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1
المؤلفون: Deirdre M. B. Hickey, Ian Stansfield, Leach Colin Andrew, Caroline M. Whittaker, Ivan Leo Pinto, Stephen A. Smith, Stephen Christopher Martin Fell, Sean Thomas Flynn, Kitty Moores, Helen F. Boyd, Colin J. Theobald, David G. Tew, Roderick A. Porter, Robert John Ife, Kevin J. Milliner, Colin H. Macphee, D. Anthony Rawlings
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:2557-2561
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Lipoproteins, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Carboxamide, Pyrimidinones, Biochemistry, Chemical synthesis, Phospholipases A, chemistry.chemical_compound, Phospholipase A2, Oral administration, Drug Discovery, medicine, Animals, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Molecular Structure, biology, Chemistry, Lipoprotein-associated phospholipase A2, Organic Chemistry, Phospholipases A2, Enzyme, Enzyme inhibitor, biology.protein, Lactam, Molecular Medicine, Rabbits
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2
المؤلفون: Martin Jones, Colin J. Theobald, Leach Colin Andrew, Sean Thomas Flynn, Deirdre M. B. Hickey, Ian Stansfield, David G. Tew, Brian Peter Slingsby, Helen F. Boyd, Stephen A. Smith, Kevin J. Milliner, Colin H. Macphee, Robert John Ife, D. Anthony Rawlings
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:395-398
مصطلحات موضوعية: Stereochemistry, High-throughput screening, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Pyrimidinones, Biochemistry, Chemical synthesis, Phospholipases A, Substrate Specificity, Inhibitory Concentration 50, Structure-Activity Relationship, Phospholipase A2, Drug Discovery, Humans, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, biology, Chemistry, Lipoprotein-associated phospholipase A2, Organic Chemistry, Substrate (chemistry), Phospholipases A2, Enzyme, Enzyme inhibitor, Drug Design, 1-Alkyl-2-acetylglycerophosphocholine Esterase, biology.protein, Molecular Medicine, Selectivity
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3
المؤلفون: Helen F. Boyd, Deirdre M. B. Hickey, Kitty Moores, Kevin J. Milliner, Colin H. Macphee, Dash Dhanak, Keith E. Suckling, Leach Colin Andrew, Rebecca A. Patterson, Robert John Ife, David S. Leake, David G. Tew
المصدر: Biochemical Journal. 338:479-487
مصطلحات موضوعية: chemistry.chemical_classification, biology, Lipoprotein-associated phospholipase A2, Fatty acid, Cell Biology, 1-Alkyl-2-acetylglycerophosphocholine Esterase, Biochemistry, chemistry.chemical_compound, Phospholipase A2, Lysophosphatidylcholine, chemistry, Low-density lipoprotein, biology.protein, lipids (amino acids, peptides, and proteins), Chemoattractant activity, Molecular Biology, Lipoprotein
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::fbda5ac7d34f8ba6f99f2e2fc0fda486
https://doi.org/10.1042/bj3380479 -
4
المصدر: Biochemistry. 37:10087-10093
مصطلحات موضوعية: Lactams, Stereochemistry, Kinetics, beta-Lactams, Biochemistry, Phospholipases A, Substrate Specificity, Hydrolysis, Phospholipase A2, Peptide bond, Lipase, Chromatography, High Pressure Liquid, biology, Chemistry, Spectrum Analysis, Stereoisomerism, Enzyme Activation, Lipoproteins, LDL, Phospholipases A2, Burst kinetics, Covalent bond, 1-Alkyl-2-acetylglycerophosphocholine Esterase, biology.protein, Azetidines, Enantiomer
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5
المؤلفون: Leach Colin Andrew, Robert John Ife, A.J. Pope, C.J. Theobald
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:543-546
