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1دورية أكاديمية
المؤلفون: Adam O. Whelan, Ian Cooper, Nicola Ooi, David Orr, Kevin Blades, James Kirkham, Amanda Lyons, Kay B. Barnes, Mark I. Richards, Anne-Marie Salisbury, Mark Craighead, Sarah V. Harding
المصدر: Antibiotics, Vol 12, Iss 6, p 983 (2023)
مصطلحات موضوعية: topoisomerase inhibitors, in vitro activity, biothreat, Burkholderia pseudomallei, Francisella tularensis, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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2
المؤلفون: Alex Swann, Roger Tan, Matthew Harper, Kevin Blades, Zacharia Joseph, Nicholas Calvert, Michael Salmon, Piers Yates
المصدر: J Orthop
مصطلحات موضوعية: 030222 orthopedics, medicine.medical_specialty, Blood management, Blood transfusion, business.industry, medicine.medical_treatment, 030229 sport sciences, Pain management, Functional recovery, Arthroplasty, Article, Surgery, 03 medical and health sciences, 0302 clinical medicine, Enhanced recovery, Cohort, Surgical site, medicine, Orthopedics and Sports Medicine, business
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3
المؤلفون: Amanda Lyons, James Kirkham, Kevin Blades, David Orr, Elizabeth Dauncey, Oliver Smith, Emma Dick, Rolf Walker, Teresa Matthews, Adam Bunt, Jonathan Finlayson, Ian Morrison, Victoria J. Savage, Emmanuel Moyo, Hayley S. Butler, Rebecca Newman, Nicola Ooi, Andrew Smith, Cédric Charrier, Andrew J. Ratcliffe, Neil R. Stokes, Stuart Best, Anne-Marie Salisbury, Mark Craighead, Ian R. Cooper
المصدر: Bioorganicmedicinal chemistry letters. 65
مصطلحات موضوعية: Topoisomerase Inhibitors, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Microbial Sensitivity Tests, Biochemistry, Anti-Bacterial Agents, Mice, Structure-Activity Relationship, DNA Gyrase, Drug Discovery, Molecular Medicine, Animals, Topoisomerase II Inhibitors, Molecular Biology, Oxazolidinones, Fluoroquinolones
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4
المؤلفون: Philip J. Jewsbury, Rajesh Odedra, Alan Lau, Sylvie Guichard, James W.T. Yates, Kevin Blades, Gary Wilkinson, Kevin Michael Foote, Dan Heathcote, Turner Paul, Christine M. Wood, J. Willem M. Nissink, Zena Wilson, Thomas M. McGuire
المصدر: Journal of Medicinal Chemistry. 61:9889-9907
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Indoles, Chemical Phenomena, Morpholines, Molecular Conformation, Regulator, Antineoplastic Agents, Context (language use), Ataxia Telangiectasia Mutated Proteins, Mice, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, Cell Line, Tumor, Drug Discovery, Animals, Humans, Tissue Distribution, Protein Kinase Inhibitors, Clinical Trials as Topic, Sulfonamides, CYP3A4, Kinase, Drug discovery, Pyrimidines, 030104 developmental biology, chemistry, Cell culture, Sulfoxides, 030220 oncology & carcinogenesis, Cancer research, Molecular Medicine, Female, DNA
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5
المؤلفون: Steven C. Glossop, Kevin Blades
المصدر: Synthesis. 49:554-556
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Stereochemistry, Heck reaction, Organic Chemistry, Key (cryptography), 010402 general chemistry, 01 natural sciences, Protocol (object-oriented programming), Catalysis, 0104 chemical sciences
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::8ecbc187a981be7817d11cc2f54b3e20
https://doi.org/10.1055/s-0036-1588364 -
6
المؤلفون: Gordon S. Currie, Kurt Gordon Pike, Janet D. Culshaw, Martin Pass, Kristy Gill, M. Raymond V. Finlay, Stuart E. Pearson, Jonathan M. Eden, Craig A. Roberts, Linette Ruston, Kevin Blades, Sarah L. Pass, Catherine Good, Ryan Greenwood, Morris Jeffrey James, Julie Demeritt, Emma J. Williams
