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1
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:43-47
مصطلحات موضوعية: Chemistry, Sodium channel, NAV1.7 Voltage-Gated Sodium Channel, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Rats, Electrophysiology, Sodium channel blocker, Dibenzazepines, Drug Discovery, Neuropathic pain, Dibenzoxazepines, Microsomes, Liver, Animals, Humans, Molecular Medicine, Potency, Molecular Biology, Sodium Channel Blockers
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2
المؤلفون: Yasuyoshi Iso, Shintani Takuya, John J. Engel, Akira Kato, Jianming Yu, Tsuyoshi Hasegawa, Toshiyuki Asaki, Yoshitaka Yamaguchi, Naoki Tsuno, Laykea Tafesse, Chiyou Ni, Noriyuki Kurose, Kevin C. Brown, Toshiyuki Kanemasa, Gang Wu, Manjunath S. Shet, Yuka Iwamoto, Aniket Patel, Donald J. Kyle, Xiaoming Zhou
المصدر: Journal of Medicinal Chemistry. 57:6781-6794
مصطلحات موضوعية: Trifluoromethyl, medicine.drug_class, Stereochemistry, TRPV1, Antagonist, Carboxamide, Pharmacology, chemistry.chemical_compound, chemistry, Pharmacokinetics, Capsaicin, In vivo, Drug Discovery, medicine, Molecular Medicine, Structure–activity relationship, lipids (amino acids, peptides, and proteins)
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3
المؤلفون: Kevin P. Carlin, Toshiyuki Kanemasa, Laykea Tafesse, Victor I. Ilyin, Gang Wu, Toshiyuki Asaki
المصدر: Biophysical Journal. 108(2)
مصطلحات موضوعية: Hyperthermia, Chemistry, Drug discovery, Analgesic, Antagonist, TRPV1, Biophysics, Endogeny, Pharmacology, medicine.disease, 3. Good health, chemistry.chemical_compound, Capsaicin, medicine, Receptor
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4
المؤلفون: Khondekar Islam, Laykea Tafesse, Qun Sun, James T. Limberis, Donald J. Kyle
المصدر: Combinatorial Chemistry & High Throughput Screening. 6:481-488
مصطلحات موضوعية: Stereochemistry, Sodium channel, Organic Chemistry, Single step, General Medicine, Condensation reaction, Combinatorial chemistry, Membrane Potentials, Computer Science Applications, Chemical library, Sodium Channel Antagonists, Xenopus laevis, chemistry.chemical_compound, Anticonvulsant Agent, chemistry, Drug Discovery, Animals, Combinatorial Chemistry Techniques, Female, Antagonism, Sodium Channel Blockers
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3571f3a68f107b9747e6e2591857fd03
https://doi.org/10.2174/138620703106298653 -
5
المؤلفون: Petros Gebreselassie, Anne M. Hudrlik, Paul F. Hudrlik, Laykea Tafesse
المصدر: Tetrahedron Letters. 44:3409-3412
مصطلحات موضوعية: Silanes, Silicon, Organic Chemistry, chemistry.chemical_element, Biochemistry, Medicinal chemistry, chemistry.chemical_compound, Elimination reaction, Stereospecificity, chemistry, Drug Discovery, Alkoxide, β elimination, Organic chemistry
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6
المؤلفون: Kevin P. Carlin, Haissam Abdelhamid, Parijat Ghatak, Stephen M. Lynch, Bin Shao, Donald J. Kyle, Laykea Tafesse
المصدر: Bioorganicmedicinal chemistry letters. 25(1)
مصطلحات موضوعية: Cell Membrane Permeability, Clinical Biochemistry, hERG, Molecular Sequence Data, Pharmaceutical Science, Pharmacology, Biochemistry, Cns penetration, Madin Darby Canine Kidney Cells, chemistry.chemical_compound, Sodium channel blocker, Dogs, Drug Discovery, Potency, Animals, Amino Acid Sequence, Molecular Biology, biology, Chemistry, Sodium channel, Aryl, Organic Chemistry, NAV1.7 Voltage-Gated Sodium Channel, Rats, Electrophysiology, biology.protein, Molecular Medicine, Selectivity, Sodium Channel Blockers
