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1
المؤلفون: Tomoyuki Tsunemi, Tomohiro Makino, Kazuo Miyazaki, Hideki Terashima, Kyoko Yamashiro, Katsushi Katayama, Maki Terakawa, Hiroaki Maeda, Kouichi Uoto, Munetada Haruyama, Ryosuke Yoshioka
المصدر: Bioorganicmedicinal chemistry letters. 30(19)
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, Phenotypic screening, Clinical Biochemistry, Cell, Pharmaceutical Science, Pharmacology, 01 natural sciences, Biochemistry, Structure-Activity Relationship, Drug Stability, In vivo, hemic and lymphatic diseases, Drug Discovery, Fetal hemoglobin, medicine, Animals, Humans, Inducer, Spiro Compounds, Globin, Molecular Biology, Fetal Hemoglobin, ADME, Erythroid Precursor Cells, Molecular Structure, 010405 organic chemistry, Chemistry, Organic Chemistry, Isoxazoles, 0104 chemical sciences, Bioavailability, 010404 medicinal & biomolecular chemistry, Macaca fascicularis, medicine.anatomical_structure, Gene Expression Regulation, Drug Design, Microsomes, Liver, Molecular Medicine, Azetidines
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2
المؤلفون: Kenji Yoshikawa, Toshiharu Yoshino, Makoto Takemura, Akiyoshi Mochizuki, Toshiharu Ohta, Tsutomu Nagata, Kouichi Uoto, Yoshihiro Yokomizo, Hiroyuki Naito, Katsuhiro Kawakami, Hideyuki Kanno, Makoto Suzuki
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2133-2140
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, Molecular model, medicine.drug_mechanism_of_action, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Factor Xa Inhibitor, Substituent, Pharmaceutical Science, Ethylenediamine, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Structure–activity relationship, Moiety, Molecular Biology, chemistry.chemical_classification, Organic Chemistry, chemistry, Drug Design, Molecular Medicine, Factor Xa Inhibitors
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3
المؤلفون: Eri Watanabe, Shozo Kobayashi, Ken-Ichi Yoshida, Tsuyoshi Otani, Yoshikazu Ishii, Kouichi Uoto, Masato Hata, Akikazu Ando
المصدر: Medical Mycology. 48:613-621
مصطلحات موضوعية: Antifungal Agents, Mutant, Saccharomyces cerevisiae, Microbial Sensitivity Tests, Biology, Reductase, Gas Chromatography-Mass Spectrometry, Microbiology, chemistry.chemical_compound, Phenols, Drug Resistance, Fungal, Oxidoreductase, Ergosterol, Candida albicans, chemistry.chemical_classification, Cell Membrane, General Medicine, Blotting, Northern, biology.organism_classification, Corpus albicans, Drug Combinations, Microscopy, Electron, Infectious Diseases, Enzyme, chemistry, Biochemistry, Chromatography, Thin Layer, Oxidoreductases, Oils
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4
المؤلفون: Kouichi Akahane, Motoko Nagata, Mayumi Kitagawa, Takao Horiuchi, Kouichi Uoto
المصدر: Bioorganic & Medicinal Chemistry. 17:7850-7860
مصطلحات موضوعية: Models, Molecular, Spectrometry, Mass, Electrospray Ionization, Magnetic Resonance Spectroscopy, Molecular model, Cell Survival, Stereochemistry, Clinical Biochemistry, Mice, Nude, Pharmaceutical Science, Hydrazone, Antineoplastic Agents, Thiophenes, Biochemistry, Chemical synthesis, Benzaldehyde, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Cell Line, Tumor, Spectroscopy, Fourier Transform Infrared, Drug Discovery, Animals, Humans, Structure–activity relationship, Moiety, Protein Kinase Inhibitors, Molecular Biology, chemistry.chemical_classification, Bicyclic molecule, Chemistry, Organic Chemistry, Hydrazones, Neoplasms, Experimental, Cyclin-Dependent Kinases, Pyrimidines, Molecular Medicine, Selectivity
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5
المؤلفون: Hiroyuki Naito, Yoshida Keisuke, Yuuichi Sugimoto, Tsunehiko Soga, Haruko Kawato, Masaki Miyazaki, Takahiko Seki, Setsuko Fukutake, Tooru Okayama, Kouichi Uoto, Masaya Miyazaki, Masashi Aonuma, Mayumi Kitagawa
المصدر: Bioorganicmedicinal chemistry. 23(10)
