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1دورية أكاديمية
المؤلفون: Leslie W Tari, Xiaoming Li, Michael Trzoss, Daniel C Bensen, Zhiyong Chen, Thanh Lam, Junhu Zhang, Suk Joong Lee, Grayson Hough, Doug Phillipson, Suzanne Akers-Rodriguez, Mark L Cunningham, Bryan P Kwan, Kirk J Nelson, Amanda Castellano, Jeff B Locke, Vickie Brown-Driver, Timothy M Murphy, Voon S Ong, Chris M Pillar, Dean L Shinabarger, Jay Nix, Felice C Lightstone, Sergio E Wong, Toan B Nguyen, Karen J Shaw, John Finn
المصدر: PLoS ONE, Vol 8, Iss 12, p e84409 (2013)
وصف الملف: electronic resource
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2
المؤلفون: Bryan P. Kwan, Kirk J. Nelson, Grayson Hough, John T. Finn, Karen Joy Shaw, Mark Hilgers, Mark L. Cunningham, Thanh Lam, Michael Trzoss, Vickie Brown-Driver, Voon Ong
المصدر: Journal of Medicinal Chemistry. 57:651-668
مصطلحات موضوعية: Models, Molecular, Staphylococcus aureus, Benzimidazole, Stereochemistry, Microbial Sensitivity Tests, Cofactor, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Sepsis, Drug Resistance, Bacterial, Drug Discovery, Dihydrofolate reductase, Animals, Humans, Potency, Structure–activity relationship, chemistry.chemical_classification, biology, Wild type, Staphylococcal Infections, Anti-Bacterial Agents, Tetrahydrofolate Dehydrogenase, Streptococcus pneumoniae, Enzyme, chemistry, Quinazolines, biology.protein, Folic Acid Antagonists, Molecular Medicine, Benzimidazoles
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3
المصدر: SLAS Discovery. 18:1018-1026
مصطلحات موضوعية: DNA, Bacterial, Staphylococcus aureus, Topoisomerase IV, Cefepime, Microbial Sensitivity Tests, Biochemistry, DNA gyrase, Analytical Chemistry, Minimum inhibitory concentration, chemistry.chemical_compound, Bacterial Proteins, Cell Wall, Drug Discovery, Escherichia coli, medicine, biology, Chloramphenicol, Kanamycin, Anti-Bacterial Agents, RNA, Bacterial, chemistry, DNA Gyrase, biology.protein, Molecular Medicine, Vancomycin, Biological Assay, Tedizolid, Biotechnology, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a345debe45ef8d15b8d1dc6858616212
https://doi.org/10.1177/1087057113487208 -
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المؤلفون: Mark L. Cunningham, Doug Phillipson, Bryan P. Kwan, John T. Finn, Kirk J. Nelson, Sergio E. Wong, Michael Trzoss, Jeff B. Locke, Jay C. Nix, Vickie Brown-Driver, Felice C. Lightstone, Zhiyong Chen, Toan B. Nguyen, Karen J. Shaw, Suzanne Akers-Rodriguez, Xiaoming Li, Suk Joong Lee, Amanda Castellano, Dean L. Shinabarger, Timothy M. Murphy, Junhu Zhang, Leslie W. Tari, Chris M. Pillar, Voon Ong, Grayson Hough, Thanh Lam, Daniel C. Bensen
المصدر: PLoS ONE, Vol 8, Iss 12, p e84409 (2013)
PLoS ONEمصطلحات موضوعية: DNA Topoisomerase IV, Models, Molecular, Indoles, Protein Conformation, Topoisomerase IV, medicine.drug_class, Antibiotics, lcsh:Medicine, Microbial Sensitivity Tests, DNA gyrase, Microbiology, Mice, chemistry.chemical_compound, Drug Resistance, Bacterial, medicine, Animals, Topoisomerase II Inhibitors, lcsh:Science, Multidisciplinary, Natural product, Bacteria, biology, Topoisomerase, lcsh:R, Anti-Bacterial Agents, Multiple drug resistance, chemistry, DNA Gyrase, Drug Design, biology.protein, Female, lcsh:Q, Topoisomerase-II Inhibitor, Antibacterial activity, Research Article
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5
المؤلفون: Vickie Brown-Driver, Christopher J. Creighton, John T. Finn, Toan B. Nguyen, Mark L. Cunningham, Zhiyong Chen, Amanda Castellano, Mark Stidham, Sergio E. Wong, Xiaoming Li, Karen J. Shaw, Thanh Lam, Junhu Zhang, Bryan P. Kwan, Kirk J. Nelson, Felice C. Lightstone, Leslie W. Tari, Daniel C. Bensen, Micheal Trzoss
المصدر: Bioorganicmedicinal chemistry letters. 23(5)
مصطلحات موضوعية: DNA Topoisomerase IV, Topoisomerase IV, Clinical Biochemistry, Pharmaceutical Science, medicine.disease_cause, Biochemistry, DNA gyrase, Microbiology, Structure-Activity Relationship, Drug Discovery, medicine, Structure–activity relationship, Humans, Topoisomerase II Inhibitors, Pyrroles, Molecular Biology, Escherichia coli, biology, Pseudomonas aeruginosa, Chemistry, Topoisomerase, Organic Chemistry, biochemical phenomena, metabolism, and nutrition, biology.organism_classification, Acinetobacter baumannii, Anti-Bacterial Agents, Pyrimidines, DNA Gyrase, Drug Design, biology.protein, bacteria, Molecular Medicine, Antibacterial activity
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المؤلفون: Michael J. Hunter, Kirk J. Nelson, Ronald V. Swanson, Duncan E. McRee, Jay C. Nix, Daniel C. Bensen, Leslie W. Tari, Isaac Hoffman
المصدر: Bioorganicmedicinal chemistry letters. 17(3)
مصطلحات موضوعية: Models, Molecular, Pyrimidine, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Aurora A kinase, Molecular Conformation, Pharmaceutical Science, Context (language use), Carboxamide, Protein Serine-Threonine Kinases, Crystallography, X-Ray, Biochemistry, Cell Line, chemistry.chemical_compound, Structure-Activity Relationship, Aurora Kinases, Drug Discovery, medicine, Structure–activity relationship, Moiety, Animals, Binding site, Enzyme Inhibitors, Molecular Biology, biology, Organic Chemistry, Active site, ErbB Receptors, Pyrimidines, chemistry, biology.protein, Molecular Medicine