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1دورية أكاديمية
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 597-605 (2022)
مصطلحات موضوعية: colchiceine tautomers, click, heck reaction, tubulin inhibitors, anticancer, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Natalia Skrzypczak, Krystian Pyta, Piotr Ruszkowski, Przemysław Mikołajczak, Małgorzata Kucińska, Marek Murias, Maria Gdaniec, Franz Bartl, Piotr Przybylski
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 36, Iss 1, Pp 1898-1904 (2021)
مصطلحات موضوعية: ansamycins, benzoquinones, chaperone hsp90, anticancer, sar, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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3
المؤلفون: Anna Janas, Krystian Pyta, Maria Gdaniec, Piotr Przybylski
المصدر: The Journal of organic chemistry. 87(5)
مصطلحات موضوعية: Lactones, Acetals, Organic Chemistry, Molecular Conformation, Macrolides, Anti-Bacterial Agents
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4
المؤلفون: Marzena Gajecka, Monika Szukowska, Marcelina M. Jaworska, Anna Janas, Krystian Pyta, Piotr Przybylski, Paulina Pecyna, Franz Bartl
المصدر: European Journal of Medicinal Chemistry. 167:96-104
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, Tertiary amine, Stereochemistry, Hydrazone, 01 natural sciences, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, polycyclic compounds, Potency, Amines, Guanidine, 030304 developmental biology, Pharmacology, chemistry.chemical_classification, 0303 health sciences, Binding Sites, 010405 organic chemistry, Chemistry, Organic Chemistry, Hydrazones, Rifamycin, General Medicine, Rifamycins, Anti-Bacterial Agents, 0104 chemical sciences, Molecular Docking Simulation, Solubility, Docking (molecular), Lipophilicity, Amine gas treating, Rifampin, Hydrophobic and Hydrophilic Interactions
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5
المؤلفون: Anna Janas, Katarzyna Pyta-Klich, Piotr Przybylski, Krystian Pyta
المصدر: Tetrahedron. 74:6335-6365
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Organic Chemistry, chemistry.chemical_element, 010402 general chemistry, 01 natural sciences, Biochemistry, Sulfur, Combinatorial chemistry, 0104 chemical sciences, Cascade reaction, Drug Discovery, Relevance (information retrieval), Pharmacophore
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6
المؤلفون: Przemysław Mikołajczak, Malgorzata Kucinska, Piotr Ruszkowski, Piotr Przybylski, Marek Murias, Franz Bartl, Natalia Skrzypczak, Maria Gdaniec, Krystian Pyta
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 36, Iss 1, Pp 1898-1904 (2021)
Journal of Enzyme Inhibition and Medicinal Chemistry
article-version (VoR) Version of Recordمصطلحات موضوعية: Lactams, Macrocyclic, Antineoplastic Agents, RM1-950, anticancer, Cell Line, HeLa, Hydrophobic effect, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, benzoquinones, Humans, Ammonium, sar, Pharmacology, Molecular Structure, biology, Spectrum Analysis, chaperone hsp90, Drug Synergism, ansamycins, General Medicine, Potentiator, Geldanamycin, biology.organism_classification, Combinatorial chemistry, Quaternary Ammonium Compounds, chemistry, Docking (molecular), Salts, Therapeutics. Pharmacology, Drug Screening Assays, Antitumor, Derivative (chemistry), Research Article, Research Paper, Quinuclidine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1d3f414f9eba80d4452f914ca6f158fc
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7
المؤلفون: Maria Gdaniec, Krystian Pyta, Piotr Przybylski, Barbara Wicher
المصدر: Crystal Growth & Design. 18:742-754
مصطلحات موضوعية: Hydrogen bond, Chemistry, Intermolecular force, Ionic bonding, Rifamycins, 02 engineering and technology, General Chemistry, 010402 general chemistry, 021001 nanoscience & nanotechnology, Condensed Matter Physics, 01 natural sciences, 0104 chemical sciences, Solvent, Crystallography, polycyclic compounds, medicine, Molecule, General Materials Science, 0210 nano-technology, Structural motif, Rifampicin, medicine.drug
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8
المؤلفون: Krystian Pyta, Piotr Przybylski, Anna Janas, Maria Gdaniec, Wojciech Schilf, Franz Bartl, Natalia Skrzypczak, Barbara Wicher
المصدر: ACS infectious diseases. 5(10)
مصطلحات موضوعية: 0301 basic medicine, Tuberculosis, Membrane permeability, medicine.drug_class, 030106 microbiology, Cell, Antibiotics, Molecular Conformation, Rifamycins, Permeability, Microbiology, 03 medical and health sciences, Structure-Activity Relationship, Gram-Negative Bacteria, polycyclic compounds, medicine, Potency, Chemistry, Cell Membrane, Rifamycin, Water, Biological Transport, DNA-Directed RNA Polymerases, medicine.disease, Anti-Bacterial Agents, 030104 developmental biology, Infectious Diseases, medicine.anatomical_structure, Models, Chemical, Rifampin, Hydrophobic and Hydrophilic Interactions
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9
المؤلفون: Paulina Pecyna, Marzena Gajecka, Marietta Blecha, Piotr Przybylski, Anna Janas, Krystian Pyta, Katarzyna Klich
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:4322-4326
مصطلحات موضوعية: Clinical Biochemistry, Triazole, Pharmaceutical Science, Alkyne, Microbial Sensitivity Tests, Hydroxylamines, 010402 general chemistry, 01 natural sciences, Biochemistry, Catalysis, chemistry.chemical_compound, Anti-Infective Agents, Drug Discovery, Organic chemistry, Molecular Biology, chemistry.chemical_classification, Ergosterol, Molecular Structure, 010405 organic chemistry, Organic Chemistry, Fungi, Gossypol, Triazoles, Tautomer, Cycloaddition, 0104 chemical sciences, chemistry, Alkynes, Intramolecular force, Molecular Medicine, Azide, Copper
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10
المؤلفون: Krystian Pyta, Marzena Gajecka, Piotr Przybylski, Lech Celewicz, Piotr Ruszkowski, Katarzyna Klich, Marcelina M. Kubicka
المصدر: Journal of Medicinal Chemistry. 59:7963-7973
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Triazole, Antineoplastic Agents, Microbial Sensitivity Tests, Gram-Positive Bacteria, 010402 general chemistry, 01 natural sciences, HeLa, Structure-Activity Relationship, chemistry.chemical_compound, Cell Line, Tumor, Spiramycin, Drug Discovery, medicine, Humans, Cycloaddition Reaction, biology, 010405 organic chemistry, Triazoles, biology.organism_classification, Cycloaddition, Anti-Bacterial Agents, 0104 chemical sciences, Aglycone, Solubility, chemistry, Lipophilicity, Thermodynamics, Molecular Medicine, Drug Screening Assays, Antitumor, Selectivity, Conjugate, medicine.drug