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المؤلفون: Laishun Chen, Parviz Ghahramani, Antonia Periclou, Nayra Gad, William M. Greenberg, Julie Wangsa, Ramesh Boinpally
المصدر: Clinical Drug Investigation. 35:601-612
مصطلحات موضوعية: Adult, Cyclopropanes, Male, medicine.medical_specialty, Adolescent, Pharmacology, Young Adult, Pharmacokinetics, Norepinephrine reuptake inhibitor, Milnacipran, Internal medicine, medicine, Humans, Drug Interactions, Pharmacology (medical), Alprazolam, business.industry, Cytochrome P-450 CYP3A Inducers, General Medicine, Carbamazepine, Middle Aged, Healthy Volunteers, Ketoconazole, Endocrinology, Area Under Curve, Delayed-Action Preparations, Cytochrome P-450 CYP3A Inhibitors, Female, business, Reuptake inhibitor, Levomilnacipran, medicine.drug
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المؤلفون: Philippe Hermann, Louise Roques, Laurence Barthe, Laishun Chen, Isabelle Hude, Bernadette Maynadier, Valérie Brunner, Sébastien Séguier
المصدر: Drug Design, Development and Therapy
مصطلحات موضوعية: Adult, Cyclopropanes, Male, medicine.medical_specialty, FETZIMA, Adolescent, tissue distribution, Pharmaceutical Science, Administration, Oral, Urine, Pharmacology, Hydroxylation, Models, Biological, Excretion, Rats, Sprague-Dawley, Young Adult, Glucuronides, Norepinephrine reuptake inhibitor, Species Specificity, Oral administration, Internal medicine, Drug Discovery, medicine, Animals, Humans, Carbon Radioisotopes, Serotonin and Noradrenaline Reuptake Inhibitors, metabolites, Biotransformation, Original Research, Drug Design, Development and Therapy, Chemistry, Milnacipran, Middle Aged, Antidepressive Agents, Macaca fascicularis, Renal Elimination, Endocrinology, Dealkylation, Renal physiology, excretion, Female, Serotonin, Glucuronide, Levomilnacipran, mass balance, Protein Binding
وصف الملف: text/html
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المؤلفون: William J. Pitts, Alaric J. Dyckman, Scott H. Watterson, Robert V. Moquin, Kim W. McIntyre, Zheng Yang, Jagabandhu Das, Katy Van Kirk, James R. Burke, David B. Wang-Iverson, Hollie Booth-Lute, James Kempson, Laishun Chen, Charles M. Langevine, Joel C. Barrish, Guchen Yang, Xiaoxia Yang, John H. Dodd, David S. Nirschl, Murray McKinnon, Steven H. Spergel, Mark A. Pattoli, Michael Galella, Kurt R. Gregor, Junquing Guo
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:7006-7012
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Biochemistry, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Acetamides, Drug Discovery, Animals, Humans, Inhibitory concentration 50, Structure–activity relationship, Potency, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Molecular Structure, Drug discovery, Organic Chemistry, Inflammatory Bowel Diseases, In vitro, I-kappa B Kinase, Rats, Enzyme Activation, chemistry, Molecular Medicine, Heterocyclic Compounds, 3-Ring, Acetamide, Tricyclic
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المؤلفون: James Kempson, Joel C. Barrish, Laishun Chen, Alaric J. Dyckman, Robert V. Moquin, Kim W. McIntyre, Kathleen M. Gillooly, William J. Pitts, James R. Burke, Steven H. Spergel, Jagabandhu Das, Mark A. Pattoli, Scott H. Watterson, John H. Dodd, Murray McKinnon, Xiao Xia Yang, Junqing Guo, Charles M. Langevine
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:2646-2649
مصطلحات موضوعية: Lipopolysaccharides, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, IκB kinase, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Structure–activity relationship, skin and connective tissue diseases, Protein Kinase Inhibitors, Molecular Biology, chemistry.chemical_classification, Tumor Necrosis Factor-alpha, Organic Chemistry, Imidazoles, I-kappa B Kinase, Rats, Pyrimidines, Enzyme, chemistry, Molecular Medicine, Amine gas treating, Lead compound, Tricyclic
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المؤلفون: Charles M. Langevine, Joseph A. Furch, Dominique Belanger, Mark A. Pattoli, Joel C. Barrish, Alaric J. Dyckman, Marco Dodier, James Kempson, Jagabandhu Das, David S. Nirschl, Laishun Chen, Punit Marathe, Kathleen M. Gillooly, Junqing Guo, Robert V. Moquin, John H. Dodd, Murray McKinnon, Anne Marinier, Zheng Yang, Steven H. Spergel, Claude A. Quesnelle, Kim W. McIntyre, Katy Van Kirk, James R. Burke, William J. Pitts, Scott H. Watterson, Alain Martel, Patrice Gill, David B. Wang-Iverson, Tianle Li
