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1
المؤلفون: David G. Breckenridge, Laurie A. Castonguay, Giuseppe A. Papalia, Swetha Pendem, Shawn S. Badal, Ford Hinojosa-Kirschenbaum, Gregory T. Notte, Sarah Wise, Michael V. Lee, Keith A. Koch, Agnes B. Fogo, Dorothy French, Britton Kenneth Corkey, Frank Y. Ma, Brian E. Schultz, Eric B. Lansdon, Melanie H. Wong, David J. Nikolic-Paterson, Tareq M Al-Tuhaifi, Theodore Sullivan, Michael Graupe, Haichun Yang, Erik Huntzicker, Grant R. Budas, John T. Liles
المصدر: Journal of Clinical Investigation. 128:4485-4500
مصطلحات موضوعية: Male, 0301 basic medicine, Nephrology, medicine.medical_specialty, MAP Kinase Signaling System, Kidney Glomerulus, Renal function, MAP Kinase Kinase Kinase 5, Rats, Sprague-Dawley, Mice, Random Allocation, 03 medical and health sciences, Fibrosis, Internal medicine, medicine, Animals, Humans, Diabetic Nephropathies, ASK1, Protein Kinase Inhibitors, Mice, Knockout, Serine/threonine-specific protein kinase, Kidney, business.industry, Glomerulosclerosis, General Medicine, Fibroblasts, medicine.disease, Oxidative Stress, Disease Models, Animal, 030104 developmental biology, medicine.anatomical_structure, Cancer research, Female, business, Research Article, Kidney disease
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2
المؤلفون: Erinn E. Pagratis, Benjamin A. Turner, Xiaohong Liu, Kelly R. Pitts, Q. Khai Huynh, Nikos Pagratis, Laurie A. Castonguay, Sarah Wise, David Koditek, Christopher B. Glascock, Keith A. Koch, Brian Reid, Magdeleine Hung, Bin Han
المصدر: SLAS Discovery. 16:724-733
مصطلحات موضوعية: Fluoroimmunoassay, Molecular Conformation, Receptor, Transforming Growth Factor-beta Type I, Smad Proteins, Protein Serine-Threonine Kinases, Mitogen-activated protein kinase kinase, Biochemistry, Analytical Chemistry, MAP2K7, Small Molecule Libraries, Growth factor receptor, Transforming Growth Factor beta, Cell Line, Tumor, Fluorescence Resonance Energy Transfer, Humans, Computer Simulation, Phosphorylation, Protein Kinase Inhibitors, biology, Cyclin-dependent kinase 4, Chemistry, Cyclin-dependent kinase 2, Molecular biology, High-Throughput Screening Assays, Adenosine Diphosphate, Kinetics, biology.protein, Molecular Medicine, Cyclin-dependent kinase 9, Receptors, Transforming Growth Factor beta, Platelet-derived growth factor receptor, ACVR2B, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::51895707278fcc75e88009c53f1325d5
https://doi.org/10.1177/1087057111405846 -
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المؤلفون: Laurie G. Castonguay, Sookhee Ha, Lex H.T. Van der Ploeg, Chun-Pyn Shen, Ihor E. Kopka, Zhege J. Lao, Mark T. Goulet, Linus S. Lin, William K. Hagmann, Tung M. Fong, James P. Jewell, Thomas J. Lanza
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:4757-4761
مصطلحات موضوعية: Models, Molecular, Molecular model, Pyridines, medicine.drug_class, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Carboxamide, Context (language use), Biochemistry, Chemical synthesis, Taranabant, Receptor, Cannabinoid, CB1, Drug Discovery, medicine, Humans, Inverse agonist, Computer Simulation, Homology modeling, Molecular Biology, Chemistry, Organic Chemistry, Amides, Molecular Medicine, Anti-Obesity Agents, Cannabinoid, Protein Binding, medicine.drug
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4
المصدر: Protein Science. 4:472-483
مصطلحات موضوعية: Models, Molecular, Protein Folding, Protein Conformation, Globular protein, Cell Adhesion Molecules, Neuronal, Molecular Sequence Data, Immunoglobulins, Biology, Biochemistry, Domain (software engineering), Protein sequencing, Molecular recognition, Animals, Drosophila Proteins, Computer Simulation, Amino Acid Sequence, Homology modeling, Molecular Biology, Integral membrane protein, chemistry.chemical_classification, Sequence Homology, Amino Acid, Protein structure prediction, Peptide Fragments, chemistry, CD4 Antigens, Immunoglobulin superfamily, Drosophila, Algorithm, Algorithms, Research Article
