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المؤلفون: Richard L. Mackman, Rao Kalla, Darius Babusis, Jared Pitts, Kimberly T. Barrett, Kwon Chun, Venice Du Pont, Lauren Rodriguez, Jasmine Moshiri, Yili Xu, Michael Lee, Gary Lee, Blake Bleier, Anh-Quan Nguyen, B. Michael O’Keefe, Andrea Ambrosi, Meredith Cook, Joy Yu, Elodie Dempah, Elaine Bunyan, Nicholas C. Riola, Xianghan Lu, Renmeng Liu, Ashley Davie, Tien-Ying Hsiang, Michael Gale, Anita Niedziela-Majka, Joy Y. Feng, Charlotte Hedskog, John P. Bilello, Raju Subramanian, Tomas Cihlar
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::f124f071d22852c94170b2ccfc17e415
https://doi.org/10.1101/2023.04.28.538473 -
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المؤلفون: Michel Perron, Xiaofeng Zhao, Richard L. Mackman, Robert Jordan, Daniel Byun, Raju Subramanian, Tomas Cihlar, Kwon Soo Chun, Diane Lye, Christopher A. Palmiotti, Darius Babusis, Hui Hon Chung, Scott Simonovich, Bin Ma, Sarah Wortman, Lijun Zhang, Gary Lee, Julie Chan, Maria M. Toteva, Eisuke Murakami, Kirsten M. Stray, Xianghan Lu, Jared Pitts, Dustin Siegel, John P. Bilello, Kimberly T. Barrett, Bindu Goyal, Cynthia Kim, Arya Vijjapurapu, Venice Du Pont, Adelle Vandersteen
المصدر: Journal of Medicinal Chemistry. 64:5001-5017
مصطلحات موضوعية: Chemistry, viruses, Metabolite, Phenotypic screening, respiratory system, Prodrug, Virology, Virus, In vitro, chemistry.chemical_compound, In vivo, Drug Discovery, Molecular Medicine, African Green Monkey, Viral load
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المؤلفون: Alexandra Schäfer, David R. Martinez, John J. Won, Rita M. Meganck, Fernando R. Moreira, Ariane J. Brown, Kendra L. Gully, Mark R. Zweigart, William S. Conrad, Samantha R. May, Stephanie Dong, Rao Kalla, Kwon Chun, Venice Du Pont, Darius Babusis, Jennifer Tang, Eisuke Murakami, Raju Subramanian, Kimberly T. Barrett, Blake J. Bleier, Roy Bannister, Joy Y. Feng, John P. Bilello, Tomas Cihlar, Richard L. Mackman, Stephanie A. Montgomery, Ralph S. Baric, Timothy P. Sheahan
المصدر: bioRxiv
article-version (status) pre
article-version (number) 3مصطلحات موضوعية: Parents, Adenosine, Alanine, SARS-CoV-2, Nucleosides, General Medicine, Antiviral Agents, Adenosine Monophosphate, Article, COVID-19 Drug Treatment, Mice, Animals, Humans, Prodrugs, Coronavirus Infections
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::414bac2018cc4bd1b40a45769213931b
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المؤلفون: Jennifer Tang, Timothy P. Sheahan, Stephanie A. Montgomery, Kendra Gully, John J. Won, Ariane J. Brown, Tomas Cihlar, Joy Y. Feng, Ralph S. Baric, Fernanado R Moreira, Kimberly T Barrett, Eisuke Murakami, Roy Bannister, Raju Subramanian, John P. Bilello, Richard L. Mackman, Darius Babusis, Venice Du Pont, Rao Kalla, David R. Martinez, Blake J. Bleier, Kwon Soo Chun, Alexandra Schäfer
مصطلحات موضوعية: Vaccination, business.industry, medicine.drug_class, Oral administration, Cell culture, In vivo, Immunology, Medicine, Prodrug, business, Monoclonal antibody, Nucleoside, Viral load
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6ce6015bc48077307a089bd765f513bb
https://doi.org/10.1101/2021.09.13.460111 -
