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1
المؤلفون: John Chan, Sandra W. Cowan-Jacob, Takanori Kanazawa, Zheng Chen, Brent A. Appleton, Aaron Smith, Qiong Zhang, Daniel Poon, Clemens Scheufler, Darrin Stuart, Kay Huh, Jeremy Murray, Kevin Shoemaker, Zilin Huang, Hanne Merritt, Susan Kaufman, Laura Tandeske, Cynthia M. Shafer, Zhi-Jie Ni, Johanna M. Jansen
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:5221-5224
مصطلحات موضوعية: Models, Molecular, Proto-Oncogene Proteins B-raf, 0301 basic medicine, MAPK/ERK pathway, Stereochemistry, VEGF receptors, Clinical Biochemistry, Pharmaceutical Science, Heterocyclic Compounds, 2-Ring, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Drug Discovery, Humans, Transferase, Benzamide, Protein Kinase Inhibitors, Molecular Biology, Dose-Response Relationship, Drug, Molecular Structure, biology, Kinase, Organic Chemistry, Combinatorial chemistry, 030104 developmental biology, chemistry, 030220 oncology & carcinogenesis, Benzamides, biology.protein, Molecular Medicine, Selectivity
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2
المؤلفون: Robert Elling, Aaron Smith, Matthew Burger, Kay Huh, Hanne Merritt, Sabina Pecchi, Charles Voliva, Jiong Lan, Wooseok Han, Daniel Menezes, John Chan, Teresa E. Williams, Yongjin Xu, Mark Knapp, Joelle Verhagen, Susan Kaufman, Zhi-Jie Ni
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:742-746
مصطلحات موضوعية: 0301 basic medicine, Imidazopyridine, Pyridines, Stereochemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Antineoplastic Agents, Stereoisomerism, Crystallography, X-Ray, Biochemistry, Mice, Phosphatidylinositol 3-Kinases, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, In vivo, Cell Line, Tumor, Drug Discovery, Animals, Humans, Structure–activity relationship, Protein Kinase Inhibitors, Molecular Biology, Phosphoinositide-3 Kinase Inhibitors, Ovarian Neoplasms, Binding Sites, Trifluoromethyl, Organic Chemistry, Protein Structure, Tertiary, Rats, Enzyme Activation, Molecular Docking Simulation, Disease Models, Animal, 030104 developmental biology, chemistry, Benzothiazole, 030220 oncology & carcinogenesis, Alkoxy group, Heterografts, Molecular Medicine, Female, Enantiomer, Half-Life
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3
المؤلفون: Alex Aycinena, Yu Ding, Audry Kauffmann, Tatiana Zavorotinskaya, Amy Lambert, John L. Langowski, Julie Chan, Cornelia Bellamacina, Robert Lowell Simmons, Yumin Dai, Min Y. Chen, Christine Fritsch, Gordana Atallah, Elaine Ginn, Victoriano Tamez, Matthew Burger, Kristine Muller, Richard Zang, Paul Feucht, Joseph Castillo, Estelle Pfister, K. Gary Vanasse, Mika Lindvall, Pablo Garcia, Michelle Mathur, Wooseok Han, Gisele Nishiguchi, Jocelyn Holash, Yingyun Wang, Kay Huh, Zhang Yanchen, Steve Basham, Jiong Lan
المصدر: Journal of Medicinal Chemistry. 58:8373-8386
مصطلحات موضوعية: Chemistry, Kinase, Myeloid leukemia, Cancer, medicine.disease, Virology, In vitro, Clinical trial, Leukemia, In vivo, hemic and lymphatic diseases, Drug Discovery, medicine, Cancer research, Molecular Medicine, Multiple myeloma
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4
المؤلفون: Matthew T, Burger, Gisele, Nishiguchi, Wooseok, Han, Jiong, Lan, Robert, Simmons, Gordana, Atallah, Yu, Ding, Victoriano, Tamez, Yanchen, Zhang, Michelle, Mathur, Kristine, Muller, Cornelia, Bellamacina, Mika K, Lindvall, Richard, Zang, Kay, Huh, Paul, Feucht, Tatiana, Zavorotinskaya, Yumin, Dai, Steve, Basham, Julie, Chan, Elaine, Ginn, Alex, Aycinena, Jocelyn, Holash, Joseph, Castillo, John L, Langowski, Yingyun, Wang, Min Y, Chen, Amy, Lambert, Christine, Fritsch, Audry, Kauffmann, Estelle, Pfister, K Gary, Vanasse, Pablo D, Garcia
المصدر: Journal of medicinal chemistry. 58(21)
مصطلحات موضوعية: Models, Molecular, Leukemia, Myeloid, Acute, Mice, Halogenation, Proto-Oncogene Proteins c-pim-1, Cell Line, Tumor, Proto-Oncogene Proteins, Animals, Humans, Protein Serine-Threonine Kinases, Picolinic Acids, Amides, Protein Kinase Inhibitors
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5
المؤلفون: Susan Kaufman, Zhang Yanchen, Joshua Haznedar, Daniel Menezes, Matthew Burger, Xiaohua Xin, Aaron Smith, Frazier Kelly, Sauveur-Michel Maira, Allan S. Wagman, Zhi-Jie Ni, Keith B. Pfister, Kay Huh, Isabel Zaror, Thomas Hendrickson, Joelle Verhagen, Gordana Atallah, Kevin Shoemaker, Bartulis Sarah, Michael Chin, Simon Ng, Kenneth Crawford, Dirksen E. Bussiere, Ed Iwanowicz, Mark Knapp, Isabelle Lee, Hanne Merritt, Marion Wiesmann, Charles Voliva, Sabina Pecchi
