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1
المؤلفون: Oksana C. Palyha, Terry D. Faidley, Joseph M. Metzger, Xiao-Ming Guan, Sheng-Ping Wang, Jennifer A. Kosinski, Ravi P. Nargund, Stephanie K. Spann, Marc L. Reitman, Liming Yang, Linus S. Lin, Lauren P. Shearman, Kate A. Raustad, Donald J. Marsh, Kathy Lyons, Theresa M. Kelly, Stephanie Craw, Alison M. Strack, Yanqing Kan, Hong Yu, Jasminka Dragovic, Iyassu K. Sebhat
المصدر: Journal of Pharmacology and Experimental Therapeutics. 336:356-364
مصطلحات موضوعية: Male, Agonist, medicine.medical_specialty, medicine.drug_class, Blood Pressure, Pharmacology, Energy homeostasis, Rats, Sprague-Dawley, Eating, Mice, Dogs, Heart Rate, Weight loss, Internal medicine, medicine, Animals, Receptor, Dose-Response Relationship, Drug, Chemistry, Body Weight, Imidazoles, Rats, Bombesin receptor, Mice, Inbred C57BL, Receptors, Bombesin, Dose–response relationship, Blood pressure, Endocrinology, Pyrazoles, Molecular Medicine, Bombesin Receptor Subtype-3, Anti-Obesity Agents, medicine.symptom, Energy Metabolism
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4f83aba6c5ca83619726b27f1351081f
https://doi.org/10.1124/jpet.110.174763 -
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المؤلفون: Junying Wang, Richard G. Ball, Chun-Pyn Shen, Richard Z. Chen, Julie Lao, Vijay Bhasker G. Reddy, Xinchun Tong, Jeffrey J. Hale, Alison M. Strack, Jing Chen Xiao, Lauren P. Shearman, John S. Debenham, Tung M. Fong, D. Sloan Stribling, Christina B. Madsen-Duggan, Pei Huo, Lin Yan, Nancy N. Tsou, Thomas Bateman
المصدر: Journal of Medicinal Chemistry. 53:4028-4037
مصطلحات موضوعية: biology, Chemistry, medicine.drug_class, Stereochemistry, medicine.medical_treatment, Drug Inverse Agonism, hERG, Glucuronidation, Carboxamide, Pyrazole, Pharmacology, chemistry.chemical_compound, Drug Discovery, medicine, biology.protein, Molecular Medicine, Inverse agonist, Cannabinoid, Receptor
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المؤلفون: Marc L. Reitman, Cheng Guo, Theresa M. Kelly, Constantin Tamvakopoulos, Joseph M. Metzger, Tianying Jian, Howard Y. Chen, Arthur A. Patchett, Oksana C. Palyha, Alison M. Strack, Allan J. Goodman, Ravi P. Nargund, Peter H. Dobbelaar, Yanqing Kan, Mark Hadden, Larry Yet, Peter R. Guzzo, Qianping Peng, Linus S. Lin, Shuwen He, Lauren P. Shearman, Alan J. Henderson, Carina P. Tan, Sargent Bruce J, Xiao-Ming Guan, Scott D. Feighner, Iyassu K. Sebhat, Jie Pan, Jian Liu, Donald J. Marsh, Matthew J. Wyvratt, Andrew D. Howard, Megan Ruenz
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1913-1917
مصطلحات موضوعية: Agonist, medicine.drug_class, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Potency, Structure–activity relationship, Molecular Biology, Biphenyl, Chemistry, Drug discovery, fungi, Organic Chemistry, Imidazoles, Rats, Bombesin receptor, Bioavailability, Receptors, Bombesin, Molecular Medicine, Bombesin Receptor Subtype-3
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المؤلفون: Alison M. Strack, Xinchun Tong, Christina B. Madsen-Duggan, Lauren P. Shearman, Cathy R.-R.C. Huang, Mark T. Goulet, Thomas F. Walsh, Yue Feng, Jing Chen Xiao, D. Sloan Stribling, Junying Wang, John S. Debenham, Tung M. Fong, Chun-Pyn Shen, Sanjeev Kumar, Julie Lao, Donald J. Marsh, Richard B. Toupence
