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1دورية أكاديمية
المؤلفون: Cecilia Ansalone, Richard I. Ainsworth, Gyrid Nygaard, Rizi Ai, Edward B. Prideaux, Deepa Hammaker, Narayanan B. Perumal, Ken Weichert, Frances Tung, Lalitha Kodandapani, J. Michael Sauder, Elisabeth C. Mertsching, Robert J. Benschop, David L. Boyle, Wei Wang, Gary S. Firestein
المصدر: ACR Open Rheumatology, Vol 4, Iss 4, Pp 288-299 (2022)
مصطلحات موضوعية: Diseases of the musculoskeletal system, RC925-935
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2578-5745
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2
المؤلفون: Cecilia Ansalone, Richard I. Ainsworth, Gyrid Nygaard, Rizi Ai, Edward B. Prideaux, Deepa Hammaker, Narayanan B. Perumal, Ken Weichert, Frances Tung, Lalitha Kodandapani, J. Michael Sauder, Elisabeth C. Mertsching, Robert J. Benschop, David L. Boyle, Wei Wang, Gary S. Firestein
المصدر: ACR Open Rheumatology. 4:288-299
مصطلحات موضوعية: Rheumatology
وصف الملف: application/pdf
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3
المؤلفون: Kevin J. Tomaselli, Julia Herrmann, Robert O. Sayers, Joe C. Wu, Lalitha Kodandapani, Kathy G. Jahangiri, Craig D. Fisher, David T. Winn, Edward D. Robinson, Steven P. Meduna, Robert J. Ternansky, Pauline Yeo, Karen L. Valentino, Jose-Luis Diaz, Vincent J. Kalish, Steven D. Linton, Kristen Sebring, Robert A. Armstrong, Joseph F. Krebs, Niel C. Hoglen, Alfred P. Spada, Brad P. Hirakawa, Ning Chen, Brett R. Ullman, Brett Weylan Ching, Cheng-zhi Zhang, Xu Bai, Xin Gu, Kip Nalley, Long-Shiuh Chen, Patricia L. Gladstone, Jeff McQuiston, Teresa Aja, Todd Groessl, Donald S. Karanewsky, Suzanne Weeks, Lawrence C. Fritz, Patricia C. Contreras
المصدر: Journal of Medicinal Chemistry. 48:6779-6782
مصطلحات موضوعية: Adult, Biological Availability, Phases of clinical research, Apoptosis, Pharmacology, Jurkat Cells, Mice, Structure-Activity Relationship, Liver disease, Pharmacokinetics, In vivo, Drug Discovery, medicine, Animals, Humans, Aspartate Aminotransferases, Pentanoic Acids, Caspase, Liver injury, Cholestasis, Clinical Trials, Phase I as Topic, biology, Caspase 3, Chemistry, Liver Diseases, Alanine Transaminase, Hepatitis C, Chronic, medicine.disease, Caspase Inhibitors, In vitro, Rats, Liver, Biochemistry, Enzyme inhibitor, Hepatocytes, biology.protein, Molecular Medicine, Half-Life
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4
المؤلفون: Markus Tschopp, Mrudula Donepudi, Joe C. Wu, Lalitha Kodandapani, Markus G. Grütter, Helen Blanchard
المصدر: Journal of Molecular Biology. 302:9-16
مصطلحات موضوعية: Caspase-9, chemistry.chemical_classification, biology, Chemistry, Stereochemistry, Caspase 8, XIAP, Enzyme, Protein structure, Biochemistry, Structural Biology, biology.protein, Binding site, Molecular Biology, Caspase, Cysteine
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5
المؤلفون: Robert Smidt, Jose-Luis Diaz, Lalitha Kodandapani, Joe C. Wu, Brian Pham, Donald S. Karanewsky, Kevin J. Tomaselli, Robert J. Ternansky, Lawrence C. Fritz, Steven D. Linton
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:2969-2971
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Peptidomimetic, Acylation, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Drug Discovery, medicine, Enzyme Inhibitors, Molecular Biology, Caspase, chemistry.chemical_classification, biology, Chemistry, Organic Chemistry, Dipeptides, Caspase Inhibitors, In vitro, Isoenzymes, Enzyme, Enzyme inhibitor, biology.protein, Molecular Medicine, Indicators and Reagents, Oligopeptides, Lactone