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5
المؤلفون: Gloria C. Koo, Laurie A. Castonguay, Mary Jo Staruch, Randal M. Bugianesi, John P. Felix, George A. Doss, Robert S. Slaughter, Marty S. Springer, Andrew Kotliar, Sookhee Ha, Kathleen M. Rupprecht, William H. Parsons, Gregory J. Kaczorowski, Kashmira Shah, Shouwu Miao, Jianming Bao, Maria L. Garcia, Frank Kayser, Robert K. Baker
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:447-451
مصطلحات موضوعية: Models, Molecular, Stereochemistry, T-Lymphocytes, T cell, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Potassium Channel Blockers, medicine, Humans, Channel blocker, Molecular Biology, Cell Proliferation, Kv1.3 Potassium Channel, Natural product, Cell growth, Organic Chemistry, Triterpenes, Potassium channel, In vitro, medicine.anatomical_structure, chemistry, Potassium Channels, Voltage-Gated, Molecular Medicine, Biological Assay, Ion Channel Gating, Enone, Immunosuppressive Agents, Ion channel blocker
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6
المؤلفون: M. Maccoss, Paul E. Finke, Bruce L. Daugherty, Youmin Weng, Di Salvo J, Julie A. DeMartino, Christopher L. Lynch, Laurie A. Castonguay, Marty S. Springer, J. J. Hale, Sander G. Mills, Adolfsen W, Charles G. Caldwell, Ruth Kilburn
المصدر: Biochemistry. 42:1544-1550
مصطلحات موضوعية: Models, Molecular, Rhodopsin, Pyrrolidines, Receptors, CCR5, Molecular model, Stereochemistry, Chemokine receptor CCR5, Molecular Sequence Data, CHO Cells, Binding, Competitive, Biochemistry, Protein Structure, Secondary, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Cricetinae, Animals, Humans, Amino Acid Sequence, Binding site, Alanine, Binding Sites, Sequence Homology, Amino Acid, biology, Aryl, Amides, Quaternary Ammonium Compounds, Transmembrane domain, Amino Acid Substitution, chemistry, Docking (molecular), CCR5 Receptor Antagonists, Butanes, Mutagenesis, Site-Directed, biology.protein, Cattle, Pharmacophore
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7
المصدر: Bioconjugate Chemistry. 10:958-964
مصطلحات موضوعية: Gadolinium DTPA, Models, Molecular, Relaxometry, Chemical Phenomena, Gadolinium, Molecular Conformation, Biomedical Engineering, Contrast Media, Pharmaceutical Science, chemistry.chemical_element, Bioengineering, Structure-Activity Relationship, Nuclear magnetic resonance, Drug Stability, Heterocyclic Compounds, Organometallic Compounds, medicine, Molecule, Chelation, Edetic Acid, Chelating Agents, Pharmacology, medicine.diagnostic_test, Chemistry, Physical, Organic Chemistry, Magnetic resonance imaging, Magnetic Resonance Imaging, chemistry, Solvents, Linear correlation, Crystallization, Algorithms, Software, Biotechnology
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المؤلفون: Laurie A. Castonguay, Ian W. Davies, Thomas R. Verhoeven, Paul J. Reider, Chris H. Senanayake, Robert D. Larsen
المصدر: Tetrahedron Letters. 36:7619-7622
مصطلحات موضوعية: Chiral auxiliary, chemistry.chemical_compound, Chemistry, Stereochemistry, Organic Chemistry, Drug Discovery, Biochemistry, Diels–Alder reaction
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المؤلفون: Laurie A. Castonguay, Ian W. Davies, Chris H. Senanayake, Robert D. Larsen, Thomas R. Verhoeven, Paul J. Reider
المصدر: ChemInform. 27
مصطلحات موضوعية: Chiral auxiliary, chemistry.chemical_compound, chemistry, Stereochemistry, General Medicine, Diels–Alder reaction
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المؤلفون: L. Gerena, Paul J. Reider, Chris H. Senanayake, Ian W. Davies, Thomas R. Verhoeven, Laurie A. Castonguay, Robert D. Larsen
المصدر: ChemInform. 27
مصطلحات موضوعية: Chemistry, Ligand, Diels alder, chemistry.chemical_element, General Medicine, Bite angle, Medicinal chemistry, Copper, Catalysis