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7
المؤلفون: Laykea, Tafesse, Toshiyuki, Kanemasa, Noriyuki, Kurose, Jianming, Yu, Toshiyuki, Asaki, Gang, Wu, Yuka, Iwamoto, Yoshitaka, Yamaguchi, Chiyou, Ni, John, Engel, Naoki, Tsuno, Aniket, Patel, Xiaoming, Zhou, Takuya, Shintani, Kevin, Brown, Tsuyoshi, Hasegawa, Manjunath, Shet, Yasuyoshi, Iso, Akira, Kato, Donald J, Kyle
المصدر: Journal of medicinal chemistry. 57(15)
مصطلحات موضوعية: Male, Analgesics, Sensory Receptor Cells, Freund's Adjuvant, Aminopyridines, Pain, TRPV Cation Channels, Stereoisomerism, CHO Cells, Hydrogen-Ion Concentration, Body Temperature, Rats, Sprague-Dawley, Structure-Activity Relationship, Cricetulus, Ganglia, Spinal, Animals, Humans, Calcium, Capsaicin
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8
المؤلفون: Kenneth J. Valenzano, Laykea Tafesse, David A. Elsemore, Jamie Boulet, Shen Shan, Lilly Mark, Leyana Rabadi, Paul I. Turchin, Gary Lee, Garth Whiteside, Mathew Toth, Suzanne M. Chaffer, Susan L. Gottshall, James E. Harrison, Lee Koetzner, Michelle S. Pearson, Yakov Rotshteyn, Wendy S. Miller
المصدر: Neuropharmacology. 48(5)
مصطلحات موضوعية: Male, Cannabinoid receptor, Indoles, Time Factors, Cyclohexanecarboxylic Acids, medicine.medical_treatment, Indomethacin, Pharmacology, Anxiety, Rats, Sprague-Dawley, Receptor, Cannabinoid, CB2, Mice, Cricetinae, Cannabinoid receptor type 2, Cyclic AMP, Amines, gamma-Aminobutyric Acid, Pain Measurement, Mice, Knockout, Analgesics, Behavior, Animal, Chemistry, Anti-Inflammatory Agents, Non-Steroidal, Chronic pain, Cannabinoid Receptor Agonists, Hyperalgesia, lipids (amino acids, peptides, and proteins), medicine.symptom, Gabapentin, Immunosuppressive Agents, Agonist, medicine.drug_class, Morpholines, Pain, CHO Cells, Naphthalenes, Partial agonist, Binding, Competitive, Cellular and Molecular Neuroscience, Cricetulus, medicine, Reaction Time, Animals, Humans, Inflammation, Catalepsy, Dose-Response Relationship, Drug, medicine.disease, Cyclohexanols, Benzoxazines, Rats, Disease Models, Animal, Ataxia, Cannabinoid, Excitatory Amino Acid Antagonists, Psychomotor Performance
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9
المؤلفون: Kenneth J. Valenzano, Xin Su, Donald J. Kyle, Lori Schmid, Laykea Tafesse, Yakov Rotshteyn, Qun Sun
المصدر: Bioorganicmedicinal chemistry letters. 14(22)
مصطلحات موضوعية: Time Factors, Stereochemistry, medicine.drug_class, Pyridines, Receptors, Drug, Clinical Biochemistry, TRPV1, Drug Evaluation, Preclinical, Pharmaceutical Science, TRPV Cation Channels, Carboxamide, Pharmacology, Biochemistry, Chemical synthesis, Piperazines, Chemical library, Cell Line, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Receptor, Molecular Biology, Molecular Structure, Organic Chemistry, Antagonist, Biological activity, Pyridazines, chemistry, Pyrazines, Molecular Medicine, Lead compound
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10
المؤلفون: Laykea Tafesse, Donald J. Kyle
المصدر: Combinatorial chemistryhigh throughput screening. 7(2)
مصطلحات موضوعية: Molecular Structure, Organic Chemistry, Total synthesis, General Medicine, Benzazepines, Combinatorial chemistry, Computer Science Applications, Benzazepine, chemistry.chemical_compound, chemistry, Drug Discovery, Tetralone, Schmidt reaction, Capsaicin, Capsazepine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::62e7b18e5e180197a317a6545554323a
https://pubmed.ncbi.nlm.nih.gov/15032662