مصطلحات موضوعية: Male, Pyrrolidines, Stereochemistry, Clinical Biochemistry, Substituent, Pharmaceutical Science, Administration, Oral, Gene Expression, Mice, Nude, Antineoplastic Agents, Bone Neoplasms, Biochemistry, Pyrrolidine, chemistry.chemical_compound, Mice, Oral administration, Cell Line, Tumor, Drug Discovery, Potency, Animals, Humans, Cytotoxicity, Molecular Biology, Octane, Cell Proliferation, Mice, Inbred BALB C, Organic Chemistry, Imidazoles, Proto-Oncogene Proteins c-mdm2, Sarcoma, Fluorine, Xenograft Model Antitumor Assays, Piperazine, Thiazoles, chemistry, Molecular Medicine, Tumor Suppressor Protein p53, Lead compound, Protein Binding
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6
المؤلفون: Takeshi Jimbo, Tsunehiko Soga, Motoko Nagata, Yasuyuki Takeda, Chiho Ono, Michio Iwahana, Hirofumi Terasawa, Kouichi Uoto, Noriko Tanaka, Ryo Atsumi
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:3209-3215
مصطلحات موضوعية: Chemistry, Organic Chemistry, Clinical Biochemistry, Melanoma, Experimental, Pharmaceutical Science, Antineoplastic Agents, General Medicine, Biochemistry, Terpene, Mice, Drug Discovery, Microsomes, Liver, Organic chemistry, Animals, Humans, Molecular Medicine, Taxoids, Molecular Biology
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7
المؤلفون: Yasuyuki, Takeda, Toshiharu, Yoshino, Kouichi, Uoto, Jun, Chiba, Takashi, Ishiyama, Michio, Iwahana, Takeshi, Jimbo, Noriko, Tanaka, Hirofumi, Terasawa, Tsunehiko, Soga
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:185-190
مصطلحات موضوعية: Paclitaxel, Cell Survival, Organic Chemistry, Clinical Biochemistry, Melanoma, Experimental, Molecular Conformation, Pharmaceutical Science, Crystallography, X-Ray, Antineoplastic Agents, Phytogenic, Biochemistry, Mice, Solubility, Drug Discovery, Tumor Cells, Cultured, Animals, Humans, Molecular Medicine, Indicators and Reagents, Drug Screening Assays, Antitumor, Molecular Biology, Neoplasm Transplantation
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8
المؤلفون: Toshiharu Yoshino, Kouichi Uoto, Takeshi Jimbo, Shin Iimura, Satoru Ohsuki, Tsunehiko Soga, Jun Chiba, Michio Iwahana, Hirofumi Terasawa
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:407-410
مصطلحات موضوعية: Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Analogue synthesis, Orally active, Docetaxel, Oral administration, In vivo, Drug Discovery, medicine, Molecular Medicine, Cytotoxicity, Molecular Biology, B16 melanoma, 10-deoxy-10-C-morpholinoethyl docetaxel, medicine.drug
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9
المؤلفون: Keiki Sato, Yasuyoshi Kawato, Hirofumi Terasawa, Y. Hirota, Kouichi Uoto, Satoru Ohsuki, Masamichi Sugimori, Ikuo Mitsui, Akio Ejima
المصدر: Journal of Medicinal Chemistry. 41:2308-2318
مصطلحات موضوعية: Ketone, Stereochemistry, Antineoplastic Agents, Irinotecan, Chemical synthesis, Mice, Structure-Activity Relationship, Drug Discovery, Tumor Cells, Cultured, medicine, Animals, Humans, Structure–activity relationship, Enzyme Inhibitors, Cytotoxicity, chemistry.chemical_classification, biology, Bicyclic molecule, Leukemia P388, Topoisomerase, chemistry, biology.protein, Molecular Medicine, Camptothecin, Drug Screening Assays, Antitumor, Topoisomerase I Inhibitors, Cell Division, Lactone, medicine.drug
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10
المؤلفون: Shuichi Ando, Tsunehiko Soga, Ikuo Mitsui, Hirofumi Terasawa, Kouichi Uoto, Haruhiro Takenoshita, Yasuhide Hirota, Toshiharu Yoshino
المصدر: Chemical and Pharmaceutical Bulletin. 46:770-776
مصطلحات موضوعية: Chemical Phenomena, Paclitaxel, Tertiary amine, Swine, Stereochemistry, Docetaxel, Microtubules, Chemical synthesis, Methanesulfonic acid, chemistry.chemical_compound, Tubulin, In vivo, Drug Discovery, medicine, Animals, Humans, Cytotoxicity, Chemistry, Physical, General Chemistry, General Medicine, Prodrug, Antineoplastic Agents, Phytogenic, Solubility, chemistry, Taxoids, Drug Screening Assays, Antitumor, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8b57cf8754b51c033a35a13f828c8b66
https://doi.org/10.1248/cpb.46.770