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المؤلفون: Tatsuhiko Fujimoto, Kentaro Rikimaru, Koichiro Fukuda, Hiromichi Sugimoto, Kei Masuda, Norio Ohyabu, Yoshihiro Banno, Norihito Tokunaga, Tetsuji Kawamoto, Yoshihide Tomata, Yasumi Kumagai, Motoo Iida, Yoichi Nagano, Mariko Yoneyama-Hirozane, Yuji Shimizu, Katsunori Sasa, Takashi Ishikawa, Hiroshi Yukitake, Mitsuhiro Ito, Kazunobu Aoyama, Takahiro Matsumoto
المصدر: ACS Medicinal Chemistry Letters. 13:457-462
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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3Sanitize It Yourself: human-based sanitization checker against machine-generated chemical structures
المؤلفون: Naruki Yoshikawa, Kentaro Rikimaru, Kazuki Yamamoto
مصطلحات موضوعية: Computer engineering, Computer science, business.industry, Deep learning, Human computation, Computer Aided Design, Web application, Artificial intelligence, business, computer.software_genre, computer, Chemical space
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::850a7645eb0e22d91c7dac460ad829e7
https://doi.org/10.33774/chemrxiv-2021-9nhm1 -
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المصدر: IPSJ Transactions on Bioinformatics. 11:41-47
مصطلحات موضوعية: 0301 basic medicine, Computer science, business.industry, Machine learning, computer.software_genre, 01 natural sciences, Biochemistry, Genetics and Molecular Biology (miscellaneous), 0104 chemical sciences, Computer Science Applications, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, 030104 developmental biology, Lead (geology), Learning to rank, Artificial intelligence, business, computer
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::e95690dde551846f63e30d20d9caa062
https://doi.org/10.2197/ipsjtbio.11.41 -
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المؤلفون: Motohisa Suzuki, Atsushi Suzuki, Hiroshi Yukitake, Haruhide Kimura, Mitsuhiro Ito, Tatsuhiko Fujimoto, Yuji Shimizu, Kentaro Rikimaru, T Ishikawa
المصدر: Pharmacology Biochemistry and Behavior. 187:172794
مصطلحات موضوعية: Male, Agonist, medicine.medical_specialty, Lateral hypothalamus, medicine.drug_class, Clinical Biochemistry, CHO Cells, Transfection, Toxicology, Biochemistry, Mice, 03 medical and health sciences, Behavioral Neuroscience, Cricetulus, 0302 clinical medicine, Orexin Receptors, Internal medicine, medicine, Animals, Humans, Wakefulness, Receptor, Biological Psychiatry, Narcolepsy, Mice, Knockout, Neurons, Pharmacology, Orexins, Chemistry, Histaminergic, medicine.disease, 030227 psychiatry, Orexin, Mice, Inbred C57BL, Endocrinology, medicine.anatomical_structure, Hypothalamic Area, Lateral, Sleep, Tuberomammillary nucleus, 030217 neurology & neurosurgery
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المؤلفون: Kentaro Rikimaru, Kenjiro Sato, Hirohisa Miyashita, Toshiki Murata, Tomoyuki Odani, Yoshiyuki Tsujihata, Hiroshi Imoto, Hiromichi Sugimoto, Nobuyuki Negoro, Masahiro Kamaura
المصدر: Bioorganic & Medicinal Chemistry. 22:1649-1666
مصطلحات موضوعية: Carbamate, Indoles, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Receptors, G-Protein-Coupled, Structure-Activity Relationship, chemistry.chemical_compound, Oral administration, Drug Discovery, medicine, Animals, Hypoglycemic Agents, Gpr119 agonist, Molecular Biology, G protein-coupled receptor, Molecular Structure, Organic Chemistry, Glucose Tolerance Test, Rats, GPR119, chemistry, Indoline, Molecular Medicine, Lead compound, Methyl group
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المؤلفون: Yoshiaki Horiguchi, Kenneth A. Bragstad, Clifford D. Mol, Tsuyoshi Maekawa, Junichi Sakamoto, Takeshi Wakabayashi, Nozomi Katayama, Chisako Nomura, Mitsuharu Matsumoto, Hidenori Abe, Kentaro Rikimaru, Miyuki Funami, Takanori Matsuo, Kazutoshi Kawakami, Hiroko Tsuge, Katsuhito Murase, Bi-Ching Sang, Gyorgy Snell, Hiroshi Imoto, Naoto Arimura, Osamu Ujikawa, Toshimasa Tanaka, Douglas R. Dougan, Yu Momose
المصدر: Bioorganic & Medicinal Chemistry. 20:714-733
مصطلحات موضوعية: Agonist, medicine.drug_class, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Carboxylic Acids, Pharmaceutical Science, Peroxisome proliferator-activated receptor, Biochemistry, Diabetes Mellitus, Experimental, Drug Discovery, medicine, Animals, Humans, Hypoglycemic Agents, Moiety, Computer Simulation, Thiazolidinedione, Molecular Biology, chemistry.chemical_classification, Sulfonyl, Sulfonamides, Binding Sites, Organic Chemistry, Protein Structure, Tertiary, Rats, PPAR gamma, Disease Models, Animal, chemistry, Docking (molecular), Drug Design, Pyrazoles, Molecular Medicine, Thiazolidinediones, Binding domain
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المؤلفون: Kentaro Rikimaru, Toshiyuki Kan, Kazuki Mori, Tohru Fukuyama
المصدر: Chem. Commun.. :394-396
مصطلحات موضوعية: Aza Compounds, Molecular Structure, Chemistry, Stereochemistry, Isocyanide, Metals and Alloys, Stereoisomerism, General Medicine, General Chemistry, Skeleton (category theory), Catalysis, Surfaces, Coatings and Films, Electronic, Optical and Magnetic Materials, Bridged Bicyclo Compounds, chemistry.chemical_compound, Tetrahydroisoquinolines, Intramolecular force, Materials Chemistry, Ceramics and Composites, Organic chemistry, Stereoselectivity, Lemonomycin
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7650545b21f16d8a5e179ca3f4546948
https://doi.org/10.1039/b415030a -
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المؤلفون: Tohru Fukuyama, Kentaro Rikimaru, Kazuki Mori, Toshiyuki Kan
المصدر: Organic Letters. 6:3095-3097
مصطلحات موضوعية: Molecular Structure, Chemistry, Stereochemistry, Organic Chemistry, Convergent synthesis, Stereoisomerism, Key features, Biochemistry, Catalysis, Hydroboration, chemistry.chemical_compound, Cyclization, Naphthyridinomycin, Intramolecular force, Indicators and Reagents, Amine gas treating, Stereoselectivity, Naphthyridines, Physical and Theoretical Chemistry, Derivative (chemistry)
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المؤلفون: Taisuke Tomita, Toshiyuki Kan, Hideaki Natsugari, Yusuke Tominari, Takeshi Iwatsubo, Tohru Fukuyama, Yuichi Morohashi, Kentaro Rikimaru
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:1983-1985
مصطلحات موضوعية: Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Benzophenones, chemistry.chemical_compound, Amide, Endopeptidases, Drug Discovery, Peptide synthesis, medicine, Protease Inhibitors, Molecular Biology, Dipeptide, Molecular Structure, biology, Organic Chemistry, Dipeptides, Condensation reaction, Amides, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Epimer, Amyloid Precursor Protein Secretases