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1
المؤلفون: Koichiro Mukoyoshi, Kaoru Yamagami, Kousei Yoshihara, Koji Yokoo, Susumu Yamaki, Fumie Takahashi, Toshihiro Hamajima, Yukihito Sugano, Koji Kato, Hidehiko Fukahori, Ayako Moritomo
المصدر: Bioorganic & Medicinal Chemistry. 26:2410-2419
مصطلحات موضوعية: 0301 basic medicine, Class I Phosphatidylinositol 3-Kinases, Pyridines, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Amide, Drug Discovery, Pyrazolopyridine, Animals, Humans, Protein Kinase Inhibitors, Molecular Biology, Phosphoinositide-3 Kinase Inhibitors, Biological evaluation, Mice, Inbred BALB C, Molecular Structure, Chemistry, Organic Chemistry, Nuclear Proteins, Stereoisomerism, Molecular Docking Simulation, 030104 developmental biology, Pyrazoles, Molecular Medicine, Female, Selectivity, Transcription Factors
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2
المؤلفون: Kazuo Nakai, Hiroyuki Usuda, Keiko Hatanaka, Hiroshi Sasaki, Ayako Moritomo, Shohei Shirakami, Yutaka Nakajima, Takayuki Inoue, Koichiro Mukoyoshi, Hisao Hamaguchi, Yasuyuki Higashi, Akira Tanaka, Masamichi Inami, Shigeki Kunikawa, Fumie Takahashi
المصدر: Bioorganic & Medicinal Chemistry. 23:4871-4883
مصطلحات موضوعية: Graft Rejection, Male, Transplantation, Heterotopic, Pyridines, medicine.drug_class, T-Lymphocytes, T cell, Clinical Biochemistry, hERG, Administration, Oral, Pharmaceutical Science, Carboxamide, Pharmacology, Biochemistry, chemistry.chemical_compound, Dogs, Immune system, In vivo, Drug Discovery, medicine, Animals, Humans, Immunologic Factors, Protein Kinase Inhibitors, Molecular Biology, Cell Proliferation, Binding Sites, biology, Chemistry, Organic Chemistry, Janus Kinase 3, Haplorhini, Janus Kinase 1, Janus Kinase 2, Amides, Protein Structure, Tertiary, Rats, Molecular Docking Simulation, medicine.anatomical_structure, Rats, Inbred Lew, Lipophilicity, Microsomes, Liver, biology.protein, Interleukin-2, Molecular Medicine, Janus kinase, Lead compound, Half-Life
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3
المؤلفون: Shigeki Kunikawa, Akira Tanaka, Fumiyuki Shirai, Koichiro Mukoyoshi, Hiroaki Tominaga, Mamoru Tasaki, Shinya Nagashima, Noboru Chida
المصدر: Bioorganic & Medicinal Chemistry. 23:3269-3277
مصطلحات موضوعية: Drug, Halogenation, T-Lymphocytes, T cell, media_common.quotation_subject, Clinical Biochemistry, Protein Kinase C-theta, Gene Expression, Pharmaceutical Science, Pharmacology, Inhibitory postsynaptic potential, Biochemistry, Dependent drug, Structure-Activity Relationship, Drug Discovery, medicine, Cytochrome P-450 CYP3A, Humans, Drug Interactions, ATP Binding Cassette Transporter, Subfamily B, Member 1, Protein Kinase Inhibitors, Molecular Biology, Protein Kinase C, media_common, CYP3A4, Chemistry, Organic Chemistry, medicine.disease, Transplant rejection, Isoenzymes, Pyrimidines, medicine.anatomical_structure, Drug Resistance, Neoplasm, Rheumatoid arthritis, Microsomes, Liver, Molecular Medicine, Signal Transduction
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4
المؤلفون: Hisao Hamaguchi, Yasuyuki Higashi, Akira Tanaka, Ayako Moritomo, Yutaka Nakajima, Masataka Morita, Takashi Tojo, Shohei Shirakami, Hiroshi Sasaki, Kazuo Nakai, Keiko Hatanaka, Fumie Takahashi, Koichiro Mukoyoshi, Takayuki Inoue