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1448-1452
مصطلحات موضوعية: Cannabinoid 1 receptor, Pyridines, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Receptor, Cannabinoid, CB1, Pharmacokinetics, Drug Discovery, Pyridine, medicine, Animals, Humans, Inverse agonist, Benzopyrans, Furans, Receptor, Molecular Biology, Biological evaluation, Mice, Knockout, Molecular Structure, Chemistry, Organic Chemistry, Haplorhini, Rats, Orally active, Drug Design, Molecular Medicine, Cannabinoid
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المؤلفون: Chun-Pyn Shen, C. DeMaula, Jing Chen Xiao, Julie Z. Lao, J. Shu, Lauren P. Shearman, J. Tyszkiewicz, A.C. Huber, Cathy C. R.-R. Huang, Alison M. Strack, A. Galijatovic-Idrizbegovic, C.L. Lanning, Tung M. Fong, D.S. Stribling, M.-F. Hubert, R. Owen
المصدر: Drug Development Research. 70:349-362
مصطلحات موضوعية: Drug, Cannabinoid receptor, medicine.medical_treatment, media_common.quotation_subject, Pharmacology, Biology, Safety profile, Taranabant, Rimonabant, In vivo, Drug Discovery, medicine, Inverse agonist, Cannabinoid, medicine.drug, media_common
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المؤلفون: Junying Wang, Jing Chen Xiao, D. Sloan Stribling, Marie-Therese Schaeffer, Alison M. Strack, Lauren P. Shearman, Cathy C. R.-R. Huang, D. Euan MacIntyre, Thomas F. Walsh, Christina B. Madsen-Duggan, Chun-Pyn Shen, John S. Debenham, Jeffrey J. Hale, Tung M. Fong, Julie Lao, Xinchun Tong
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:2591-2594
مصطلحات موضوعية: Cannabinoid receptor, Chemistry, Pharmaceutical, medicine.medical_treatment, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Biochemistry, Chemical synthesis, Receptor, Cannabinoid, CB2, Inhibitory Concentration 50, Structure-Activity Relationship, Receptor, Cannabinoid, CB1, Drug Discovery, medicine, Animals, Humans, Inverse agonist, Structure–activity relationship, Obesity, Receptor, Molecular Biology, Cannabinoid Receptor Agonists, Cannabinoids, Chemistry, Organic Chemistry, Biological activity, Protein Structure, Tertiary, Rats, Pyrimidines, Drug Design, Molecular Medicine, Cannabinoid
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المؤلفون: Sloan Stribling, Donald F. Thompson, Junying Wang, Xinchun Tong, Lauren P. Shearman, Cathy C. R.-R. Huang, Joana Achanfuo-Yeboah, Susan Nicolich, Andrea Frassetto, Tung M. Fong, Donald F. Hora, Chun-Pyn Shen, Nancy N. Tsou, Alison M. Strack, Richard G. Ball, Julie Lao, Gerard J. Hickey, Terry D. Faidley, Jeffrey J. Hale, Joan M. Fletcher, William K. Hagmann, Petr Vachal, Richard Z. Chen, Jing Chen Xiao
المصدر: Journal of Medicinal Chemistry. 52:2550-2558
مصطلحات موضوعية: Models, Molecular, Drug Inverse Agonism, medicine.medical_treatment, Biological Availability, In Vitro Techniques, Pharmacology, Piperazines, Eating, Structure-Activity Relationship, Dogs, Receptor, Cannabinoid, CB1, In vivo, Drug Discovery, medicine, Animals, Humans, Potency, Inverse agonist, Structure–activity relationship, Receptor, Sulfonamides, Chemistry, Body Weight, Antagonist, Stereoisomerism, Macaca mulatta, Rats, Biochemistry, Hepatocytes, Microsomes, Liver, Molecular Medicine, Anti-Obesity Agents, Cannabinoid
