-
1
المؤلفون: Walter G. Smith, Suzanne H Kim, Doreen Villani-Price, Matthew W Mahoney, Nayereh S Ghoreishi-Haack, Helen Y. Chen, Thomas D. Penning, Stella Siu-Tzyy Yu, James W. Malecha, Leslie J Askonas, Chi-Dean Liang, Elizabeth I Harding, E.Yvonne Pyla, Maureen K Highkin, James K. Gierse, Julie M Miyashiro, Mark A Russell, James F Kachur, Chen Barbara B
المصدر: Journal of Medicinal Chemistry. 45:3482-3490
مصطلحات موضوعية: Epoxide Hydrolases, chemistry.chemical_classification, biology, Stereochemistry, Administration, Oral, Leukotriene A4, Chemical synthesis, Proinflammatory cytokine, Leukotriene-A4 hydrolase, Mice, Structure-Activity Relationship, Enzyme, chemistry, Enzyme inhibitor, In vivo, Drug Discovery, Hydrolase, beta-Alanine, biology.protein, Animals, Humans, Molecular Medicine, Structure–activity relationship, Enzyme Inhibitors
-
2
المؤلفون: Leslie J Askonas, Mark A Russell, Walter G. Smith, James F. Kachur, Chi-Dean D. Liang, D Villani-Price
المصدر: Journal of Pharmacology and Experimental Therapeutics. 300:577-582
مصطلحات موضوعية: beta-Alanine, Enzyme-Linked Immunosorbent Assay, In Vitro Techniques, Pharmacology, Aminopeptidases, Substrate Specificity, Mice, chemistry.chemical_compound, Dogs, Species Specificity, In vivo, Hydrolase, Animals, Humans, Enzyme Inhibitors, Epoxide hydrolase, Chromatography, High Pressure Liquid, Epoxide Hydrolases, Leukotriene, Arachidonic Acid, Ionophores, Leukotriene A4, Macaca mulatta, Recombinant Proteins, Rats, Kinetics, chemistry, Biochemistry, Eicosanoids, Leukotriene Antagonists, Molecular Medicine, Arachidonic acid, Ex vivo
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8a43488c1feb896fd592f6e43e83a9e0
https://doi.org/10.1124/jpet.300.2.577 -
3
المؤلفون: Thomas D. Penning, Nizal S. Chandrakumar, Barbara B. Chen, Helen Y. Chen, Bipin N. Desai, Stevan W. Djuric, Stephen H. Docter, Alan F. Gasiecki, Richard A. Haack, Julie M. Miyashiro, Mark A. Russell, Stella S. Yu, David G. Corley, Richard C. Durley, Brian F. Kilpatrick, Barry L. Parnas, Leslie J. Askonas, James K. Gierse, Elizabeth I. Harding, Maureen K. Highkin, James F. Kachur, Suzanne H. Kim, Gwen G. Krivi, Doreen Villani-Price, E. Yvonne Pyla, Walter G. Smith, Nayereh S. Ghoreishi-Haack
المصدر: Journal of Medicinal Chemistry. 43:721-735
مصطلحات موضوعية: Male, Pyrrolidines, Tertiary amine, Administration, Oral, In Vitro Techniques, Pharmacology, Leukotriene B4, Leukotriene-A4 hydrolase, Mice, Structure-Activity Relationship, Drug Discovery, Hydrolase, Animals, Humans, Structure–activity relationship, Enzyme Inhibitors, Epoxide Hydrolases, chemistry.chemical_classification, biology, In vitro, Enzyme, Biochemistry, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Ex vivo
-
4
المؤلفون: Gwen Grabowski Krivi, E.Yvonne Pyla, Stevan W. Djuric, Thomas D. Penning, Richard A. Haack, Leslie J Askonas, Stella S. Yu, Marshall L. Michener
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:2517-2522
مصطلحات موضوعية: chemistry.chemical_classification, Leukotriene A4, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Peptide, Biochemistry, Aminopeptidase, Leukotriene-A4 hydrolase, chemistry.chemical_compound, Enzyme, chemistry, Drug Discovery, Hydrolase, Molecular Medicine, Kelatorphan, Molecular Biology
-
5
المؤلفون: Doreen Villani-Price, Suzanne H Kim, Walter G. Smith, Leslie J Askonas, Elizabeth I Harding, Maureen K Highkin, Thomas D. Penning, Alan F. Gasiecki, Nayereh S Ghoreishi-Haack, Nizal S Chandrakumar, E.Yvonne Pyla, Bipin N Desai, James F Kachur, Mark A Russell, Stevan W Djuric, James W. Malecha, James K. Gierse, Julie M Miyashiro
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:1137-1139