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6
المؤلفون: Teresa Aja, Kevin J. Tomaselli, Edward D. Robinson, Joe C. Wu, Steven D. Linton, Xin Gu, Robert O. Sayers, Steven P. Meduna, Kip Nalley, Lalitha Kodandapani, Silvio Roggo, Vincent J. Kalish, Jose-Luis Diaz, Donald S. Karanewsky, Ning Chen, Albert Schmitz, Julia Herrmann, Brett R. Ullman, Joseph J. Krebs, Robert J. Ternansky
المصدر: Bioorganicmedicinal chemistry letters. 15(15)
مصطلحات موضوعية: Programmed cell death, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Naphthols, Cysteine Proteinase Inhibitors, Biochemistry, Chemical synthesis, Models, Biological, Mice, Structure-Activity Relationship, Heterocyclic Compounds, Drug Discovery, Animals, Molecular Biology, Caspase, Cells, Cultured, chemistry.chemical_classification, Aspartic Acid, biology, Bicyclic molecule, Cell Death, Organic Chemistry, Valine, Ketones, Caspase Inhibitors, In vitro, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Cellular model
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7
المصدر: Biochemistry. 42(14)
مصطلحات موضوعية: chemistry.chemical_classification, Models, Molecular, Caspase inhibitors, Binding Sites, biology, Sequence Homology, Amino Acid, Stereochemistry, Protein Conformation, Molecular Sequence Data, Biochemistry, Homology (biology), Recombinant Proteins, Amino acid, Structure-Activity Relationship, Protein structure, chemistry, Caspases, biology.protein, Structure–activity relationship, Humans, Amino Acid Sequence, Binding site, Peptide sequence, Caspase
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8
المؤلفون: Xian Guo, Robert J. Ternansky, Brett R. Ullman, Lawrence C. Fritz, Robert Smidt, Ning Chen, Albert Schmitz, Lalitha Kodandapani, Donald S. Karanewsky, Jose-Luis Diaz, Steven D. Linton, Vincent J. Kalish, Brian Pham, U. von Krosigk, Kathy G. Jahangiri, Kevin J. Tomaselli, Steven P. Meduna, Joe C. Wu, Silvio Roggo, Edward D. Robinson
المصدر: Bioorganicmedicinal chemistry letters. 12(20)
مصطلحات موضوعية: Stereochemistry, medicine.drug_class, Acylation, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Caspase 8, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Drug Discovery, medicine, Enzyme Inhibitors, Molecular Biology, Caspase, chemistry.chemical_classification, biology, Organic Chemistry, Dipeptides, Caspase Inhibitors, In vitro, Isoenzymes, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Indicators and Reagents, Oligopeptides, Lactone
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9
المؤلفون: Joe C. Wu, Kevin J. Tomaselli, Joseph F. Krebs, Lalitha Kodandapani, Peer R. E. Mittl, Helen Blanchard, Markus G. Grütter, Stefania Di Marco
المصدر: Structure. (9):1125-1133
مصطلحات موضوعية: Models, Molecular, Protein Conformation, drug design, Molecular Sequence Data, Apoptosis, inhibitor binding, Caspase 8, Crystallography, X-Ray, Substrate Specificity, 03 medical and health sciences, 0302 clinical medicine, Protein structure, Structural Biology, Zymogen, Protease Inhibitors, Amino Acid Sequence, Binding site, Protein Structure, Quaternary, Molecular Biology, Caspase, 030304 developmental biology, structure comparison, 0303 health sciences, Binding Sites, biology, Chemistry, Active site, Cysteine protease, Caspase Inhibitors, Caspase 9, Cell biology, Biochemistry, caspases, biology.protein, X-ray structure, Dimerization, Oligopeptides, 030217 neurology & neurosurgery
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::569978eccd67925895ed331123b9a1c4