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المؤلفون: Sebastien Andre Campos, Sorif Uddin, Daniel Thomas, Paul Rowland, Birgit Duempelfeld, Douglas W. Thomson, Andrew Sharpe, James E. Rowedder, Kenneth David Down, Máire A. Convery, Augustin Amour, Michael Daniel Goldsmith, Grant A. McGonagle, David N. Mallett, Edith M. Hessel, Jana Krause, Kevin James Doyle, J. Nicole Hamblin, Srividya Sriskantharajah, Edward P. Cannons, Vipulkumar Kantibhai Patel, Chris D. Edwards, Cole Clissold, Nick Barton, Anderson Niall Andrew, John J. Coward
المصدر: Journal of medicinal chemistry. 64(18)
مصطلحات موضوعية: Male, Class I Phosphatidylinositol 3-Kinases, Crystallography, X-Ray, chemistry.chemical_compound, Structure-Activity Relationship, Pharmacokinetics, Drug Discovery, Potency, Animals, Rats, Wistar, Phosphoinositide-3 Kinase Inhibitors, chemistry.chemical_classification, Mice, Inbred BALB C, Sulfonamides, Molecular Structure, Glutathione, Highly selective, Combinatorial chemistry, Sulfonamide, Bioavailability, chemistry, Molecular Medicine, Amine gas treating, Female, Selectivity, Protein Binding
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المؤلفون: Kevin James Doyle, Amanda Van de Poël, Helena Käck, Samantha Jayne Hughes, Hans Lönn, Nicholas John Palmer, Michael S. Bodnarchuk
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Nitrile, Stereochemistry, Organic Chemistry, Drug Discovery, Potency, Biochemistry, Pyrrolidine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ec722f2da594ec7527fb9b43258631f0
https://europepmc.org/articles/PMC6691682/ -
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المؤلفون: Göran Dahl, Amanda Van de Poël, James Root, Steve Swallow, Philip Gardiner, Hans Lönn, Cecilia Wikell, Helena Käck, Kevin James Doyle, Kristina Stenvall, Petra Johannesson, Stephen Connolly
المصدر: Journal of medicinal chemistry. 59(20)
مصطلحات موضوعية: 0301 basic medicine, Administration, Oral, 01 natural sciences, Cathepsin C, 03 medical and health sciences, Mice, Structure-Activity Relationship, Dogs, Drug Discovery, Structure–activity relationship, Animals, Humans, Protease Inhibitors, Benzoxazoles, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Drug discovery, U937 Cells, Combinatorial chemistry, 0104 chemical sciences, Rats, 010404 medicinal & biomolecular chemistry, Oxazepines, 030104 developmental biology, Covalent bond, Molecular Medicine, Rabbits, Once daily