مصطلحات موضوعية: Imidazopyridine, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Purine analogue, In Vitro Techniques, Biochemistry, Chemical synthesis, Leukotriene-A4 hydrolase, Mice, Structure-Activity Relationship, Heterocyclic Compounds, Drug Discovery, Animals, Humans, Structure–activity relationship, Enzyme Inhibitors, Purine metabolism, Molecular Biology, Epoxide Hydrolases, biology, Chemistry, Organic Chemistry, Recombinant Proteins, stomatognathic diseases, Purines, Enzyme inhibitor, biology.protein, Molecular Medicine, Indicators and Reagents, Ex vivo
-
6
المؤلفون: Trevor M. Penning, Leslie J. Askonas
المصدر: Biochemistry. 30:11553-11560
مصطلحات موضوعية: 3-Hydroxysteroid Dehydrogenases, Binding Sites, Affinity labeling, biology, Affinity label, Anti-Inflammatory Agents, Non-Steroidal, Indomethacin, Affinity Labels, Pharmacology, Biochemistry, Enzyme Activation, Kinetics, Structure-Activity Relationship, chemistry.chemical_compound, chemistry, Drug Design, biology.protein, Anthranilic acid, Drug Binding Site, Prostaglandin-F synthase, Binding site, Hydroxysteroid dehydrogenase, Prostaglandin H2
-
7
المؤلفون: Leslie J. Askonas, Ronald J. Parry, Angelika Muscate
المصدر: Biochemistry. 30:9988-9997
مصطلحات موضوعية: chemistry.chemical_classification, Protein Denaturation, Adenosine, Binding Sites, biology, Hydrolases, Stereochemistry, Adenosylhomocysteinase, NAD, Biochemistry, Cofactor, Enzyme Activation, Kinetics, Enzyme, chemistry, Affinity chromatography, Enzyme inhibitor, Dideoxyadenosine, Enzyme Stability, Hydrolase, biology.protein, Nucleotide, NAD+ kinase
-
8
المؤلفون: Maureen K Highkin, Leslie J Askonas, Doreen Villani-Price, Chi-Dean Liang, Bipin N Desai, Thomas D. Penning, James F Kachur, Elizabeth I Harding, Nayereh S Ghoreishi-Haack, Mark A Russell, Julie M Miyashiro, Walter G. Smith, E.Yvonne Pyla, Nizal S Chandrakumar, Stevan W Djuric, Suzanne H Kim, James K. Gierse, Alan F. Gasiecki
المصدر: Bioorganicmedicinal chemistry letters. 12(23)
مصطلحات موضوعية: Pyrrolidines, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Biochemistry, Chemical synthesis, Pyrrolidine, Leukotriene-A4 hydrolase, chemistry.chemical_compound, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, Piperidines, In vivo, Drug Discovery, Hydrolase, Structure–activity relationship, Animals, Humans, Enzyme Inhibitors, Molecular Biology, Epoxide Hydrolases, biology, Chemistry, Organic Chemistry, stomatognathic diseases, Enzyme inhibitor, biology.protein, beta-Alanine, Molecular Medicine, Ex vivo
-
9
المؤلفون: James F. Kachur, Leslie J. Askonas, Doreen Villani-Price, Nayereh Ghoreishi-Haack, Suzanne Won-Kim, Chi-Dean D. Liang, Mark A. Russell, Walter G. Smith
المصدر: The Journal of pharmacology and experimental therapeutics. 300(2)
مصطلحات موضوعية: Pharmacology, Epoxide Hydrolases, Administration, Topical, Administration, Oral, Dermatitis, In Vitro Techniques, Leukotriene A4, Rats, Mice, Arthus Reaction, beta-Alanine, Molecular Medicine, Animals, Edema, Eicosanoids, Hydroxyurea, Leukotriene Antagonists, Lipoxygenase Inhibitors, Enzyme Inhibitors, Peritoneum, Skin
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::85dd328be3aae29c01487cfa97414149
https://pubmed.ncbi.nlm.nih.gov/11805220 -
10
المؤلفون: Trevor M. Penning, Leslie J. Askonas, Mark S. Tang
المصدر: Advances in Experimental Medicine and Biology ISBN: 9781461374305
مصطلحات موضوعية: biology, Mefenamic acid, ATP synthase, Affinity label, Cleavage (embryo), chemistry.chemical_compound, Biochemistry, chemistry, biology.protein, medicine, Anthranilic acid, Arachidonic acid, Cyclooxygenase, Prostaglandin H2, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::3025944b235a1e636e6155d7cfc9da6e
https://doi.org/10.1007/978-1-4615-5325-0_11