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المؤلفون: D. Euan MacIntyre, Yue Feng, Lauren P. Shearman, Xiao-Ming Guan, Mark T. Goulet, Christopher W. Plummer, Sharon Tong, Quang Truong, D. Sloan Stribling, Donald J. Marsh, Junying Wang, Hong Yu, Kimberly Rosko, Sander G. Mills, Paul E. Finke, Alison M. Strack, Stephanie K. Spann, L. H. T. Van Der Ploeg, Shrenik K. Shah, Douglas J. MacNeil, Ramon E. Camacho, Joseph M. Metzger, William K. Hagmann, Tung M. Fong
المصدر: European Journal of Pharmacology. 579:215-224
مصطلحات موضوعية: Male, medicine.medical_specialty, Cannabinoid receptor, Drug Inverse Agonism, medicine.drug_class, medicine.medical_treatment, Administration, Oral, In Vitro Techniques, Rats, Sprague-Dawley, Receptor, Cannabinoid, CB2, Eating, Mice, Dexfenfluramine, Receptor, Cannabinoid, CB1, In vivo, Internal medicine, medicine, Animals, Humans, Inverse agonist, Obesity, Receptor, Mice, Knockout, Pharmacology, Dose-Response Relationship, Drug, Chemistry, Imidazoles, Brain, Receptor antagonist, Rats, Disease Models, Animal, Endocrinology, Autoradiography, Anti-Obesity Agents, Cannabinoid, Ex vivo, Protein Binding, medicine.drug
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المؤلفون: Tung M. Fong, Helen E. Armstrong, Thomas J. Lanza, Sookhee Ha, Julie Lao, James P. Jewell, Quang Truong, Lauren P. Shearman, Vincent J. Colandrea, Grace M. Quaker, William K. Hagmann, Guthikonda Ravi N, D. Sloan Stribling, Junying Wang, Chun-Pyn Shen, Sherry Xu, Linus S. Lin, Amy Galka, Xinchun Tong, Mark T. Goulet, Shrenik K. Shah, Linda L. Chang, Lex H.T. Van der Ploeg, Alison M. Strack, Jing Chen, Kimberly Rosko
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:2184-2187
مصطلحات موضوعية: Stereochemistry, medicine.drug_class, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Hypothermia, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Taranabant, Receptor, Cannabinoid, CB1, Amide, Cannabinoid Receptor Modulators, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Potency, Inverse agonist, Pharmacokinetics, Molecular Biology, Brain Chemistry, chemistry.chemical_classification, Sulfonamides, Organic Chemistry, Rats, Sulfonamide, chemistry, Molecular Medicine, Anti-Obesity Agents, Cannabinoid, medicine.drug
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المؤلفون: Xinchun Tong, Yue Feng, Lauren P. Shearman, William K. Hagmann, Koppara Samuel, Jing Chen Xiao, Shrenik K. Shah, Hongbo Qi, Junying Wang, Sanjeev Kumar, Kimberly Rosko, Tung M. Fong, Wenji Yin, Ping Liu, D. Sloan Stribling, Linus S. Lin, Alison M. Strack, Chun-Pyn Shen, Julie Lao, Donald J. Marsh, James P. Jewell, Lex H.T. Van der Ploeg, Thomas J. Lanza, Mark T. Goulet, Suoyu S. Xu
المصدر: Journal of Medicinal Chemistry. 49:7584-7587
مصطلحات موضوعية: Trifluoromethyl, Stereochemistry, Propanamide, Chemical synthesis, chemistry.chemical_compound, Taranabant, chemistry, In vivo, Amide, Drug Discovery, medicine, Molecular Medicine, Inverse agonist, Receptor, medicine.drug