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1
المؤلفون: Peter T. Buckley, James J. Foley, Edward F. Webb, Roderick S. Davis, Dulcie B. Schmidt, Jakob Busch-Petersen, Michael Salmon, Jian Jin, Widdowson Katherine L, Kristen E. Belmonte, Henry M. Sarau, Yonghui Wang, Qi Jin, Palovich Michael R, Ann M. Bullion
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:7087-7091
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Bronchi, Muscarinic Antagonists, Biochemistry, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Solid-phase synthesis, In vivo, Drug Discovery, Muscarinic acetylcholine receptor, Animals, Urea, Structure–activity relationship, Moiety, Ammonium, Tyrosine, Molecular Biology, Chemistry, Organic Chemistry, Receptors, Muscarinic, Quaternary Ammonium Compounds, Molecular Medicine
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2
المؤلفون: Yonghui Wang, Henry M. Sarau, Dongchuan Shi, Dwight M. Morrow, Miriam Burman, Michael L. Moore, Palovich Michael R, Ralph A. Rivero, Edward F. Webb, Dramane I. Laine, Jian Jin, Brian Budzik, Kristen E. Belmonte, Feng Wang, James J. Foley, Haibo Xie, Michael Salmon, Chongye Zhu, Manuela Berlanga, Zehong Wan
المصدر: Journal of Medicinal Chemistry. 51:5915-5918
مصطلحات موضوعية: medicine.medical_specialty, Bronchoconstriction, Drug Evaluation, Preclinical, Pharmacology, Bronchial Provocation Tests, Piperazines, Bronchoconstrictor Agents, Mice, Structure-Activity Relationship, In vivo, Internal medicine, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Administration, Intranasal, Methacholine Chloride, Acetylcholine receptor, Molecular Structure, Chemistry, Antagonist, Muscarinic acetylcholine receptor M3, Stereoisomerism, Biological activity, Receptors, Muscarinic, Bronchodilator Agents, Disease Models, Animal, Endocrinology, Molecular Medicine, Nasal administration, medicine.symptom
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3
المؤلفون: Palovich Michael R, Miriam Burman, Edward F. Webb, Roderick S. Davis, Henry M. Sarau, Yonghui Wang, Wei Fu, Dwight M. Morrow, Jian Jin, Feng Wang, Qi Jin, Kristen E. Belmonte, Parvathi Rao, Michael L. Moore, Manuela Berlanga, James J. Foley, Chris J. Dehaas, Michael Salmon, Ralph A. Rivero, Lorena A. Kallal, Jakob Busch-Petersen, Dongchuan Shi
المصدر: Journal of Medicinal Chemistry. 51:4866-4869
مصطلحات موضوعية: medicine.drug_class, Bronchoconstriction, Guinea Pigs, Drug Evaluation, Preclinical, Muscarinic Antagonists, Pharmacology, Inhibitory postsynaptic potential, Mice, In vivo, Bronchodilator, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Acetylcholine receptor, Chemistry, Phenylurea Compounds, Antagonist, Bridged Bicyclo Compounds, Heterocyclic, Rats, Quaternary Ammonium Compounds, Biochemistry, Tyrosine, Molecular Medicine, Nasal administration, medicine.symptom
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4
المؤلفون: Widdowson Katherine L, Edward F. Webb, Palovich Michael R, James J. Foley, Kristen E. Belmonte, Haibo Xie, Peter T. Buckley, Noémie Buffet, Dramane I. Laine
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:6066-6069
مصطلحات موضوعية: Carbamate, medicine.medical_treatment, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Muscarinic Antagonists, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Mice, Pulmonary Disease, Chronic Obstructive, chemistry.chemical_compound, In vivo, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Receptor, Molecular Biology, Acetylcholine receptor, Molecular Structure, Chemistry, Organic Chemistry, Antagonist, Tropane, Bridged Bicyclo Compounds, Heterocyclic, Receptors, Muscarinic, Bronchodilator Agents, Molecular Medicine, Carbamates, Tropanes
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5
المؤلفون: Victoria J. Barrett, Feng Wang, Christopher Browning, Matthew J Lindon, Henry M. Sarau, James A. Fornwald, Andy J. Harker, Guido Hartmann, Jeffery K. Kerns, David P. Andrew, Graeme Irvine Stevenson, Ashley Paul Hancock, Victoria Vinader, Michael L. Moore, James J. Foley, Jian Jin, Parvathi Rao, Anthony J. Jurewicz, Helen E. Connor, Dwight M. Morrow, Kristen E. Belmonte, Yonghui Wang, Ralph A. Rivero, Cuc Nguyen
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:1722-1725
