-
1
المؤلفون: Karren D. Beattie, Topul Rali, Troy E. Messick, Frederick Keeney, Lily D. Lu, Rohan A. Davis, Emery T. Register, Joseph M. Salvino, Luis J. Montaner, Xiangyang Zhou, Ian Tietjen, Joel Cassel, Pablo Tebas, Hildegund C.J. Ertl
المصدر: Antimicrobial Agents and Chemotherapy
مصطلحات موضوعية: natural products, coronavirus, Resveratrol, Antiviral Agents, 01 natural sciences, stilbenoids, 03 medical and health sciences, chemistry.chemical_compound, Phenols, Viral entry, Stilbenes, Humans, Pharmacology (medical), Receptor, Cytotoxicity, Pandemics, 030304 developmental biology, Cytopathic effect, Pharmacology, 0303 health sciences, SARS-CoV-2, 010405 organic chemistry, Chemistry, Ligand binding assay, COVID-19, Ligand (biochemistry), Virology, In vitro, 3. Good health, 0104 chemical sciences, Infectious Diseases, Spike Glycoprotein, Coronavirus, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b6ab9ced861bf84f6fc1c81f25f01192
https://doi.org/10.1128/aac.00772-21 -
2
المؤلفون: Karren D. Beattie, Frederick Keeney, Rohan A. Davis, Luis J. Montaner, Emery T. Register, Joel Cassel, Xiangyang Zhou, Hildegund C.J. Ertl, Lily D. Lu, Troy E. Messick, Topul Rali, Ian Tietjen, Joseph M. Salvino
مصطلحات موضوعية: Infectivity, chemistry.chemical_compound, chemistry, Viral entry, Ligand binding assay, Resveratrol, Biology, Receptor, Ligand (biochemistry), Virology, In vitro, Cytopathic effect
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::313f69e8af68ad533f529397176b915b
https://doi.org/10.1101/2021.04.29.442010 -
3
المؤلفون: William Hockeimer, Kristine L. Stump, Matthew M. Seavey, Bruce Ruggeri, Nate H. Wallace, Teresa M. O'Kane, Lily D. Lu, Pawel Dobrzanski
المصدر: Molecular Cancer Therapeutics. 11:984-993
مصطلحات موضوعية: Cancer Research, Pyridines, Colorectal cancer, Angiogenesis, Mouse model of colorectal and intestinal cancer, medicine.disease_cause, Proinflammatory cytokine, Mice, Cell Line, Tumor, medicine, Animals, Humans, Phosphorylation, Protein Kinase Inhibitors, STAT5, Mice, Inbred BALB C, biology, Cancer, Interleukin, Janus Kinase 2, Triazoles, Colitis, medicine.disease, Disease Models, Animal, Oncology, Immunology, Cancer research, biology.protein, Female, Colorectal Neoplasms, Carcinogenesis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f11cea5144fe26bcfd3d18f611dea74d
https://doi.org/10.1158/1535-7163.mct-11-0951 -
4
المؤلفون: Thomas J. Connors, Jie Qian, Zeck Huang, Joanne R. Mathiasen, Edward R. Bacon, Thelma S. Angeles, Mark J. Huffman, Emir Duzic, Joseph M. Salvino, Beth Ann McKenna, Hervé Schaffhauser, Robert J. McHugh, Lily D. Lu, George C. Morton, Beverly P. Holskin, Karla Kopec, Amy DiCamillo, Gerard C. Rosse, Chrysanthe Spais, Rabindranath Tripathy, Lisa D. Aimone
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:1421-1426
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Stereoisomerism, Biochemistry, Sulfone, chemistry.chemical_compound, In vivo, Drug Discovery, 5-HT6 receptor, Molecular Medicine, Pharmacophore, Receptor, Molecular Biology, 5-HT receptor
-
5
المؤلفون: Beverly P. Holskin, Karla Kopec, Joanne R. Mathiasen, Amy DiCamillo, Babu G. Sundar, Thomas J. Connors, Emir Duzic, Edward R. Bacon, Gerard C. Rosse, Chrysanthe Spais, Thomas R. Bailey, Beth Ann McKenna, Rebecca A. Brown, Jie Qian, Derek Dunn, Mark J. Huffman, Joseph M. Salvino, Huang Zeqi, Lisa D. Aimone, Hervé Schaffhauser, Deborah Galinis, Thelma S. Angeles, Lily D. Lu, George C. Morton
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:120-123
مصطلحات موضوعية: biology, Organic Chemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Pharmacology, Biochemistry, Social recognition, chemistry.chemical_compound, chemistry, Drug Discovery, biology.protein, 5-HT6 receptor, Molecular Medicine, Structure–activity relationship, Serotonin Antagonists, Penetrant (biochemical), Receptor, Molecular Biology, 5-HT receptor