المصدر: ACS Medicinal Chemistry Letters. 2:774-779
مصطلحات موضوعية: Phosphoinositide 3-kinase, biology, business.industry, Kinase, Organic Chemistry, Buparlisib, Phases of clinical research, Cancer, Pharmacology, medicine.disease, Biochemistry, chemistry.chemical_compound, chemistry, In vivo, Drug Discovery, biology.protein, Medicine, Signal transduction, business, PI3K/AKT/mTOR pathway
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6
المؤلفون: Victoriano Tamez, Kay Huh, John L. Langowski, Tatiana Zavorotinskaya, Min Y. Chen, Gisele Nishiguchi, Matthew Burger, Zhang Yanchen, Jocelyn Holash, Cornelia Bellamacina, Pablo Garcia, Kristine Muller, Michelle Mathur, Wooseok Han, Jiong Lan, Joseph Castillo, Christopher McBride, Paul Feucht, Mika Lindval, Yu Ding, Yumin Dai, Gordana Atallah, Elizabeth L. Beans, Yingyun Wang
مصطلحات موضوعية: Myeloid, Kinase, Organic Chemistry, Myeloid leukemia, PIM1, Biology, medicine.disease, Biochemistry, Virology, In vitro, Lymphoma, Haematopoiesis, medicine.anatomical_structure, In vivo, hemic and lymphatic diseases, Drug Discovery, medicine, Cancer research
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::944da92389832ca637e9d382159688c5
https://europepmc.org/articles/PMC4027555/ -
7
المؤلفون: Aaron Smith, Matthew Burger, Charles Voliva, Kay Huh, John Chan, Sabina Pecchi, Johanna Janssen, Jiong Lan, Hanne Merritt, Marion Wiesmann, Wooseok Han, Zhi-Jie Ni, Susan Kaufman, Mark Knapp
المصدر: Bioorganicmedicinal chemistry letters. 23(16)
مصطلحات موضوعية: Models, Molecular, Imidazopyridine, Pyridines, Clinical Biochemistry, Cell, Pharmaceutical Science, Imides, Biochemistry, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, Gene duplication, medicine, Humans, Benzothiazoles, Enzyme Inhibitors, Molecular Biology, PI3K/AKT/mTOR pathway, Phosphoinositide-3 Kinase Inhibitors, Chemistry, Kinase, Organic Chemistry, Cancer, medicine.disease, In vitro, Enzyme Activation, medicine.anatomical_structure, Benzothiazole, Solubility, Cancer research, Molecular Medicine, Female, Azo Compounds
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8
المؤلفون: Daniel T. Chu, Mike Langhorne, Kelly Young, Christy Hiebert, Jolene Kidney, J. J. Plattner, Scott Anderson, Georgia Law Carroll, Kay Huh, Mehran Seid, Xiaodong Lin, Alice Rico, Manoj C. Desai, Lynn Barker, Ribhi Shawar, Burger Matthew
المصدر: Journal of medicinal chemistry. 49(5)
مصطلحات موضوعية: Lung Diseases, Male, Ketolides, Staphylococcus aureus, Haemophilus Infections, Vinyl Compounds, Stereochemistry, Streptococcus pyogenes, Telithromycin, Erythromycin, Biological Availability, macromolecular substances, Microbial Sensitivity Tests, Chemical synthesis, Pneumococcal Infections, Rats, Sprague-Dawley, Structure-Activity Relationship, In vivo, Drug Discovery, Drug Resistance, Bacterial, medicine, Enterococcus faecalis, Structure–activity relationship, Animals, Ketolide, Chemistry, organic chemicals, Antimicrobial, Haemophilus influenzae, Anti-Bacterial Agents, Rats, Streptococcus pneumoniae, Molecular Medicine, lipids (amino acids, peptides, and proteins), Antibacterial activity, medicine.drug, Half-Life
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9دورية أكاديمية
المؤلفون: Matthew T. Burger, Gisele Nishiguchi, Wooseok Han, Jiong Lan, Robert Simmons, Gordana Atallah, Yu Ding, Victoriano Tamez, Yanchen Zhang, Michelle Mathur, Kristine Muller, Cornelia Bellamacina, MikaK. Lindvall, Richard Zang, Kay Huh, Paul Feucht, Tatiana Zavorotinskaya, Yumin Dai, Steve Basham, Julie Chan
المصدر: Journal of Medicinal Chemistry; Nov2015, Vol. 58 Issue 21, p8373-8386, 14p
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المؤلفون: Nancy Pryer, Isabelle Lee, Yoko Oei, Kay Huh, Marion Wiesmann, Susan Kaufman, Janet Sim, Tao Wang, Victoria Sung, Lenahan William P, Ursula Jeffry, Dylan Daniel, James Sutton
المصدر: Cancer Research. 70:3629-3629
مصطلحات موضوعية: Cancer Research, Pathology, medicine.medical_specialty, Osteolysis, biology, business.industry, Bone metastasis, Tyrosine phosphorylation, medicine.disease, Receptor tyrosine kinase, Bone resorption, chemistry.chemical_compound, medicine.anatomical_structure, Oncology, Growth factor receptor, chemistry, Osteoclast, medicine, biology.protein, Cancer research, Kinase activity, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::00e7ddf71622c6d195dfbe82cc3a1b0a
https://doi.org/10.1158/1538-7445.am10-3629