المصدر: Journal of Medicinal Chemistry. 52:1994-2005
مصطلحات موضوعية: Lipopolysaccharides, Recombinant Fusion Proteins, IκB kinase, In Vitro Techniques, Crystallography, X-Ray, Chemical synthesis, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Animals, Humans, Thiazole, Oxazoles, Glutathione Transferase, Oxazole, chemistry.chemical_classification, Mice, Inbred BALB C, Tumor Necrosis Factor-alpha, Imidazoles, Biological activity, I-kappa B Kinase, Rats, Thiazoles, Enzyme, chemistry, Biochemistry, Leukocytes, Mononuclear, Microsomes, Liver, Molecular Medicine, Female, Signal transduction, Heterocyclic Compounds, 3-Ring, Tricyclic
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المؤلفون: Parviz Ghahramani, Carl Gommoll, Laishun Chen, S. Zukin, Joann O’Connor, William M. Greenberg, Antonia Periclou
المصدر: Clinical therapeutics. 37(9)
مصطلحات موضوعية: Adult, Cyclopropanes, Male, medicine.medical_specialty, Pharmacology, Placebo, Reuptake, Pharmacokinetics, Double-Blind Method, Internal medicine, medicine, Humans, Pharmacology (medical), Dosing, Serotonin Plasma Membrane Transport Proteins, Depressive Disorder, Major, Norepinephrine Plasma Membrane Transport Proteins, business.industry, Milnacipran, medicine.disease, Healthy Volunteers, Endocrinology, Area Under Curve, Delayed-Action Preparations, Major depressive disorder, Female, Serotonin, business, Reuptake inhibitor, Levomilnacipran, Selective Serotonin Reuptake Inhibitors
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المؤلفون: Bin Guo, Chuan Li, Guangji Wang, Laishun Chen
المصدر: Rapid Communications in Mass Spectrometry. 20:39-47
مصطلحات موضوعية: Male, Analyte, Fluoxetine, Time Factors, Chromatography, Metabolite, Organic Chemistry, Ultrafiltration, Blood proteins, Analytical Chemistry, Fluoxetine Hydrochloride, chemistry.chemical_compound, Dogs, Pharmacokinetics, chemistry, Pharmacodynamics, medicine, Animals, Spectroscopy, Protein Binding, medicine.drug
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المؤلفون: Robert K. Hofbauer, Antonia Periclou, Ramesh Boinpally, S. Zukin, Laishun Chen
المصدر: Alzheimer's & Dementia. 10
مصطلحات موضوعية: Epidemiology, business.industry, Health Policy, Fixed-dose combination, Memantine, Capsule, Phase i trials, Pharmacology, Psychiatry and Mental health, Cellular and Molecular Neuroscience, Developmental Neuroscience, Pharmacokinetics, medicine, Neurology (clinical), Geriatrics and Gerontology, Once daily, Extended release, Donepezil, business, medicine.drug
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المؤلفون: William M. Greenberg, Antonia Periclou, Ramesh Boinpally, Laishun Chen, Parviz Ghahramani, Julie Wangsa
المصدر: Clinical drug investigation. 34(5)
مصطلحات موضوعية: Adult, Cyclopropanes, Male, medicine.medical_specialty, Adolescent, Metabolite, Administration, Oral, Capsules, Pharmacology, chemistry.chemical_compound, Young Adult, Pharmacokinetics, Norepinephrine reuptake inhibitor, Internal medicine, medicine, Humans, Pharmacology (medical), Adverse effect, Aged, Dose-Response Relationship, Drug, business.industry, Liver Diseases, Milnacipran, General Medicine, Middle Aged, medicine.disease, Endocrinology, chemistry, Case-Control Studies, Delayed-Action Preparations, Major depressive disorder, Female, Liver function, business, Reuptake inhibitor, Levomilnacipran
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المؤلفون: Ming Yao, Nuggehally R. Srinivas, Laishun Chen
المصدر: Journal of Chromatography B: Biomedical Sciences and Applications. 752:9-16
مصطلحات موضوعية: Quality Control, Antifungal Agents, Chromatography, Chemistry, Reproducibility of Results, General Chemistry, Reversed-phase chromatography, Reference Standards, Triazoles, Mass spectrometry, Sensitivity and Specificity, High-performance liquid chromatography, Mass Spectrometry, Piperazines, Rats, Standard curve, chemistry.chemical_compound, Atmospheric Pressure, Liquid chromatography–mass spectrometry, Ammonium formate, Animals, Protein precipitation, Itraconazole, Quantitative analysis (chemistry), Chromatography, High Pressure Liquid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c4b722cbb38bb15cebd73c239c1f8cfb
https://doi.org/10.1016/s0378-4347(00)00505-3