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1
المؤلفون: Laura Llauger Bufi, Caterina Torrisi, Christian Steinkühler, Philip Jones, Claudia Giomini, Wu Hao, Sergio Serafini, Alberto Bresciani, Jesus Maria Ontoria Ontoria, Hu Bin, Michael Rowley
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:5274-5282
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, Dogs, Microsomes, Drug Discovery, Animals, Humans, Urea, Hedgehog Proteins, Molecular Biology, Hedgehog, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Antagonist, Stereoisomerism, Hedgehog signaling pathway, Rats, Novel agents, Molecular Medicine, Smoothened, Signal Transduction
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2
المؤلفون: Jesus Maria Ontoria Ontoria, Gabriella Dessole, Massimiliano Fonsi, Michael Rowley, Claudio Giuliano, Edith Monteagudo, Christian Steinkühler, Ester Muraglia, Caterina Torrisi, Maria Cecilia Palumbi, Danila Branca, Philip Jones, Laura Llauger Bufi, Alberto Bresciani
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:5283-5288
مصطلحات موضوعية: Molecular Structure, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Stereoisomerism, Amides, Smoothened Receptor, Biochemistry, Piperazines, Hedgehog signaling pathway, Receptors, G-Protein-Coupled, Structure-Activity Relationship, Piperazine, chemistry.chemical_compound, In vivo, Drug Discovery, Molecular Medicine, Amine gas treating, Signal transduction, Smoothened, Molecular Biology, Hedgehog
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3
المؤلفون: Fabrizio Fiore, Michael Rowley, Philip Jones, Odalys Gonzalez Paz, Massimiliano Fonsi, Edith Monteagudo, Olaf Kinzel, Carsten Schultz-Fademrecht, Christian Steinkühler, Giovanna Pescatore, Laura Llauger-Bufi
المصدر: Journal of Medicinal Chemistry. 52:3453-3456
مصطلحات موضوعية: Ketone, medicine.drug_class, Antineoplastic Agents, Mice, Dogs, Pharmacokinetics, In vivo, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Enzyme Inhibitors, Vorinostat, chemistry.chemical_classification, biology, Chemistry, Histone deacetylase inhibitor, Biological activity, Rats, Histone Deacetylase Inhibitors, Biochemistry, Enzyme inhibitor, Quinolines, biology.protein, Molecular Medicine, Histone deacetylase, Drug Screening Assays, Antitumor, HeLa Cells, medicine.drug
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4
المؤلفون: Philip Jones, Caterina Torrisi, Samuele Lillini, Olaf Kinzel, Costanza Bergami, Laura Llauger, Giovanna Pescatore
المصدر: Tetrahedron Letters. 50:172-177
مصطلحات موضوعية: chemistry.chemical_classification, Nucleophilic addition, Base (chemistry), Double bond, medicine.drug_class, Aryl, Organic Chemistry, Carboxamide, Biochemistry, Medicinal chemistry, chemistry.chemical_compound, chemistry, Intramolecular force, Drug Discovery, medicine, Hydroamination, Isomerization
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5
المؤلفون: Laura Llauger, Julia Aguirre, Nian Wu, Gabriela Chiosis, Joungnam Kim, Huazhong He, R.M. Immormino, Danuta Zatorska, Daniel T. Gewirth, Yuhong She
المصدر: Journal of Medicinal Chemistry. 49:381-390
مصطلحات موضوعية: Purine, Molecular Structure, biology, Chemistry, Water, Hsp90, In vitro, Structure-Activity Relationship, chemistry.chemical_compound, Solubility, Biochemistry, Purines, Cell Line, Tumor, Chaperone (protein), Heat shock protein, Drug Discovery, Cancer cell, biology.protein, Humans, Molecular Medicine, Structure–activity relationship, HSP90 Heat-Shock Proteins, Drug Screening Assays, Antitumor, Signal transduction, Cell Proliferation
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6
المؤلفون: Gabriela Chiosis, Neal Rosen, Julia Aguirre, Joungnam Kim, Peter Davies, Laura Llauger, Huazhong He, Ulf Peters
المصدر: Journal of Medicinal Chemistry. 48:2892-2905
مصطلحات موضوعية: Purine, Antineoplastic Agents, Binding, Competitive, Cell Line, Hsp90 inhibitor, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Cell Line, Tumor, Heat shock protein, Drug Discovery, Animals, Humans, Structure–activity relationship, HSP90 Heat-Shock Proteins, Sulfones, Sulfonyl, chemistry.chemical_classification, biology, Adenine, Hsp90, chemistry, Biochemistry, Sulfoxides, Chaperone (protein), Cancer cell, biology.protein, Molecular Medicine, Drug Screening Assays, Antitumor
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7
المؤلفون: Joan Bosch, Laura Llauger, Cecilia Juan, M.-Lluïsa Bennasar, Ester Zulaica
المصدر: Tetrahedron Letters. 40:3961-3964
مصطلحات موضوعية: Acylation, Nucleophile, Chemistry, Organic Chemistry, Drug Discovery, Trichloroacetic anhydride, chemistry.chemical_element, Organic chemistry, Biochemistry, Carbon, Adduct
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8
المؤلفون: J. C. Scaiano, Miguel A. Miranda, Laura Llauger, Gonzalo Cosa
المصدر: Organic Letters. 4:3083-3085
مصطلحات موضوعية: Anions, chemistry.chemical_classification, Photochemistry, Anti-Inflammatory Agents, Non-Steroidal, Organic Chemistry, Water, Protonation, Absolute rate, Hydrogen-Ion Concentration, Decarboxylation, Biochemistry, Carbon, Benzophenones, Kinetics, Reaction rate constant, chemistry, Ketoprofen, Computational chemistry, Protons, Physical and Theoretical Chemistry, Alkyl, Carbanion
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9
المؤلفون: M.-Lluïsa Bennasar, Joan Bosch, Ester Zulaica, Laura Llauger, Cecilia Juan
المصدر: ChemInform. 30
مصطلحات موضوعية: Acylation, Nucleophile, Chemistry, Trichloroacetic anhydride, Organic chemistry, chemistry.chemical_element, General Medicine, Carbon, Adduct
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10
المؤلفون: Samuele Lillini, Carsten Schultz-Fademrecht, Edith Monteagudo, Carlo Toniatti, Ester Muraglia, Olaf Kinzel, Caterina Torrisi, Danila Branca, Laura Llauger Bufi, Federica Ferrigno, Michael Rowley, Philip Jones
المصدر: Bioorganicmedicinal chemistry letters. 20(3)
مصطلحات موضوعية: Poly ADP ribose polymerase, Clinical Biochemistry, hERG, Poly (ADP-Ribose) Polymerase-1, Pharmaceutical Science, Poly(ADP-ribose) Polymerase Inhibitors, Biochemistry, Piperazines, Drug Discovery, Animals, Humans, Molecular Biology, chemistry.chemical_classification, biology, Chemistry, BRCA1 Protein, Organic Chemistry, Wild type, In vitro, Rats, Pyridazines, Enzyme, Enzyme inhibitor, Cancer cell, biology.protein, Microsome, Microsomes, Liver, Molecular Medicine, Poly(ADP-ribose) Polymerases, HeLa Cells