مصطلحات موضوعية: ERG1 Potassium Channel, Stereochemistry, High-throughput screening, Clinical Biochemistry, Drug Evaluation, Preclinical, Human immunodeficiency virus (HIV), Pharmaceutical Science, CHO Cells, Computational biology, Protein Serine-Threonine Kinases, medicine.disease_cause, Biochemistry, Chemical synthesis, Myotonin-Protein Kinase, Receptors, CCR8, Structure-Activity Relationship, Cricetulus, Th2 Cells, Cricetinae, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Computer Simulation, Molecular Biology, Oxazolidinones, Chemistry, Organic Chemistry, Ether-A-Go-Go Potassium Channels, Chemotaxis, Leukocyte, Lung disease, Molecular Medicine, Indicators and Reagents, Receptors, Chemokine
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6
المصدر: American Journal of Respiratory Cell and Molecular Biology. 34:233-241
مصطلحات موضوعية: Adult, Male, Pulmonary and Respiratory Medicine, Neutrophils, Receptor expression, Clinical Biochemistry, Gene Expression, Biology, Receptors, Interleukin-8A, chemistry.chemical_compound, Reference Values, Sphingosine, Cell surface receptor, Lysophosphatidic acid, Humans, Protein Isoforms, Sphingosine-1-phosphate, Receptors, Lysophosphatidic Acid, Receptor, Molecular Biology, Aged, Aged, 80 and over, Chemotaxis, organic chemicals, Pneumonia, Cell Biology, Middle Aged, Molecular biology, Blot, Receptors, Lysophospholipid, chemistry, Case-Control Studies, Female, lipids (amino acids, peptides, and proteins), Lysophospholipids, biological phenomena, cell phenomena, and immunity, Dimerization
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7
المؤلفون: Kristen E. Belmonte
المصدر: Proceedings of the American Thoracic Society. 2:297-304
مصطلحات موضوعية: Pulmonary and Respiratory Medicine, medicine.medical_specialty, medicine.drug_class, Cholinergic Antagonists, Pulmonary Disease, Chronic Obstructive, Aclidinium bromide, Parasympathetic Nervous System, Internal medicine, Administration, Inhalation, Muscarinic acetylcholine receptor, Anticholinergic, Humans, Medicine, Receptor, Lung, Asthma, business.industry, medicine.disease, Receptors, Muscarinic, Bronchodilator Agents, Endocrinology, Immunology, Cholinergic, Drug Therapy, Combination, Bronchoconstriction, Bronchial Hyperreactivity, medicine.symptom, business, Acetylcholine, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::38af4224038cd050443285a2472a56fd
https://doi.org/10.1513/pats.200504-043sr -
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المؤلفون: Richard W. Costello, Gerald J. Gleich, Kristen E. Belmonte, David B. Jacoby, Allison D. Fryer, Christopher M. Evans
المصدر: Europe PubMed Central
مصطلحات موضوعية: Pulmonary and Respiratory Medicine, Quinuclidines, medicine.medical_specialty, Physiology, Guinea Pigs, Substance P, Biology, Antibodies, chemistry.chemical_compound, Ribonucleases, Neurokinin-1 Receptor Antagonists, Piperidines, Physiology (medical), Internal medicine, Muscarinic acetylcholine receptor, medicine, Animals, Receptor, Cyclophosphamide, Acetylcholine receptor, Neurons, Receptor, Muscarinic M2, Heparin, Vagus Nerve, Muscarinic acetylcholine receptor M2, Blood Proteins, Cell Biology, Eosinophil Granule Proteins, Receptors, Muscarinic, Electric Stimulation, Endocrinology, medicine.anatomical_structure, chemistry, Autoreceptor, Female, Neuron, Bronchial Hyperreactivity, Acetylcholine, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0ac8d56001d917e1d002cb3130a5d8a4
https://doi.org/10.1152/ajplung.2000.279.3.l477 -
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المصدر: British Journal of Pharmacology. 124:267-276
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, Chemistry, Muscarinic acetylcholine receptor M2, Muscarinic agonist, chemistry.chemical_compound, Endocrinology, Pilocarpine, Internal medicine, Muscarinic acetylcholine receptor, medicine, NK1 receptor antagonist, Bronchoconstriction, medicine.symptom, Receptor, Histamine, medicine.drug
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10
المؤلفون: Allison D. Fryer, Kristen E. Belmonte, David B. Jacoby
المصدر: British Journal of Pharmacology. 121:1287-1294
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, business.industry, Muscarinic acetylcholine receptor M3, Muscarinic acetylcholine receptor M2, Muscarinic acetylcholine receptor M1, Muscarinic agonist, Endocrinology, Pilocarpine, Internal medicine, Muscarinic acetylcholine receptor, Muscarinic acetylcholine receptor M4, Medicine, business, Acetylcholine, medicine.drug