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المؤلفون: Erika Rehnström, Thomas Lundböck, Anna Novén, Jan Holmgren, Linda Fredlund, Johan Wernevik, Fredrik Bergström, Dan Addison, Johan Hulthe, Per-Erik Strömstedt
المصدر: Assay and Drug Development Technologies
مصطلحات موضوعية: Computer science, Computational biology, 030226 pharmacology & pharmacy, Mass Spectrometry, Automation, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, assay panels, Drug Discovery, Animals, Humans, Profiling (information science), Chromatography, High Pressure Liquid, 030304 developmental biology, 0303 health sciences, Human liver, business.industry, Original Articles, Metabolic stability, Rats, Workflow, Pharmaceutical Preparations, Drug development, Hepatocytes, Microsomes, Liver, Molecular Medicine, profiling, business, Drug metabolism, DMPK
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a14e880c484c3f3b630ddc5a788747f0
https://doi.org/10.1089/adt.2020.970 -
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المؤلفون: Christian Tyrchan, Anna-Pia Palmgren, Hui-Fang Amy Chang, Yunhua Chen, Victoria Ullah, Karin Björhall, Annika Westin Eriksson, Rebecca Fransson, Mickael Mogemark, Tiiu Wennberg, Shuchun Zhao, Bold Peter, Linda Fredlund, Matthew Thomas, Eva Lamm Bergström, Nils Pemberton, Ulf Börjesson, Reed W. Smith, Mikael Brűlls, Johan Carlsson, Britt-Marie Fihn, Linda Öster, Mio Rodrigo Blomqvist, Hongbin Ge, Antonios Nikitidis, Wenzhen Yang, Anders Eriksson, Haijuan Huang, Sarah Lever, Perry Matthew, Kostas Karabelas, Helena Lindmark, Jens Petersen
المصدر: Journal of medicinal chemistry. 64(12)
مصطلحات موضوعية: Male, Class I Phosphatidylinositol 3-Kinases, Ovalbumin, High selectivity, Pharmacology, Crystallography, X-Ray, 01 natural sciences, 03 medical and health sciences, Phosphatidylinositol 3-Kinases, Structure-Activity Relationship, Rats, Inbred BN, Drug Discovery, medicine, Asthmatic patient, Potency, Structure–activity relationship, Animals, Class Ib Phosphatidylinositol 3-Kinase, Humans, Short duration, Protein Kinase Inhibitors, 030304 developmental biology, Asthma, 0303 health sciences, Sulfonamides, biology, Inhalation, Molecular Structure, Chemistry, medicine.disease, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Thiazoles, biology.protein, Leukocytes, Mononuclear, Molecular Medicine, Protein Binding
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المؤلفون: Christian Tyrchan, Neil S. Holden, Nils Pemberton, Anders Eriksson, Ina Terstiege, Yunhua Chen, Hai'e Hao, Kostas Karabelas, Karin Björhall, Tor Svensson, Linda Fredlund, Wenzhen Yang, Jens Petersen, Shuchun Zhao, Perry Matthew, Johan Carlsson, Helena Lindmark, Sandra Rodrigo Blomqvist, Britta Bonn, Feifei Liu, Reed W. Smith, Linda Öster
المصدر: Journal of medicinal chemistry. 60(12)
مصطلحات موضوعية: 0301 basic medicine, Cell, Drug Evaluation, Preclinical, Biological Availability, Mice, Transgenic, Chemistry Techniques, Synthetic, Pharmacology, Permeability, 03 medical and health sciences, Structure-Activity Relationship, In vivo, B200 Pharmacology, Toxicology and Pharmacy, Drug Discovery, Administration, Inhalation, medicine, Structure–activity relationship, Potency, Animals, Enzyme Inhibitors, B100 Anatomy, Physiology and Pathology, Cell potency, Phosphoinositide-3 Kinase Inhibitors, Inhalation, Chemistry, Kinase, Rats, Isoenzymes, Thiazoles, 030104 developmental biology, medicine.anatomical_structure, Solubility, Drug Design, Lipophilicity, Molecular Medicine, Half-Life
وصف الملف: application/pdf
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المؤلفون: Susanne Winiwarter, Linda Fredlund, Constanze Hilgendorf
المصدر: Molecular pharmaceutics. 14(5)
مصطلحات موضوعية: 0301 basic medicine, Membrane permeability, In silico, Pharmaceutical Science, Biological Transport, Active, 030226 pharmacology & pharmacy, Intestinal absorption, 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, ATP Binding Cassette Transporter, Subfamily G, Member 2, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, Chemistry, Transporter, In vitro, Multidrug Resistance-Associated Protein 2, Permeability (earth sciences), 030104 developmental biology, Biochemistry, Intestinal Absorption, Caco-2, Drug Design, Molecular Medicine, Efflux, Caco-2 Cells, Multidrug Resistance-Associated Proteins
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المؤلفون: Johan Wernevik, Lars Carlsson, Linda Fredlund, Ioana Oprisiu, Susanne Winiwarter, Ernst Ahlberg, Barry Jones, Claus Bendtsen, Tobias Noeske, Per-Erik Strömstedt
المصدر: Toxicology Letters. 280:S285
مصطلحات موضوعية: Property (philosophy), Computer science, In silico, General Medicine, Computational biology, Toxicology, In vitro