المصدر: CHEMICAL & PHARMACEUTICAL BULLETIN. 63:341-353
مصطلحات موضوعية: Stereochemistry, Chemistry, T cell, Janus kinase 3, Substituent, Chemical modification, General Chemistry, General Medicine, chemistry.chemical_compound, medicine.anatomical_structure, Docking (molecular), Drug Discovery, Pyridine, medicine, Immune Mediators, Janus kinase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::46a152d038420cc6b471f5ce5284ea06
https://doi.org/10.1248/cpb.c15-00036 -
5
المؤلفون: Yutaka, Nakajima, Takashi, Tojo, Masataka, Morita, Keiko, Hatanaka, Shohei, Shirakami, Akira, Tanaka, Hiroshi, Sasaki, Kazuo, Nakai, Koichiro, Mukoyoshi, Hisao, Hamaguchi, Fumie, Takahashi, Ayako, Moritomo, Yasuyuki, Higashi, Takayuki, Inoue
المصدر: Chemicalpharmaceutical bulletin. 63(5)
مصطلحات موضوعية: Male, Models, Molecular, Molecular Structure, Pyridines, Janus Kinase 3, Rats, Immunomodulation, Rats, Sprague-Dawley, Microsomes, Liver, Animals, Lymphocytes, Medical Informatics, Spleen, Cell Proliferation, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::06929a07b6bd29059c79e7eec1721dfe
https://pubmed.ncbi.nlm.nih.gov/25786493 -
6
المؤلفون: Akira Tanaka, Masamichi Inami, Hisao Hamaguchi, Yasuyuki Higashi, Yutaka Nakajima, Ayako Moritomo, Hiroyuki Usuda, Shohei Shirakami, Koichiro Mukoyoshi, Kazuo Nakai, Hiroshi Sasaki, Shigeki Kunikawa, Fumie Takahashi, Keiko Hatanaka, Takayuki Inoue
المصدر: Bioorganic & Medicinal Chemistry. 25:2813
مصطلحات موضوعية: Chemistry, Stereochemistry, medicine.drug_class, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, 030226 pharmacology & pharmacy, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, 030220 oncology & carcinogenesis, Drug Discovery, Pyridine, medicine, Molecular Medicine, Molecular Biology
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7
المصدر: Chirality. 14:713-715
مصطلحات موضوعية: Pharmacology, Spiropyran, chemistry.chemical_classification, Stereochemistry, fungi, Organic Chemistry, Optically active, Catalysis, Analytical Chemistry, Amino acid, chemistry.chemical_compound, chemistry, Drug Discovery, Moiety, Merocyanine, Enantiomer, Chirality (chemistry), Spectroscopy, Derivative (chemistry)
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8
المؤلفون: Kazunori Tsubaki, Koichiro Mukoyoshi, Tadamune Otsubo, Kaoru Fuji
المصدر: ChemInform. 31
مصطلحات موضوعية: chemistry.chemical_compound, Monomer, chemistry, Dimer, Polymer chemistry, Phenol, General Medicine, Condensation reaction
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9
المؤلفون: Koichiro Mukoyoshi, Tadamune Otsubo, Kazunori Tsubaki, Kaoru Fuji
المصدر: Chemicalpharmaceutical bulletin. 48(6)
مصطلحات موضوعية: Molecular Structure, Macromolecular Substances, Dimer, Spectrum Analysis, General Chemistry, General Medicine, Condensation reaction, Chemical synthesis, Inclusion compound, chemistry.chemical_compound, Monomer, chemistry, Drug Discovery, Polymer chemistry, Calixarene, Phenol, Organic chemistry, Calixarenes, Cyclophane
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e3a8bed20c56ec091f3e56600eb7e4ae
https://pubmed.ncbi.nlm.nih.gov/10866155