مصطلحات موضوعية: Bicyclic molecule, biology, Stereochemistry, ATPase, Organic Chemistry, Clinical Biochemistry, Quinoline, Gastric H+/K+ ATPase, Pharmaceutical Science, Protonation, Biochemistry, chemistry.chemical_compound, chemistry, Drug Discovery, Pyridine, biology.protein, Molecular Medicine, Molecule, Thiazole, Molecular Biology
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6
المؤلفون: David J. Keeling, M. E. Parsons, Robert John Ife, S. M. Laing, C. A. Price, K. J. Wiggall, Leach Colin Andrew, T. H. Brown
المصدر: ChemInform. 24
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Stereochemistry, Gastric H+/K+ ATPase, Substituent, General Medicine
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7
المؤلفون: Leach Colin Andrew, David G. Tew, Deirdre M. B. Hickey, Stephen A. Smith, Robert John Ife, Colin H. Macphee
المصدر: ChemInform. 32
مصطلحات موضوعية: chemistry.chemical_classification, biology, Monocyte, General Medicine, Pharmacology, Proinflammatory cytokine, chemistry.chemical_compound, Enzyme, medicine.anatomical_structure, Phospholipase A2, chemistry, Low-density lipoprotein, Phosphatidylcholine, biology.protein, medicine, lipids (amino acids, peptides, and proteins), Lipase, Lipoprotein
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8
المؤلفون: Leach Colin Andrew, David R. Reavill, Kenneth Wiggall, Colin J. Theobald, David J. Keeling, Robert John Ife, Thomas Henry Brown, Malcolm L. Meeson, Michael E. Parsons
المصدر: Journal of Medicinal Chemistry. 35:3413-3422
مصطلحات موضوعية: Stereochemistry, Substituent, Gastric Acid, H(+)-K(+)-Exchanging ATPase, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, In vivo, Drug Discovery, Animals, Enzyme Inhibitors, Adenosine Triphosphatases, chemistry.chemical_classification, biology, Bicyclic molecule, Hydrogen bond, Quinoline, Rats, Enzyme, chemistry, Gastric Mucosa, Enzyme inhibitor, Quinolines, biology.protein, Molecular Medicine, Gastric acid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::79cebd31e4331d8b5aab573022f2e5ce
https://doi.org/10.1021/jm00096a018 -
9
المؤلفون: Michael E. Parsons, Leach Colin Andrew, Kenneth Wiggall, David J. Keeling, Thomas Henry Brown, Carolyn A. Price, Shiona M. Laing, Robert John Ife
المصدر: Journal of Medicinal Chemistry. 35:1845-1852
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, Stereochemistry, Substituent, Reversible reaction, H(+)-K(+)-Exchanging ATPase, chemistry.chemical_compound, Dogs, In vivo, Drug Discovery, Animals, Adenosine Triphosphatases, chemistry.chemical_classification, biology, Stomach, Biological activity, In vitro, Rats, Enzyme Activation, Enzyme, chemistry, Enzyme inhibitor, Aminoquinolines, biology.protein, Molecular Medicine, Gastric acid, Pentagastrin
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::634fc359e90b5a4b3a2eb6a38fac940b
https://doi.org/10.1021/jm00088a021 -
10
المؤلفون: Leach Colin Andrew, David J. Keeling, Colin J. Theobald, Malcolm L. Meeson, Robert John Ife, Michael E. Parsons, Peter Blurton, Thomas Henry Brown
المصدر: Journal of medicinal chemistry. 38(14)
مصطلحات موضوعية: chemistry.chemical_classification, Magnetic Resonance Spectroscopy, biology, Bicyclic molecule, Stereochemistry, Chemistry, ATPase, Stomach, Substituent, Proton Pump Inhibitors, H(+)-K(+)-Exchanging ATPase, Chemical synthesis, In vitro, Rats, chemistry.chemical_compound, Structure-Activity Relationship, Enzyme, Dogs, Pyrimidines, Enzyme inhibitor, Drug Discovery, biology.protein, Quinazolines, Molecular Medicine, Animals
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c4916b337cd6a2d8d714e94e54e26f02
https://pubmed.ncbi.nlm.nih.gov/7629814