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1دورية أكاديمية
المؤلفون: Kelly Bleasby, Robert Houle, Michael Hafey, Meihong Lin, Jingjing Guo, Bing Lu, Rosa I. Sanchez, Kerry L. Fillgrove
المصدر: Viruses, Vol 13, Iss 8, p 1566 (2021)
مصطلحات موضوعية: 4′-ethynyl-2-fluoro-2′-deoxyadenosine (EFdA), islatravir, MK-8591, cytochrome p450, drug–drug interaction, drug transporters, Microbiology, QR1-502
وصف الملف: electronic resource
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المؤلفون: Anthony J. Roecker, Kathy M. Schirripa, H. Marie Loughran, Ling Tong, Tao Liang, Kerry L. Fillgrove, Yuhsin Kuo, Kelly Bleasby, Hannah Collier, Michael D. Altman, Melissa C. Ford, Robert E. Drolet, Mali Cosden, Sarah Jinn, Nathan G. Hatcher, Lihang Yao, Monika Kandebo, Joshua D. Vardigan, Rosemarie B. Flick, Xiaomei Liu, Christina Minnick, Laura A. Price, Marla L. Watt, Wei Lemaire, Christine Burlein, Gregory C. Adam, Lauren A. Austin, Jacob N. Marcus, Sean M. Smith, Mark E. Fraley
المصدر: ACS Medicinal Chemistry Letters. 14:146-155
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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المؤلفون: Grace Chan, Kelly Bleasby, Raymond Evers, Xiaoyan Chu, Irene Nunes
المصدر: Clinical Pharmacology & Therapeutics. 100:437-440
مصطلحات موضوعية: 0301 basic medicine, Drug, Drug-Related Side Effects and Adverse Reactions, Organic Cation Transport Proteins, media_common.quotation_subject, Renal function, Pharmacology, Models, Biological, behavioral disciplines and activities, 030226 pharmacology & pharmacy, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Animals, Humans, Medicine, Pharmacology (medical), media_common, Creatinine, Kidney, Organic cation transport proteins, biology, urogenital system, business.industry, Acute kidney injury, Transporter, Acute Kidney Injury, medicine.disease, 030104 developmental biology, medicine.anatomical_structure, chemistry, biology.protein, Biomarker (medicine), business, Biomarkers
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المؤلفون: Kerry L. Fillgrove, Grace Chan, Rosa I. Sanchez, Meihong Lin, Bing Lu, Deborah J. Newton, Robert Houle, Jairam Palamanda, Kelly Bleasby
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, 0303 health sciences, Organic anion transporter 1, biology, CYP3A4, Abcg2, 030306 microbiology, Chemistry, CYP1A2, Transporter, 030226 pharmacology & pharmacy, Antiviral Agents, In vitro, Organic anion-transporting polypeptide, 03 medical and health sciences, 0302 clinical medicine, Infectious Diseases, Enzyme, Biochemistry, biology.protein, Pharmacology (medical)
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0f76b0224ecf19334aa1e470533a76d3
https://europepmc.org/articles/PMC6437506/ -
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المؤلفون: Xiaoyan Chu, Raymond Evers, Kelly Bleasby
المصدر: Expert Opinion on Drug Metabolism & Toxicology. 9:237-252
مصطلحات موضوعية: Drug, Organic Cation Transport Proteins, Abcg2, media_common.quotation_subject, Drug Evaluation, Preclinical, Organic Anion Transporters, ATP-binding cassette transporter, Pharmacology, Toxicology, Absorption, Species Specificity, Pharmacokinetics, Animals, Humans, Distribution (pharmacology), Drug Interactions, Tissue Distribution, ATP Binding Cassette Transporter, Subfamily B, Member 1, media_common, biology, Biological Transport, Transporter, General Medicine, Multiple drug resistance, Disease Models, Animal, biology.protein, ATP-Binding Cassette Transporters, Efflux
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المؤلفون: Maria Madeira, Wendy D. Cornell, Andreas Verras, Robert P. Sheridan, William K. Hagmann, Edward C. Sherer, Drew Roberts, Kelly Bleasby
المصدر: Molecular Informatics. 31:231-245
مصطلحات موضوعية: Quantitative structure–activity relationship, Molecular model, Chemistry, business.industry, Organic Chemistry, Cross prediction, Computer Science Applications, Random forest, Passive permeability, Structural Biology, Permeability (electromagnetism), Drug Discovery, Line (geometry), Molecular Medicine, Artificial intelligence, business, Biological system, ADME
