مصطلحات موضوعية: Diarrhea, Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Receptors, Opioid, mu, Pharmaceutical Science, Pharmacology, Biochemistry, Irritable Bowel Syndrome, Structure-Activity Relationship, Clinical Trials, Phase II as Topic, Opioid receptor, Receptors, Opioid, delta, Drug Discovery, medicine, Humans, Structure–activity relationship, Receptor, Molecular Biology, Irritable bowel syndrome, Molecular Structure, Chemistry, Organic Chemistry, Antagonist, medicine.disease, Opioid, Molecular Medicine, medicine.symptom, medicine.drug
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6
المصدر: Journal of Molecular Graphics and Modelling. 23:409-418
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, Stereochemistry, Molecular Sequence Data, In Vitro Techniques, Aminopeptidases, Sincalide, Structure-Activity Relationship, Catalytic Domain, Computer Graphics, Materials Chemistry, Computer Simulation, Amino Acid Sequence, Homology modeling, Physical and Theoretical Chemistry, Dipeptidyl-Peptidases and Tripeptidyl-Peptidases, Spectroscopy, Sequence Homology, Amino Acid, biology, Chemistry, Serine Endopeptidases, Tripeptidyl peptidase II, Active site, Computer Graphics and Computer-Aided Design, Drug Design, biology.protein, Thermodynamics, Pharmacophore, Butabindide
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7دورية أكاديمية
المؤلفون: Breslin, Henry J., Diamond, Craig J., Kavash, Robert W., Cai, Chaozhong, Dyatkin, Alexey B., Miskowski, Tamara A., Zhang, Sui-Po, Wade, Paul R., Hornby, Pamela J., He, Wei
المصدر: In Bioorganic & Medicinal Chemistry Letters 15 July 2012 22(14):4869-4872
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8
المؤلفون: Peter Walter Maria Roevens, Hans De Winter, Kavash Robert W, Michael Joseph Kukla, Maria V. F. Somers, Henry J. Breslin, Tamara A. Miskowski
المصدر: ChemInform. 35
مصطلحات موضوعية: Serine protease, biology, Stereochemistry, Chemistry, biology.protein, Tripeptidyl peptidase II, General Medicine, Pharmacophore, Inhibitory postsynaptic potential, IC50
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9
المؤلفون: Maria V. F. Somers, Tamara A. Miskowski, Michael Joseph Kukla, Peter Walter Maria Roevens, Hans De Winter, Kavash Robert W, Henry J. Breslin
المصدر: Bioorganicmedicinal chemistry letters. 13(24)
مصطلحات موضوعية: Models, Molecular, Indoles, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Aminopeptidases, Structure-Activity Relationship, Drug Discovery, Protease Inhibitors, Dipeptidyl-Peptidases and Tripeptidyl-Peptidases, Molecular Biology, IC50, chemistry.chemical_classification, Serine protease, biology, Bicyclic molecule, Molecular Structure, Organic Chemistry, Serine Endopeptidases, Imidazoles, Tripeptidyl peptidase II, Kinetics, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Pharmacophore
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10
المؤلفون: Lewi, Paul, de Jonge, Frederik, Daeyaert, Frits, Koymans, Luc, Vinkers, Maarten, Heeres, Jan, Janssen, Paul A.J., Arnold, Eddy, Das, Kalyan, Clark, Art D., Stephen, H. Hughes, Boyer, Paul L., de Béthune, Marie-Pierre, Pauwels, Rudi, Andries, Koen, Kukla, Mike, Ludovici, Donald, de Corte, Bart, Kavash, Robert, Ho, Chih
المصدر: Journal of computer-aided molecular design