المصدر: Journal of Medicinal Chemistry. 58:2326-2349
مصطلحات موضوعية: Models, Molecular, Molecular Structure, Chemistry, Drug discovery, TOR Serine-Threonine Kinases, High-throughput screening, Thiourea, Mechanistic Target of Rapamycin Complex 2, mTORC1, Mechanistic Target of Rapamycin Complex 1, Combinatorial chemistry, mTORC2, Chemical space, Structure-Activity Relationship, Pyrimidines, Multiprotein Complexes, Drug Discovery, Hepatocytes, Humans, Molecular Medicine, Potency, Structure–activity relationship, Solubility, Protein Kinase Inhibitors, Cells, Cultured
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7
المؤلفون: Nicholas J. Howe, Kevin Blades, Gillian M. Lamont
المصدر: Synlett. 26:228-232
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, Scaffold, chemistry, Aryl, Organic Chemistry, Hydrazine, Lactam, Pyrazole, Ring (chemistry), Combinatorial chemistry, Dieckmann condensation, Alkyl
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::179cdfc16f78b2d8573cc6b3d9fb0228
https://doi.org/10.1055/s-0034-1379504 -
8
المؤلفون: Kevin Blades, Piers Yates, Michael Kent, Nick Calvert, Alex Swann
مصطلحات موضوعية: musculoskeletal diseases, 030222 orthopedics, medicine.medical_specialty, Blood transfusion, Revision arthroplasty, business.industry, medicine.medical_treatment, Incidence (epidemiology), Revision hip replacement, Outcome measures, Arthroplasty, Article, Surgery, 03 medical and health sciences, 0302 clinical medicine, Enhanced recovery, Pain control, Anesthesia, medicine, Orthopedics and Sports Medicine, 030212 general & internal medicine, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::89081a90ad955c30ca89c96fa2962e49
https://europepmc.org/articles/PMC5581381/ -
9
المؤلفون: William McCoull, Roman D. Abrams, Erica Anderson, Kevin Blades, Peter Barton, Matthew Box, Jonathan Burgess, Kate Byth, Qing Cao, Claudio Chuaqui, Rodrigo J. Carbajo, Tony Cheung, Erin Code, Andrew D. Ferguson, Shaun Fillery, Nathan O. Fuller, Eric Gangl, Ning Gao, Matthew Grist, David Hargreaves, Martin R. Howard, Jun Hu, Paul D. Kemmitt, Jennifer E. Nelson, Nichole O’Connell, D. Bryan Prince, Piotr Raubo, Philip B. Rawlins, Graeme R. Robb, Junjie Shi, Michael J. Waring, David Whittaker, Marta Wylot, Xiahui Zhu
المصدر: Journal of medicinal chemistry. 60(14)
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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المؤلفون: Jennifer E. Nelson, Graeme R. Robb, Martin R. Howard, Piotr Raubo, Paul D. Kemmitt, Kevin Blades, Junjie Shi, Tony Cheung, Qing Cao, Peter Barton, Andrew D. Ferguson, D. Bryan Prince, Shaun M. Fillery, Jun Hu, David J. Hargreaves, Roman D. Abrams, Nathan O. Fuller, Claudio Chuaqui, Eric Gangl, Matthew R. Box, Ning Gao, William McCoull, Kate Byth, Michael J. Waring, Jonathan Burgess, Xiahui Zhu, Matthew Grist, Erica Anderson, Nichole O'Connell, Philip B. Rawlins, Marta Wylot, David Whittaker, Rodrigo J. Carbajo, Erin Code
المصدر: Journal of medicinal chemistry. 60(10)
مصطلحات موضوعية: 0301 basic medicine, Pyrimidine, Pyridines, 03 medical and health sciences, chemistry.chemical_compound, immune system diseases, hemic and lymphatic diseases, Cell Line, Tumor, Drug Discovery, medicine, Transferase, Potency, Humans, Protein Interaction Maps, B-cell lymphoma, Cell Proliferation, Chemistry, Kinase, medicine.disease, BCL6, Combinatorial chemistry, Lymphoma, Molecular Docking Simulation, 030104 developmental biology, Biochemistry, Cell culture, Drug Design, Proto-Oncogene Proteins c-bcl-6, Molecular Medicine, Pyrazoles, Lymphoma, Large B-Cell, Diffuse