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المؤلفون: Richard L, Mackman, Hon C, Hui, Michel, Perron, Eisuke, Murakami, Christopher, Palmiotti, Gary, Lee, Kirsten, Stray, Lijun, Zhang, Bindu, Goyal, Kwon, Chun, Daniel, Byun, Dustin, Siegel, Scott, Simonovich, Venice, Du Pont, Jared, Pitts, Darius, Babusis, Arya, Vijjapurapu, Xianghan, Lu, Cynthia, Kim, Xiaofeng, Zhao, Julie, Chan, Bin, Ma, Diane, Lye, Adelle, Vandersteen, Sarah, Wortman, Kimberly T, Barrett, Maria, Toteva, Robert, Jordan, Raju, Subramanian, John P, Bilello, Tomas, Cihlar
المصدر: Journal of medicinal chemistry. 64(8)
مصطلحات موضوعية: Male, Alanine, Drug Evaluation, Preclinical, Epithelial Cells, Respiratory Syncytial Virus Infections, Viral Load, Antiviral Agents, Adenosine Monophosphate, Tubercidin, Rats, Sprague-Dawley, Disease Models, Animal, Macaca fascicularis, Structure-Activity Relationship, Dogs, Respiratory Syncytial Virus, Human, Chlorocebus aethiops, Animals, Humans, Prodrugs, Tissue Distribution, Caco-2 Cells, Cells, Cultured
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المصدر: Nature
مصطلحات موضوعية: Molecular switch, Quantitative Biology::Biomolecules, Multidisciplinary, Molecular Structure, Rotation, Chemistry, Stereochemistry, Diastereomer, Enantioselective synthesis, Stereoisomerism, Bromine, Article, Carbon, Catalysis, Stereocenter, Kinetics, Pharmaceutical Preparations, Benzamides, Molecule, Thermodynamics, Enantiomer, Chirality (chemistry), Isomerization
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المؤلفون: Scott J. Miller, Kimberly T. Barrett
المصدر: Journal of the American Chemical Society. 135:2963-2966
مصطلحات موضوعية: Tertiary amine, Chemistry, Enantioselective synthesis, Regioselectivity, Halogenation, Stereoisomerism, General Chemistry, Electrophilic aromatic substitution, Bromine, Biochemistry, Article, Catalysis, Colloid and Surface Chemistry, Benzamides, Organic chemistry, Peptides, Brønsted–Lowry acid–base theory, Racemization
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المؤلفون: Daniel Lim, Scott J. Miller, Jeffrey L. Gustafson, Kimberly T. Barrett
المصدر: Angewandte Chemie International Edition. 50:5125-5129
مصطلحات موضوعية: Atropisomer, Halogenation, Chemistry, Ligand, Stereochemistry, Enantioselective synthesis, Stereoisomerism, General Medicine, General Chemistry, Inherent chirality, Small molecule, Article, Catalysis, Kinetic resolution, chemistry.chemical_compound, Terphenyl Compounds, Tetrazole, Peptides, Palladium
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المؤلفون: Scott J. Miller, Kimberly T. Barrett
مصطلحات موضوعية: Alkylation, Molecular Structure, Chemistry, Stereochemistry, Organic Chemistry, Enantioselective synthesis, Regioselectivity, Stereoisomerism, Biochemistry, Article, Catalysis, Hydrocarbons, Brominated, chemistry.chemical_compound, Tsuji–Trost reaction, Functional group, Benzamides, Combinatorial Chemistry Techniques, Physical and Theoretical Chemistry, Benzamide, Derivative (chemistry), Palladium
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b0fd9dbecf6ce8c0df8a16ae01a908e4
https://europepmc.org/articles/PMC4364386/ -
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المؤلفون: Scott J. Miller, Kimberly T. Barrett
المصدر: ChemInform. 44
مصطلحات موضوعية: chemistry.chemical_classification, Chemistry, Enantioselective synthesis, Halogenation, Peptide, General Medicine, Combinatorial chemistry, Catalysis