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1
المؤلفون: Gary E. Zurenko, Betty H. Yagi, Douglas K Hutchinson, D E Emmert, David R. Graber, Jackson B. Hester, Stuart A. Garmon, Judith C. Hamel, Michael R Barbachyn, Ronda D. Schaadt, Michael J. Genin, Douglas Stapert, Joel Morris, David J. Anderson, Debra A. Allwine, R J Reischer, Charles W. Ford, Kevin C. Grega
المصدر: Journal of Medicinal Chemistry. 43:953-970
مصطلحات موضوعية: Azoles, Stereochemistry, Triazole, Administration, Oral, Microbial Sensitivity Tests, Pyrazole, medicine.disease_cause, Haemophilus influenzae, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Eperezolid, Animals, Humans, Organic chemistry, Oxazoles, Moraxella, Antibacterial agent, chemistry.chemical_classification, biology, biology.organism_classification, Anti-Bacterial Agents, chemistry, Molecular Medicine, Azole, Methicillin Resistance, Antibacterial activity, Moraxella catarrhalis
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2
المؤلفون: Ford Charles W, Robert A. Conradi, Jenifer L. Adamski, Randy M. Jensen, Debra A. Allwine, Barbachyn Michael R, John A. Tucker, Gary E. Zurenko, Jennifer L. Klock, Hutchinson Douglas K, Steven J. Brickner, Phillip S. Burton, Kevin C. Grega
المصدر: Journal of Medicinal Chemistry. 41:3727-3735
مصطلحات موضوعية: Staphylococcus aureus, Pyrimidine, Pyridines, Stereochemistry, Microbial Sensitivity Tests, Chemical synthesis, Permeability, Piperazines, Pyridazine, Structure-Activity Relationship, chemistry.chemical_compound, Morpholine, Acetamides, Drug Discovery, Enterococcus faecalis, Eperezolid, Humans, Triazene, Oxazoles, Oxazolidinones, Antibacterial agent, Linezolid, Staphylococcal Infections, Anti-Bacterial Agents, Piperazine, Streptococcus pneumoniae, chemistry, Molecular Medicine, Methicillin Resistance, Caco-2 Cells, Triazenes
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3
المؤلفون: Betty H. Yagi, Suzanne E. Glickman, Susan K. Hendges, Ford Charles W, Toops Dana S, Jonda D. Schaadt, Barbachyn Michael R, Douglas Stapert, Kevin C. Grega, Jerry M. Buysse, Judith C. Hamel, James O. Kilburn, Gary E. Zurenko, William F. Demyan
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:1009-1014
مصطلحات موضوعية: Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, chemistry.chemical_element, Ring (chemistry), Biochemistry, Combinatorial chemistry, In vitro, chemistry.chemical_compound, Meta, chemistry, In vivo, Drug Discovery, Fluorine, Molecular Medicine, Tropone, Antibacterial activity, Molecular Biology
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4
المؤلفون: Sally P. Klemens, Toops Dana S, James O. Kilburn, Susan K. Hendges, Ford Charles W, S. E. Glickman, Gary E. Zurenko, Kevin C. Grega, Steven J. Brickner, Michael H. Cynamon, Hutchinson Douglas K, Barbachyn Michael R
المصدر: Journal of Medicinal Chemistry. 39:680-685
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, medicine.drug_class, SQ109, Microbial Sensitivity Tests, Pharmacology, Antimycobacterial, Mass Spectrometry, Mycobacterium tuberculosis, chemistry.chemical_compound, In vivo, Acetamides, Drug Discovery, medicine, Eperezolid, Animals, Oxazoles, Antibacterial agent, biology, Chemistry, Isoniazid, Biological activity, biology.organism_classification, Anti-Bacterial Agents, Rats, Molecular Medicine, Mycobacterium avium, medicine.drug
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5
المؤلفون: Susan K. Hendges, Toops Dana S, Hutchinson Douglas K, Manninen Peter Rudolph, Barbachyn Michael R, Gary E. Zurenko, Stuart A. Garmon, Steven J. Brickner, Ford Charles W, Kevin C. Grega, Debra A. Ulanowicz
المصدر: Journal of Medicinal Chemistry. 39:673-679
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, medicine.drug_class, Antibiotics, Microbial Sensitivity Tests, medicine.disease_cause, Mass Spectrometry, Microbiology, Mice, chemistry.chemical_compound, Dogs, Antibiotic resistance, Anti-Infective Agents, Acetamides, Drug Discovery, medicine, Eperezolid, Animals, Oxazoles, Oxazolidinones, Antibacterial agent, Linezolid, Drug Resistance, Microbial, Combinatorial chemistry, Drug Resistance, Multiple, Rats, Multiple drug resistance, chemistry, Staphylococcus aureus, Molecular Medicine, Vancomycin, Female, Antibacterial activity, medicine.drug
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6
المصدر: The Journal of Organic Chemistry. 60:5255-5261
مصطلحات موضوعية: Chemistry, Metalation, Organic Chemistry, Regioselectivity, Combinatorial chemistry
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7
المصدر: ChemInform. 26
مصطلحات موضوعية: Metalation, Chemistry, Organic chemistry, Regioselectivity, General Medicine, Combinatorial chemistry
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8
المؤلفون: Betty H. Yagi, Kevin C. Grega, Ronda D. Schaadt, W. F. Demyan, Toops Dana S, Gary E. Zurenko, Steven J. Brickner, J. O. Kilburn, Barbachyn Michael R, Debra A. Ulanowicz, Ford Charles W, S. E. Glickman, Judith C. Hamel, J. M. Buysse, Douglas Stapert
المصدر: ChemInform. 27
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Substitution (logic), Identification (biology), General Medicine, Tropone, Antibacterial activity, Combinatorial chemistry
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9
المؤلفون: Susan K. Hendges, Kevin C. Grega, Hutchinson Douglas K, Gary E. Zurenko, Manninen Peter Rudolph, Toops Dana S, Stuart A. Garmon, Ford Charles W, Steven J. Brickner, Debra A. Ulanowicz, Barbachyn Michael R
المصدر: ChemInform. 27
مصطلحات موضوعية: biology, Chemistry, medicine.drug_class, Antibiotics, General Medicine, biology.organism_classification, Microbiology, Multiple drug resistance, Mycobacterium tuberculosis, Antibiotic resistance, Mechanism of action, In vivo, medicine, Vancomycin, medicine.symptom, Antibacterial activity, medicine.drug
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10
المؤلفون: Michael H. Cynamon, Steven J. Brickner, Susan K. Hendges, Sally P. Klemens, Hutchinson Douglas K, Gary E. Zurenko, James O. Kilburn, S. E. Glickman, Barbachyn Michael R, Kevin C. Grega, Ford Charles W, Toops Dana S
المصدر: ChemInform. 27
مصطلحات موضوعية: Tuberculosis, biology, Chemistry, medicine.drug_class, Antibiotics, Isoniazid, General Medicine, Pharmacology, biology.organism_classification, medicine.disease, Antimycobacterial, In vitro, Mycobacterium tuberculosis, In vivo, medicine, Antibacterial agent, medicine.drug