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المؤلفون: Sebastien Dropsit, Pieter F. W. Stouten, Linda Tomaskovic, Thierry Christophe, Ellen van der Aar, Maarten Gees, Luc Nelles, Mia Jans, Monica Borgonovi, Evelyne M. Quinton, Katja Conrath, Jan Van Der Schueren, Caroline Joannesse, Hans Kelgtermans, Martin James Inglis Andrews, Sebastien Laurent Xavier Martina, Oscar Mammoliti, Ann De Blieck, Steven Emiel Van Der Plas, Tom De Munck
المصدر: Journal of Medicinal Chemistry. 61:1425-1435
مصطلحات موضوعية: 0301 basic medicine, congenital, hereditary, and neonatal diseases and abnormalities, Mutant, Pharmacology, medicine.disease_cause, Cystic fibrosis, Ivacaftor, 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, medicine, Structure–activity relationship, Mutation, biology, Chemistry, Drug discovery, respiratory system, Potentiator, medicine.disease, digestive system diseases, Cystic fibrosis transmembrane conductance regulator, respiratory tract diseases, 030104 developmental biology, 030220 oncology & carcinogenesis, biology.protein, Molecular Medicine, medicine.drug
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المؤلفون: Donatella Verbanac, Mihaela Perić, Mario Matijašić, Andrea Fajdetić, Linda Tomaskovic, Hana Čipčić Paljetak, Mirjana Bukvić
المصدر: Current Topics in Medicinal Chemistry. 17:919-940
مصطلحات موضوعية: 0301 basic medicine, medicine.drug_class, Antibiotics, Azalide, Biology, Pharmacology, Anti-inflammatory, Antimalarials, 03 medical and health sciences, Polyketide, In vivo, Chloroquine, Drug Discovery, medicine, Animals, Humans, Inflammation, Bacteria, macrolide hybrid, azalide, antibacterial, antimalarial, anti-inflammatory, quinolone, quinoline, corticosteroid, Anti-Inflammatory Agents, Non-Steroidal, General Medicine, Quinolone, Anti-Bacterial Agents, Malaria, 030104 developmental biology, Macrolides, Pharmacophore, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c36d459192d76e02e59d7b870b41e46a
https://doi.org/10.2174/1568026616666160927160036 -
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المؤلفون: Dijana Pesic, Ivaylo Jivkov Elenkov, Antun Hutinec, Linda Tomaskovic, Sanja Koštrun, Mirjana Bukvić, Sulejman Alihodžić, Dinko Žiher, Gordon Saxty
مصطلحات موضوعية: 010405 organic chemistry, Drug discovery, Political science, Patent literature, 010402 general chemistry, 01 natural sciences, Data science, 0104 chemical sciences
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::0773aeccbb559a31abb85103d691d875
https://doi.org/10.1016/bs.pmch.2018.01.002 -
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المؤلفون: Steven E, Van der Plas, Hans, Kelgtermans, Tom, De Munck, Sébastien L X, Martina, Sébastien, Dropsit, Evelyne, Quinton, Ann, De Blieck, Caroline, Joannesse, Linda, Tomaskovic, Mia, Jans, Thierry, Christophe, Ellen, van der Aar, Monica, Borgonovi, Luc, Nelles, Maarten, Gees, Pieter, Stouten, Jan, Van Der Schueren, Oscar, Mammoliti, Katja, Conrath, Martin, Andrews
المصدر: Journal of medicinal chemistry. 61(4)
مصطلحات موضوعية: Structure-Activity Relationship, Cystic Fibrosis, Drug Discovery, Mutation, Animals, Cystic Fibrosis Transmembrane Conductance Regulator, Humans, Pyrazoles, Mutant Proteins, Quinolones, Aminophenols, Chloride Channel Agonists, Rats
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المصدر: Structural Chemistry. 20:73-80
مصطلحات موضوعية: Stereochemistry, Hydrogen bond, Chemistry, Intermolecular force, Stacking, 5-dihydroxy-2-nitrobenzoic acid, 3, 5-dihydroxy-4-nitrobenzoic acid, alpha-resorcylic acid, X-ray structure, aromatic nitration, Crystal structure, Condensed Matter Physics, law.invention, Crystallography, chemistry.chemical_compound, law, Intramolecular force, Nitration, Molecule, Physical and Theoretical Chemistry, Crystallization
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المؤلفون: Jasna Padovan, Linda Tomaskovic, Stribor Markovic, Milan Mesic, Hana Čipčić Paljetak, Mladen Mercep, Ines Glojnarić, Mihailo Banjanac, Barbara Stanić, Jovica Ralić, Vesna Munić, Oresta Makaruha Stegić, Marijana Komac, Vesna Eraković Haber, Boska Hrvacic
المساهمون: University of Zurich, Tomašković, Linda
مصطلحات موضوعية: Male, 1303 Biochemistry, Phagocyte, medicine.drug_class, medicine.medical_treatment, Clinical Biochemistry, Anti-Inflammatory Agents, Carboxylic Acids, 3003 Pharmaceutical Science, Pharmaceutical Science, 610 Medicine & health, Pharmacology, 1308 Clinical Biochemistry, Biochemistry, Anti-inflammatory, Steroid, Cell Line, Mice, Immune system, In vivo, 10183 Swiss Institute of Allergy and Asthma Research, Rats, Inbred BN, Drug Discovery, medicine, 1312 Molecular Biology, Animals, Molecular Biology, Glucocorticoids, Mice, Inbred BALB C, biology, Chemistry, 3002 Drug Discovery, Organic Chemistry, In vitro, Asthma, Rats, Ovalbumin, medicine.anatomical_structure, Drug Design, 1313 Molecular Medicine, concept, anti-inflammatory, glucocorticoid, macrolides, biology.protein, Molecular Medicine, Steroids, Macrolides, Glucocorticoid, medicine.drug, 1605 Organic Chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ef738a49ddc32a931c0b944f69099b06
https://www.zora.uzh.ch/id/eprint/76109/ -
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المؤلفون: Sulejman Alihodžić, Denis Polančec, Marjorie A. Smith, Ivica Malnar, Vesna Eraković Haber, Michael Lee, Krunoslav Nujić, Daniela Belamarić, Linda Tomaskovic, Klaus Schneider
المصدر: European journal of pharmacology. 677(1-3)
مصطلحات موضوعية: Proteomics, medicine.drug_class, Valosin-containing protein, Anti-Inflammatory Agents, Cell Cycle Proteins, Biology, Azithromycin, Macrolide Antibiotics, Cell Line, Mice, Affinity chromatography, In vivo, Valosin Containing Protein, Clarithromycin, medicine, Gene silencing, Animals, Humans, Gene Silencing, Pharmacology, Adenosine Triphosphatases, Reproducibility of Results, In vitro, Anti-Bacterial Agents, macrolide, chemical proteomics, target identification, valosin containing protein, inflammation, Biochemistry, Cell culture, Drug Design, biology.protein, Protein Binding