-
6
المؤلفون: Matthew M. Seavey, Kristine L. Stump, Lily D. Lu, Nate H. Wallace, Bruce Ruggeri
المصدر: International Immunopharmacology. 12:257-270
مصطلحات موضوعية: Threonine, Proteasome Endopeptidase Complex, medicine.medical_specialty, Anti-nuclear antibody, Immunology, Lupus nephritis, Kidney, Mice, immune system diseases, Internal medicine, medicine, Animals, Lupus Erythematosus, Systemic, Immunology and Allergy, skin and connective tissue diseases, Pharmacology, Systemic lupus erythematosus, Proteinuria, Bortezomib, business.industry, Drug Administration Routes, Glomerulonephritis, medicine.disease, Boronic Acids, Lupus Nephritis, Disease Models, Animal, Endocrinology, Tolerability, Antibodies, Antinuclear, Proteasome inhibitor, Cytokines, Female, medicine.symptom, business, Proteasome Inhibitors, Spleen, medicine.drug
-
7
المؤلفون: Rabindranath, Tripathy, Robert J, McHugh, Edward R, Bacon, Joseph M, Salvino, George C, Morton, Lisa D, Aimone, Zeck, Huang, Joanne R, Mathiasen, Amy, DiCamillo, Mark J, Huffman, Beth A, McKenna, Karla, Kopec, Lily D, Lu, Jie, Qian, Thelma S, Angeles, Thomas, Connors, Chrysanthe, Spais, Beverly, Holskin, Emir, Duzic, Hervé, Schaffhauser, Gerard C, Rossé
المصدر: Bioorganicmedicinal chemistry letters. 22(3)
مصطلحات موضوعية: Molecular Structure, Brain, Stereoisomerism, Rats, Inhibitory Concentration 50, Mice, Dogs, Receptors, Serotonin, Microsomes, Liver, Animals, Humans, Serotonin Antagonists, Sulfones, Heterocyclic Compounds, 3-Ring
-
8
المؤلفون: Babu G, Sundar, Thomas R, Bailey, Derek D, Dunn, Edward R, Bacon, Joseph M, Salvino, George C, Morton, Lisa D, Aimone, Huang, Zeqi, Joanne R, Mathiasen, Amy, Dicamillo, Mark J, Huffman, Beth A, McKenna, Karla, Kopec, Lily D, Lu, Rebecca, Brown, Jie, Qian, Thelma, Angeles, Thomas, Connors, Chrysanthe, Spais, Beverly, Holskin, Deborah, Galinis, Emir, Duzic, Herve, Schaffhauser, Gerard C, Rosse
المصدر: Bioorganicmedicinal chemistry letters. 22(1)
مصطلحات موضوعية: ERG1 Potassium Channel, Brain, Ether-A-Go-Go Potassium Channels, Rats, Inhibitory Concentration 50, Kinetics, Structure-Activity Relationship, Memory, Short-Term, Models, Chemical, Piperidines, Receptors, Serotonin, Schizophrenia, Animals, Humans, Serotonin Antagonists, Benzofurans
-
9
المؤلفون: Kristine L. Stump, Matthew M. Seavey, Lily D. Lu
المصدر: Current Protocols in Pharmacology
مصطلحات موضوعية: Autoimmune disease, Systemic lupus erythematosus, Lupus erythematosus, Drug discovery, business.industry, General Medicine, medicine.disease, Disease Models, Animal, New chemical entity, Immunology, Drug Discovery, medicine, Animals, Humans, Lupus Erythematosus, Systemic, skin and connective tissue diseases, business, Organ system, Ex vivo, Immunosuppressive Agents
-
10
المؤلفون: Kristine L. Stump, Benjamin J. Dugan, Lily D. Lu, Matthew M. Seavey, Jennifer L. Mason, Thelma S. Angeles, Diane E. Gingrich, Cynthia Serdikoff, Mark A. Ator, Mark S. Albom, Pawel Dobrzanski, Bruce D. Dorsey, Nate H. Wallace, Bruce Ruggeri
المصدر: Journal of immunology (Baltimore, Md. : 1950). 187(7)
مصطلحات موضوعية: Mice, Inbred MRL lpr, Cyclophosphamide, Pyridines, medicine.medical_treatment, Immunology, Plasma Cells, Lupus nephritis, Administration, Oral, Spleen, Autoimmunity, Enzyme-Linked Immunosorbent Assay, Cell Separation, Proinflammatory cytokine, Mice, Immune system, immune system diseases, Immunology and Allergy, Medicine, Animals, Enzyme Inhibitors, skin and connective tissue diseases, Dexamethasone, biology, business.industry, Janus Kinase 2, Triazoles, medicine.disease, Flow Cytometry, Lupus Nephritis, Disease Models, Animal, Cytokine, medicine.anatomical_structure, Antibodies, Antinuclear, biology.protein, Cytokines, Female, Antibody, business, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e3a3b8bd6b9c256b884ac8efb0f4a3f2
https://pubmed.ncbi.nlm.nih.gov/21880982