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المؤلفون: Thomas H. Graham, Urmi R. Bhatt, Dong-Ming Shen, Xinchun Tong, Mike E. Lassman, Kelly Bleasby, Dan Xie, Qing Chen, Shirly Pinto, Margarita Garcia-Calvo, Andreas Verras, Renee M. Chabin, Zhicai Wu, Steven L. Colletti, Suoyu Xu, Cangming Yang, James R. Tata, Zhu Shen, Ranabir SinhaRoy, Jeffrey J. Hale
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:1727-1730
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Carboxypeptidases, Pharmacology, Biochemistry, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, Enzyme activator, chemistry.chemical_compound, Heterocyclic Compounds, Drug Discovery, Animals, Inhibitory concentration 50, Structure–activity relationship, Amines, Enzyme Inhibitors, Molecular Biology, Molecular Structure, Chemistry, Drug discovery, Organic Chemistry, Brain, Amides, Enzyme Activation, Molecular Medicine, Penetrant (biochemical)
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المؤلفون: Raymond Evers, Xiaoyan Chu, Kelly Bleasby, Irene Nunes, Grace Chan
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 44(9)
مصطلحات موضوعية: 0301 basic medicine, medicine.medical_specialty, Organic anion transporter 1, Cmax, Pharmaceutical Science, Renal function, Organic Anion Transporters, Sodium-Independent, Kidney, Kidney Function Tests, 030226 pharmacology & pharmacy, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Internal medicine, medicine, Humans, Pharmacology, Creatinine, biology, Acute kidney injury, Kidney metabolism, Organic Cation Transporter 2, medicine.disease, 030104 developmental biology, medicine.anatomical_structure, Endocrinology, Elevated serum creatinine, chemistry, Drug Design, biology.protein, Biomarkers
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ccb0a71e78a8b1f3c53258f8aa7753b9
https://pubmed.ncbi.nlm.nih.gov/26825641 -
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المؤلفون: Kelly Bleasby, Dwight Macdonald, Bruce Mackay, Richard Tschirret-Guth, Robert Houle, Sebastien Laliberte, Patrick Lacombe, Robert Papp, Erich L. Grimm, Amandine Chefson, Jean-François Lévesque, Michael J. Hafey, Pierre-André Fournier, Sébastien Gagné, Yongxin Han, Yves Ducharme, Michel Gallant, Austin Chen, Daniel Dube
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:5547-5551
مصطلحات موضوعية: ATP Binding Cassette Transporter, Subfamily B, Cell Membrane Permeability, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmaceutical Science, ATP-binding cassette transporter, Absorption (skin), Pharmacology, Biochemistry, Mice, Structure-Activity Relationship, Piperidines, Renin, Drug Discovery, Renin–angiotensin system, Animals, Structure–activity relationship, Molecular Biology, Mice, Knockout, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Biological Transport, Stereoisomerism, Transporter, Rats, Bioavailability, Permeability (electromagnetism), Molecular Medicine, Efflux
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المؤلفون: Kelly Bleasby, Yui Sing Tang, Emmanuel O. Nketiah, Lauren Smith, Margaret E. McCann, Feroze Ujjainwalla, Brande S. Williams, Michael J. Hafey, Jessica Aijia Liu, Gregory J. Kaczorowski, William A. Schmalhofer, Joseph F. Leone, Matthew P. Braun, Lindsey Beers, Anu Thomas, Martin Köhler, Maria L. Garcia, Adam B. Weinglass
المصدر: Molecular Pharmacology. 73:1072-1084
مصطلحات موضوعية: medicine.drug_class, Pharmacology, Transfection, Tritium, beta-Lactams, Cell Line, chemistry.chemical_compound, Dogs, Ezetimibe, medicine, Animals, Humans, Cholesterol absorption inhibitor, Cloning, Molecular, Sulfonamides, biology, Cholesterol, Membrane Proteins, Membrane Transport Proteins, Reproducibility of Results, Sitosterols, Biochemistry, chemistry, Caco-2, Cell culture, HMG-CoA reductase, biology.protein, Azetidines, Molecular Medicine, Lovastatin, Caco-2 Cells, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0fee59cbd56dba6e1cebfc2f3a19d052
https://doi.org/10.1124/mol.107.043844